Issue 17, 2005
From the journal:

Organic & Biomolecular Chemistry

A straightforward approach towards thiazoles and endothiopeptides via Ugi reaction†

Uli Kazmaier*a  and  Stefanie Ackermanna  

* Corresponding authors

a Institut für Organische Chemie, Universität des Saarlandes, D-66123 Saarbrücken, Germany
E-mail: u.kazmaier@mx.uni-saarland.de
Fax: +49 681 302 2409
Tel: +49 681 302 2409

Abstract

Endothiopeptides can easily be obtained via Ugi reaction using thio acids as acid components. If isonitriles with an acetal group are applied, the endothiopeptides can directly be converted into thiazoles using TMSCl–NaI under microwave irradiation.

Graphical abstract: A straightforward approach towards thiazoles and endothiopeptides via Ugi reaction

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Article information

DOI
https://doi.org/10.1039/B507028G
Article type
Paper
Submitted
18 May 2005
Accepted
29 Jun 2005
First published
26 Jul 2005

Org. Biomol. Chem., 2005,3, 3184-3187

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A straightforward approach towards thiazoles and endothiopeptides via Ugi reaction

U. Kazmaier and S. Ackermann, Org. Biomol. Chem., 2005, 3, 3184 DOI: 10.1039/B507028G

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