Rhodium(II)-catalyzed intramolecular annulation of 1-sulfonyl-1,2,3-triazoles with indoles: facile synthesis of functionalized tetrahydro-β-carbolines

Hai Shang; Yu Tian; Jun Luo; Lingyu Li; Yefeng Tang; Zhongmei Zou

doi:10.1039/C6RA02923J

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Rhodium(ii)-catalyzed intramolecular annulation of 1-sulfonyl-1,2,3-triazoles with indoles: facile synthesis of functionalized tetrahydro-β-carbolines†

Hai Shang,^a Yu Tian,^a Jun Luo,^a Lingyu Li,^a Yefeng Tang*^b and Zhongmei Zou*^a

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* Corresponding authors

^a Institute of Medicinal Plant Development, Chinese Academy of Medical Sciences and Peking Union Medical College, Beijing 100193, P. R. China
E-mail: zmzou@implad.ac.cn

^b Comprehensive AIDS Research Center, Department of Pharmacology & Pharmaceutical Sciences, School of Medicine, Tsinghua University, Beijing 100084, China

Abstract

A novel rhodium(II)-catalyzed intramolecular annulation of 1-sulfonyl-1,2,3-triazoles with indoles has been developed, which enables the facile synthesis of various 4-functionalized tetrahydro-β-carbolines as well as relevant scaffolds from readily available starting materials.

This article is part of the themed collection: Elegant Synthetic Routes to Indole Derivatives

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Article information

DOI: https://doi.org/10.1039/C6RA02923J
Article type: Communication
Submitted: 01 Kol 2016
Accepted: 15 Ube 2016
First published: 17 Ube 2016

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RSC Adv., 2016,6, 30835-30839

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Rhodium(II)-catalyzed intramolecular annulation of 1-sulfonyl-1,2,3-triazoles with indoles: facile synthesis of functionalized tetrahydro-β-carbolines

H. Shang, Y. Tian, J. Luo, L. Li, Y. Tang and Z. Zou, RSC Adv., 2016, 6, 30835 DOI: 10.1039/C6RA02923J

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Rhodium(ii)-catalyzed intramolecular annulation of 1-sulfonyl-1,2,3-triazoles with indoles: facile synthesis of functionalized tetrahydro-β-carbolines†

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Rhodium(II)-catalyzed intramolecular annulation of 1-sulfonyl-1,2,3-triazoles with indoles: facile synthesis of functionalized tetrahydro-β-carbolines

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