Indazole – an emerging privileged scaffold: synthesis and its biological significance

Anuradha Singampalli, Pardeep Kumar, Rani Bandela, Sri Mounika Bellapukonda, Srinivas Nanduri and Venkata Madhavi Yaddanapudi

RSC Med. Chem., 2025, 16, 5196
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An efficient and simple approach for synthesizing indazole compounds using palladium-catalyzed Suzuki–Miyaura cross-coupling

Bandaru Gopi and Vijayaparthasarathi Vijayakumar

RSC Adv., 2024, 14, 26494
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Synthesis molecular docking and DFT studies on novel indazole derivatives

Bandaru Gopi and Vijayaparthasarathi Vijayakumar

RSC Adv., 2024, 14, 13218
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Importance of Indazole against Neurological Disorders

Dilipkumar Pal and Pooja Sahu

CTMC, 2022, 22, 1136
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Unveiling the hidden harms: a review on the deeper exploration of side effects of oncotherapy

Amrutashree Hota and Badal Kumar Mandal

Med Oncol, 2025, 43
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Synthesis of 3‐(Phenylcarbonyl)‐1H‐indazole Derivatives through Intramolecular Cyclization under Mild Conditions

Sota Kuroyanagi, Shumpei Kikuchi, Shunsuke Sumikoshi, Mizuho Uwano, Takayuki Chiba, Ryohei Yamakado and Shuji Okada

Asian J Org Chem, 2022, 11
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Study of the Addition Mechanism of 1H-Indazole and Its 4-, 5-, 6-, and 7-Nitro Derivatives to Formaldehyde in Aqueous Hydrochloric Acid Solutions

Ibon Alkorta, Rosa M. Claramunt, José Elguero, Enrique Gutiérrez-Puebla, M. Ángeles Monge, Felipe Reviriego and Christian Roussel

J. Org. Chem., 2022, 87, 5866
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Indazole, a privileged scaffold: Synthetic strategies, biological potential, and future prospects

Sanjay Kumar, Ajay Kumar, Shashi Kiran Misra, Ashish Tiwari, Shweta Singh Verma and Amrita Singh

Letters in Drug Design & Discovery, 2025, 22, 100249
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Expanding Therapeutic Horizons with Indazole-Based Compounds: A Review of Anticancer, Antimicrobial, and Neuroprotective Applications

Pooja Dinkar Bhane and Sarita Suryabhan Pawar

MC, 2026, 22, 30
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Recent Advances in Indazole‐Derived Heterocycles: Synthetic Strategies, Functionalization, and Therapeutic Potential

Uday V. Bhat, Glanish Jude Martis, Dinesh Chikkanna, Santosh L. Gaonkar and Munmun Bardhan

Journal of Chemistry, 2025, 2025
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Discovery of Tropomyosin Receptor Kinase Inhibitors as New Generation Anticancer Agents: A Review

Ishan Panchal, Rati Kailash Prasad Tripathi, Kinjal Parmar and Mange Ram Yadav

CTMC, 2024, 24, 3
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Microwave-Assisted Facile Synthesis of 1,2-Benzisoxazoles, Isoxazoloquinolines, and Isothiazoloquinolines in [BMIM(SO2Cl)][OTs] Ionic Liquid as a Recyclable System

I. Jamadar, R. B. Manami, S. Kurahatti, A. Anchi, V. Jadhav, R. G. Kalkhambkar, M. Kurkuri, M. S. Refat and A. M. Alsuhaibani

Russ J Gen Chem, 2025, 95, 393
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Design, Synthesis, and Evaluation of EA-Sulfonamides and Indazole-Sulfonamides as Promising Anticancer Agents: Molecular Docking, ADME Prediction, and Molecular Dynamics Simulations

Nassima Saghdani, Nabil El Brahmi, Abdelmoula El Abbouchi, Rachid Haloui, Souad Elkhattabi, Gérald Guillaumet and Saïd El Kazzouli

Chemistry, 2024, 6, 1396
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Synthesis, in silico Biological Profile and MMP-9 Inhibitory Activity of Some Isonicotinic Acid Hydrazide Incorporated Novel Indazoles

Rajasekhar Komarla Kumarachari, Mayandigari Guruvareddy, Aithepalli Thanuja, Agraharam Shresta, Gilla Shalini, Kalikiri Sindhu and Jampana Bhargavi

Asian J. Chem., 2023, 35, 1264
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A comprehensive review on the indazole based derivatives as targeted anticancer agents

Sachin Puri, Siddhi Sawant and Kapil Juvale

Journal of Molecular Structure, 2023, 1284, 135327
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1‐Benzyl‐1H‐indazol‐3‐ol Copper(II) Derivatives as Anticancer Agents: In‐vitro Interaction with DNA/BSA, DFT, Molecular Docking and Cytotoxicity on MCF7 Cells

Shivabasayya V Salimath and Madhvesh Pathak

ChemistrySelect, 2024, 9
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A review on synthetic strategy, molecular pharmacology of indazole derivatives, and their future perspective

Suvadeep Mal, Udita Malik, Monalisa Mahapatra, Abhishek Mishra, Dilipkumar Pal and Sudhir K. Paidesetty

Drug Development Research, 2022, 83, 1469
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Microwave‐Assisted Rapid and Efficient Synthesis of Novel Indazole‐Based 1,3,4‐Oxadiazole Derivatives with Molecular Docking, ADME, and DFT Studies

Bandaru Gopi and Vijayaparthasarathi Vijayakumar

Asian J Org Chem, 2025, 14
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A comprehensive review on: Organic benzo-fused five-membered N-heterocyclic molecules in mimicry of cancer cell lines and importance of iso-steric replacement

Parasuraman R, Vardhineedi Shirisha, Ravichandra Vandal and Anand KumarTengli

Journal of Molecular Structure, 2026, 1371, 146552
DOI: 10.1016/j.molstruc.2026.146552

Synthesis, anticancer activity and molecular modeling study of novel substituted triazole linked tetrafluoronaphthalene hybrid derivatives

Musa Erdoğan and Ferah Comert Onder

Journal of Biomolecular Structure and Dynamics, 2024, 42, 9767
DOI: 10.1080/07391102.2023.2252914