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2,5-Diazabicyclo[2.2.1]heptane in medicinal chemistry: a treasure trove of therapeutic opportunities

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A decennary update on applications of metal nanoparticles (MNPs) in the synthesis of nitrogen- and oxygen-containing heterocyclic scaffolds

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Molecular iodine-catalysed oxidative CO–C(alkyl) bond cleavage of aryl/heteroaryl alkyl ketones: an efficient strategy to access fused polyheterocycles

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Ynones as versatile electrophiles for the divergent synthesis of 4H-chromenes and 1,4-dihydroquinolines

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Rh(iii)-Catalyzed switchable C–H monoalkenylation and dialkenylation of 2-(1H-pyrazol-1-yl)pyridine with alkenes via rollover cyclometalation

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A decade update on the application of β-oxodithioesters in heterocyclic synthesis

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Multi-functionalization of Rh-carbynoids with alcohols/carbamates and α-propargylic-3-indolymethanols

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Design, synthesis, and anti-mycobacterial evaluation of 1,8-naphthyridine-3-carbonitrile analogues

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Iron-catalyzed cascade one-pot reaction between azlactones and O-acetyl oximes to afford 6H-pyrrolo[3,2-d]oxazole and pyrrol-2-one nucleus

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Reductive stability evaluation of 6-azopurine photoswitches for the regulation of CKIα activity and circadian rhythms

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Organic acid catalysed Minisci-type arylation of heterocycles with aryl acyl peroxides

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Transition-metal-free approaches to access N-heterocycles and valuable intermediates from aryldiazonium salts

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Cycloamination strategies for renewable N-heterocycles

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A direct entry to polycyclic quinoxaline derivativesviaI2-DMSO mediated oxidative decarboxylation of α-amino acids and the subsequent Pictet–Spengler cyclization reaction

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Silver/molybdenum-promoted skeletal reconstructive cyclization of N-quinolinyl indoles and anthranils

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Recent advances in metal-free catalysts for the synthesis of N-heterocyclic frameworks focusing on 5- and 6-membered rings: a review

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Nickel-catalyzed borrowing hydrogen annulations: access to diversified N-heterocycles

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Multicomponent reactions as a potent tool for the synthesis of benzodiazepines

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Stereoselective synthesis of 3,3′-spirooxindoles with higher order heterocycles

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Indazolin-3-ylidenes (Indy*): easily accessible, sterically-hindered indazole-derived N-heterocyclic carbenes and their application in gold catalysis

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UV/visible light-promoted external photocatalyst-free transformations: A Decade's Journey of N-heterocycles and their functionalisation

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Biocompatible de novo indolylchalcones as platelet aggregation inhibition and diabetic wound healing agents

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Single-atom molecular editing: transformative advances in carbocyclic and heterocyclic frameworks

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