Issue 13, 2016

Copper(ii)-mediated regioselective N-arylation of pyrroles, indoles, pyrazoles and carbazole via dehydrogenative coupling

Abstract

A copper(II)-mediated regioselective N-arylation of azoles has been developed using 8-aminoquinoline amide as a directing group. This reaction shows a broad substrate scope with different azoles such as pyrroles, indoles, pyrazoles and carbazole with good yields.

Graphical abstract: Copper(ii)-mediated regioselective N-arylation of pyrroles, indoles, pyrazoles and carbazole via dehydrogenative coupling

Supplementary files

Article information

Article type
Communication
Submitted
01 Oct 2015
Accepted
07 Jan 2016
First published
07 Jan 2016

Chem. Commun., 2016,52, 2803-2806

Author version available

Copper(II)-mediated regioselective N-arylation of pyrroles, indoles, pyrazoles and carbazole via dehydrogenative coupling

P. Sadhu and T. Punniyamurthy, Chem. Commun., 2016, 52, 2803 DOI: 10.1039/C5CC08206D

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