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Catalytic Asymmetric Mono‐Fluorination of α‐Keto Esters: Synthesis of Optically Active β‐Fluoro‐α‐Hydroxy and β‐Fluoro‐α‐Amino Acid Derivatives

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Angew Chem Int Ed, 2012, 51, 4581
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Alkali Carbonates Improve β,β-Diaryl Serine-Catalyzed Enantioselective α-Fluorination of β-Dicarbonyl Compounds

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New insights on reaction pathway selectivity promoted by crown ether phase-transfer catalysis: Model ab initio calculations of nucleophilic fluorination

Josefredo R. Pliego and Jose M. Riveros

Journal of Molecular Catalysis A: Chemical, 2012, 363-364, 489
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Asymmetric catalysis as a method for the synthesis of chiral organophosphorus compounds

Oleg I. Kolodiazhnyi, Valery P. Kukhar and Anastasy O. Kolodiazhna

Tetrahedron: Asymmetry, 2014, 25, 865
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Cinchona Alkaloid Catalyzed Enantioselective Fluorination of Allyl Silanes, Silyl Enol Ethers, and Oxindoles

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Angewandte Chemie, 2008, 120, 4225
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Convenient Electrophilic Fluorination of Functionalized Aryl and Heteroaryl Magnesium Reagents

Shigeyuki Yamada, Andrei Gavryushin and Paul Knochel

Angewandte Chemie, 2010, 122, 2261
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Selective Fluorination of Multi-Substituted Aldehydes or Ketones Using Amino Catalysts

Satoru Arimitsu

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Review of recent advances in nucleophilic C–F bond-forming reactions at sp3 centers

Jimmy Wu

Tetrahedron Letters, 2014, 55, 4289
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2,2′-Bipyridine-3,3′-dicarboxylic carbohydrate esters and amides. Synthesis and preliminary evaluation as ligands in Cu(II)-catalysed enantioselective electrophilic fluorination

Aurélie Assalit, Thierry Billard, Stéphane Chambert, Bernard R. Langlois, Yves Queneau and Diane Coe

Tetrahedron: Asymmetry, 2009, 20, 593
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Catalytic enantioselective chlorination of cyclic β-keto esters in the presence of chiral Pd(II) complexes

Young Ku Kang, Hee Hun Kim, Kwang Oh Koh and Dae Young Kim

Tetrahedron Letters, 2012, 53, 3811
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Stereocontrolled Approach to Bromofluoroalkenes and Their Use for the Synthesis of Tri- and Tetrasubstituted Fluoroalkenes

Grégory Landelle, Pier Alexandre Champagne, Xavier Barbeau and Jean-François Paquin

Org. Lett., 2009, 11, 681
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Ruthenium‐Catalyzed CC Coupling of Fluorinated Alcohols with Allenes: Dehydrogenation at the Energetic Limit of β‐Hydride Elimination

Brannon Sam, Tom Luong and Michael J. Krische

Angewandte Chemie, 2015, 127, 5555
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N‐Trifluoromethylthiophthalimide: A Stable Electrophilic SCF3‐Reagent and its Application in the Catalytic Asymmetric Trifluoromethylsulfenylation

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Angew Chem Int Ed, 2013, 52, 12856
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Selective Synthesis of Monofluorinated Compounds Applying Amine/HF Reagents

Günter Haufe

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Fluorinated Aromatic Ketones as Nucleophiles in the Asymmetric Organocatalytic Formation of CC and CN Bonds: A Facile Route to the Construction of Fluorinated Quaternary Stereogenic Centers

Yujun Zhao, Yuanhang Pan, Hongjun Liu, Yuanyong Yang, Zhiyong Jiang and Choon‐Hong Tan

Chemistry A European J, 2011, 17, 3571
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Recent Progress in Synthesis of Alkyl Fluorinated Compounds with Multiple Contiguous Stereogenic Centers

Xuemei Yin, Xihong Wang, Lei Song, Junxiong Zhang and Xiaoling Wang

Molecules, 2024, 29, 3677
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Asymmetric Fluorofunctionalizations with Carboxylate‐Based Phase‐Transfer Catalysts

Hiromichi Egami and Yoshitaka Hamashima

The Chemical Record, 2023, 23
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Functionalization of Fluorinated Molecules by Transition-Metal-Mediated C–F Bond Activation To Access Fluorinated Building Blocks

Theresia Ahrens, Johannes Kohlmann, Mike Ahrens and Thomas Braun

Chem. Rev., 2015, 115, 931
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Stereoselective Difluoromethylenation Using Me3SiCF2SPh: Synthesis of Chiral 2,4‐Disubstituted 3,3‐Difluoropyrrolidines

Ya Li and Jinbo Hu

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Enantioselective Fluorination of α-Substituted β-Diketones Using β,β-Diaryl Serines

Samira Poorsadeghi, Katsuki Endo and Satoru Arimitsu

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Olefin Metathesis Reactions with Fluorinated Substrates, Catalysts, and Solvents

Santos Fustero, Antonio Simón-Fuentes, Pablo Barrio and Günter Haufe

Chem. Rev., 2015, 115, 871
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Selection between Diastereomeric Kinetic vs Thermodynamic Carbonyl Binding Modes Enables Enantioselective Iridium-Catalyzed anti-(α-Aryl)allylation of Aqueous Fluoral Hydrate and Difluoroacetaldehyde Ethyl Hemiacetal

James M. Cabrera, Johannes Tauber, Wandi Zhang, Ming Xiang and Michael J. Krische

J. Am. Chem. Soc., 2018, 140, 9392
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Synthesis of novel chiral fluorinating agents, (+)- and (−)-N-fluoro-3-methyl-3-(4-methylphenyl)-2H-benzo[e][1,2]thiazine-1,1,4-triones

Hui Min Sun, Zhao Peng Liu and Long Qian Tang

Chinese Chemical Letters, 2008, 19, 907
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Pinacolatoboron fluoride (pinBF) is an efficient fluoride transfer agent for diastereoselective synthesis of benzylic fluorides

Alexander J. Cresswell, Stephen G. Davies, Aude L.A. Figuccia, Ai M. Fletcher, Dorus Heijnen, James A. Lee, Melloney J. Morris, Alice M.R. Kennett, Paul M. Roberts and James E. Thomson

Tetrahedron Letters, 2015, 56, 3373
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Enantioselective Fluorination of β-Ketoesters Catalyzed by Chiral Sodium Phosphate: Remarkable Enhancement of Reactivity by Simultaneous Utilization of Metal Enolate and Metal Phosphate

Keiji Mori, Ayaka Miyake and Takahiko Akiyama

Chemistry Letters, 2014, 43, 137
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Beyond the Balz–Schiemann Reaction: The Utility of Tetrafluoroborates and Boron Trifluoride as Nucleophilic Fluoride Sources

Alexander J. Cresswell, Stephen G. Davies, Paul M. Roberts and James E. Thomson

Chem. Rev., 2015, 115, 566
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