Identification of novel natural inhibitors of Mycobacterium tuberculosis DNA-directed RNA polymerase via extensive computational screening and MMGBSA

Muhammad Bilal Azmi, Muhammad Waqas, Shahid Durran, Palvasha Hussain, Muhammad Yahya Noori, Syed Danish Haseen Ahmed, Gehan Ahmed Othman, Mesaik M. Ahmed, Sobia Ahsan Halim, Ajmal Khan and Ahmed Al-Harrasi

Journal of Molecular Liquids, 2025, 427, 127360
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Nanoenabling MbtI Inhibitors for Next-Generation Tuberculosis Therapy

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J. Med. Chem., 2025, 68, 5312
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Targeted isolation of natural analogs of anti-mycobacterial hit compounds based on the metabolite profiling of a large collection of plant extracts

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Front. Nat. Prod., 2023, 2
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Isolation and Characterization of Anti-Mycobacterial Natural Products from a Petrosia sp. Marine Sponge

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Quinoline heterocyclic containing plant and marine candidates against drug-resistant Mycobacterium tuberculosis: A systematic drug-ability investigation

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European Journal of Medicinal Chemistry, 2022, 232, 114173
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Microbial-based natural products as potential inhibitors targeting DNA gyrase B of Mycobacterium tuberculosis: an in silico study

Tilal Elsaman, Magdi Awadalla Mohamed, Malik Suliman Mohamed, Eyman Mohamed Eltayib and Abualgasim Elgaili Abdalla

Front. Chem., 2025, 13
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Natural products and their analogues acting against Mycobacterium tuberculosis: A recent update

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Alkaloids of Dicranostigma franchetianum (Papaveraceae) and Berberine Derivatives as a New Class of Antimycobacterial Agents

Viriyanata Wijaya, Ondřej Janďourek, Jana Křoustková, Kateřina Hradiská-Breiterová, Jan Korábečný, Kateřina Sobolová, Eliška Kohelová, Anna Hošťálková, Klára Konečná, Marcela Šafratová, Rudolf Vrabec, Jiří Kuneš, Lubomír Opletal, Jakub Chlebek and Lucie Cahlíková

Biomolecules, 2022, 12, 844
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Plant-Derived Antimicrobials and Their Crucial Role in Combating Antimicrobial Resistance

Paola Angelini

Antibiotics, 2024, 13, 746
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Study on the Anti-Mycobacterium marinum Activity of a Series of Marine-Derived 14-Membered Resorcylic Acid Lactone Derivatives

Qian-Qian Jing, Jun-Na Yin, Ya-Jie Cheng, Qun Zhang, Xi-Zhen Cao, Wei-Feng Xu, Chang-Lun Shao and Mei-Yan Wei

Marine Drugs, 2024, 22, 135
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Microbial-derived peptides with anti-mycobacterial potential

Pengchao Zhao, Pu Hou, Zhishen Zhang, Xin Li, Chunshan Quan, Yun Xue, Kun Lei, Jinghua Li, Weina Gao and Fangfang Fu

European Journal of Medicinal Chemistry, 2024, 276, 116687
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Unique Remote Regiocontrol by an N‐Oxide Group in the Synthesis of Isocaulibugulones A, B, C, and D

Joaquim A. M. Castro, Bruno K. Serikava, Fabrício F. Naciuk, Carolina B. P. Ligiéro, Nelson H. Morgon and Paulo C. M. L. Miranda

ChemistrySelect, 2023, 8
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Vitamin K (Menaquinone) from marine Kocuria sp. RAM1: optimization, characterization and potential in vitro biological activities

Rasha A. Metwally, Nermeen A. El-Sersy, Amany El Sikaily, Soraya A. Sabry and Hanan A. Ghozlan

Microb Cell Fact, 2025, 24
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The anti-tubercular callyaerins target the Mycobacterium tuberculosis-specific non-essential membrane protein Rv2113

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Jolkinolide B inhibits mycobacterial growth by down-regulating ribosomal proteins and interfering with protein synthesis

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Bioorganic & Medicinal Chemistry, 2025, 129, 118294
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Revisiting the potential of natural products in antimycobacterial therapy: advances in drug discovery and semisynthetic solutions

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Screening of Microbial Fermentation Products for Anti-M. tuberculosis Activity

Aikebaier Reheman, Di Lu, Yifan Wang, Xi Chen, Gang Cao and Chuanxing Wan

Animals, 2022, 12, 1947
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Safety evaluation and bioassay-guided isolation of antimycobacterial compounds from Morella salicifolia root ethanolic extract

Alphonce Ignace Marealle, Ester Innocent, Kerstin Andrae-Marobela, Michael Qwarse, Francis Machumi, Ramadhani S.O. Nondo, Matthias Heydenreich and Mainen Julius Moshi

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Imaging‐based profiling for elucidation of antibacterial mechanisms of action

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An O-methylflavone from Artemisia afra kills non-replicating hypoxic Mycobacterium tuberculosis

Joshua J. Kellogg, Maria Natalia Alonso, R. Teal Jordan, Junpei Xiao, Juan Hilario Cafiero, Trevor Bush, Xiaoling Chen, Melissa Towler, Pamela Weathers and Scarlet S. Shell

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Multitargeting: An Alternative Approach to Tackle Multidrug Resistance in Tuberculosis

Satakshi Hazra, Risha Hazarika and Sanjukta Patra

CDT, 2023, 24, 751
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Oxidative Cyclization at ortho-Position of Phenol: Improved Total Synthesis of 3-(Phenethylamino)demethyl(oxy)aaptamine

Yuki Nakatani, Risa Kimura, Tomoyo Kimata and Naoyuki Kotoku

Marine Drugs, 2023, 21, 311
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Boosting the antibacterial potency of natural products through nanotechnologies

Min Jiao, Weiwen Kong, Wenjuan Liu, Zirong Dong, Jinlong Yang, Zibo Wei, Xinrui Lu, Yuning Wei and Jie Zhuang

International Journal of Pharmaceutics, 2025, 674, 125437
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Nuclear Magnetic Resonance Fingerprinting and Principal Component Analysis Strategies Lead to Anti-Tuberculosis Natural Product Discovery from Actinomycetes

Jianying Han, Xueting Liu, Lixin Zhang, Ronald J. Quinn and Miaomiao Liu

Antibiotics, 2025, 14, 108
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Identification of Axinellamines A and B as Anti-Tubercular Agents

Emily J. Strong, Lendl Tan, Sasha Hayes, Hayden Whyte, Rohan A. Davis and Nicholas P. West

Marine Drugs, 2024, 22, 298
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