Issue 13, 2012
From the journal:

Organic & Biomolecular Chemistry

Gold catalysis on immobilized substrates: a heteroannulation approach to the solid-supported synthesis of indoles†

Agustina La-Venia,a   Sebastián A. Testero,a   Mirta P. Mischne*a  and  Ernesto G. Mata*a  

* Corresponding authors

a Instituto de Química Rosario (CONICET – UNR), Facultad de Ciencias Bioquímicas y Farmacéuticas, Universidad Nacional de Rosario, Suipacha 531, 2000 – Rosario, Argentina
E-mail: mischne@iquir-conicet.gov.ar, mata@iquir-conicet.gov.ar
Fax: +54-341-4370477
Tel: +54-341-4370477

Abstract

A gold-catalyzed cyclization of immobilized 2-alkynylanilines was developed as the key step in the synthetic sequence for the preparation of 2-substituted indoles. These results demonstrate the potential of the unexplored combination of gold catalysis and solid-phase organic synthesis.

Graphical abstract: Gold catalysis on immobilized substrates: a heteroannulation approach to the solid-supported synthesis of indoles

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Article information

DOI
https://doi.org/10.1039/C2OB06881H
Article type
Communication
Submitted
08 Nov 2011
Accepted
18 Jan 2012
First published
19 Jan 2012

Org. Biomol. Chem., 2012,10, 2514-2517

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Gold catalysis on immobilized substrates: a heteroannulation approach to the solid-supported synthesis of indoles

A. La-Venia, S. A. Testero, M. P. Mischne and E. G. Mata, Org. Biomol. Chem., 2012, 10, 2514 DOI: 10.1039/C2OB06881H

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