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Covalent drugs based on small molecules and peptides for disease theranostics

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Solid Phase Synthesis of Fluorosulfate Containing Macrocycles for Chemoproteomic Workflows

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SuFEx Chemistry Enables Covalent Assembly of a 280-kDa 18-Subunit Pore-Forming Complex

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Covalent Proteomimetic Inhibitor of the Bacterial FtsQB Divisome Complex

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Stretching Peptides to Generate Small Molecule β-Strand Mimics

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Recent developments in catalysis and inhibition of the Jumonji histone demethylases

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Atypical histone targets of PHD fingers

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Trimethyllysine Reader Proteins Exhibit Widespread Charge-Agnostic Binding via Different Mechanisms to Cationic and Neutral Ligands

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The Promise of Epigenetics Research in the Treatment of Appendiceal Neoplasms

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Recent advances in the development of therapeutic peptides

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HTS Identifies NUP98-KDM5A-PHD3 Domain Ligands with Novel Scaffolds

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Recent advances in the development of peptide-based inhibitors targeting epigenetic readers of histone lysine acetylation and methylation marks

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An Intrinsically Disordered Region of Histone Demethylase KDM5A Activates Catalysis Through Interactions With the Nucleosomal Acidic Patch and DNA

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Intrastrand Peptide Staples That Promote β-Sheet Folding, Self-Assembly, and Amyloid Seeding

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Application of a MALDI mass spectrometry assay to identify covalent fragments targeting the methyl-lysine reader protein MPP8

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Advances in sulfur fluoride exchange for chemical biology

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