Issue 53, 2017

Exhaustive Suzuki–Miyaura reactions of polyhalogenated heteroarenes with alkyl boronic pinacol esters

Abstract

A novel Suzuki–Miyaura protocol is described that enables the exhaustive alkylation of polychlorinated pyridines. This method facilitates a formal synthesis of normuscopyridine and the rapid assembly of a dumbbell shaped portion of a [2]rotaxane.

Graphical abstract: Exhaustive Suzuki–Miyaura reactions of polyhalogenated heteroarenes with alkyl boronic pinacol esters

Supplementary files

Article information

Article type
Communication
Submitted
07 Kol 2017
Accepted
28 Kol 2017
First published
03 Ube 2017

Chem. Commun., 2017,53, 7270-7273

Exhaustive Suzuki–Miyaura reactions of polyhalogenated heteroarenes with alkyl boronic pinacol esters

S. Laulhé, J. M. Blackburn and J. L. Roizen, Chem. Commun., 2017, 53, 7270 DOI: 10.1039/C7CC00997F

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