Rapid preparation of triazolyl substituted NH-heterocyclic kinase inhibitorsvia one-pot Sonogashira coupling–TMS-deprotection–CuAAC sequence†‡
Abstract
The one-pot, three-component
* Corresponding authors
a
Lehrstuhl für Organische Chemie, Institut für Organische Chemie und Makromolekulare Chemie, Heinrich-Heine-Universität Düsseldorf, Universitätsstraße 1, Düsseldorf, Germany
E-mail:
ThomasJJ.Mueller@uni-duesseldorf.de
Fax: ++49 (0)211 8114324
Tel: ++49 (0)211 8112298
b Merck Serono Research & Development, Merck KGaA, Darmstadt, Germany
The one-pot, three-component
E. Merkul, F. Klukas, D. Dorsch, U. Grädler, H. E. Greiner and T. J. J. Müller, Org. Biomol. Chem., 2011, 9, 5129 DOI: 10.1039/C1OB05586K
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