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Dihydrobenzothiazole coupled N‐piperazinyl acetamides as antimicrobial agents: Design, synthesis, biological evaluation and molecular docking studies

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The Condition of Contemporary Murals in Sun-Exposed Urban Environments: A Model Study Based on Spray-Painted Mock-Ups and Simulated Light Ageing

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Design, synthesis and antibacterial evaluation of piperazine urea–pyrazole-pyrimidine hybrids: in-vitro and in-silico studies

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Piperazinyl-N-aryl acetamides and 1,3,4-thiadiazole Hybrids as Potential DprE1 Inhibitors: Design, Synthesis and Biological Evaluation as antitubercular agents

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Development of Piperazine- and Oxazine-Linked Pyrimidines as p65 Subunit Binders of NF–κB in Human Breast Cancer Cells

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Antimicrobial and Phytochemistry study of Dendrobium linearifolium Teijsm. & Binn. from Gumitir, Jember, Indonesia

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Study of the Anti-klebsiella Activity of Quinazoline Compounds Containing a Piperazine Ring

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Medicinal chemistry perspectives on the development of piperazine-containing HIV-1 inhibitors

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Design, synthesis, X-ray crystal structure and antibacterial activity of ferulic acid derivatives bearing sulfonamide moiety

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Synthesis of Antifungal Heterocycle-Containing Mannich Bases: A Comprehensive Review

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Novel pyrazoline-piperazine conjugates as anticancer and antibacterial agents: integrating synthesis, in vitro, QSAR, molecular docking, and MD simulation studies

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Synthesis and DNA Cleavage Activity of Cationic Methylene-Blue-Backboned Polymers

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Rearrangement reactions: Important tool for the synthesis of piperazines

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Recent Developments in the Antimicrobial Potential of Some Nitrogenous Heterocycles and their SAR Studies: A Review

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Discovery of Arylpiperazines with Broad‐Spectrum Antimicrobial Activity and Favorable Pharmacokinetic Profiles

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Fragmentation of Polyfunctional Compounds Recorded Using Automated High-Throughput Desorption Electrospray Ionization

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Design, Synthesis, Computational Study, and Biological Evaluation of Sulfonyl Tethered Piperazine Derivatives as Antimicrobial Agents

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Experimental and Theoretical Investigations of the Inhibition of the Corrosion of Mild Steel in HCl by Synthesized Piperazin Derivatives

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Leveraging the MMV Pathogen Box to Engineer an Antifungal Compound with Improved Efficacy and Selectivity against Candida auris

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One-Pot Synthesis of Polyvinyl Alcohol-Piperazine Cross-Linked Polymer for Antibacterial Applications

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Asymmetric Construction of α,α‐Disubstituted Piperazinones Enabled by Benzilic Amide Rearrangement

Yu‐Ping He, Rui Quan, Xing‐Zi Li, Jieping Zhu and Hua Wu

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Design and synthesis of fluorescent calix[4]arene-1,8-Naphthalimide derivatives: Transparent biofilms, antioxidant and antimicrobial properties, and real-samples applications

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Synthesis, crystal structure and negative hyperconjugation study of quinoxaline derivatives containing piperazine

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Novel pyrimidine-piperazine hybrids as potential antimicrobial agents: in-vitro antimicrobial and in-silico studies

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Recent advances in piperazine derivatives as antibacterial agents: a comprehensive review (2020–2024)

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Mol Divers, 2025
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A practical and environmentally sustainable approach to dye removal: Synthesis and characterization of a highly efficient crosslinked chitosan-Schiff base adsorbent for Eriochrome Black T removal

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Design, synthesis, and antimicrobial evaluation of novel quinazoline piperazine phosphorodiamidate hybrids as potent DNA gyrase inhibitors

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Piperazine as a privileged scaffold in medicinal chemistry: biological activities, synthetic strategies, and multitarget drug design

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Synthesis, molecular docking, ADME study, and antimicrobial potency of piperazine based cinnamic acid bearing coumarin moieties as a DNA gyrase inhibitor

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2,3-Diketopiperazine as potential scaffold to develop new anti-Chagasic agents

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Discovery of piperazine‐tethered N‐heterocycle derivatives as anticancer agents

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Novel Hybrid Heterocycles Based on 1,4-Diphenylpiperazine Moiety: Synthesis via Hantzsch and Biginelli Reactions, Molecular Docking Simulation, and Antimicrobial Activities

Hadeer M. Diab, Mostafa E. Salem, Manal Abdellatif, Mona M. Soliman, Ismail A. Abdelhamid, Ahmed H. M. Elwahy, Nadeem Raza and Yassmen A. El-Gabry

ACS Omega, 2025, 10, 38014
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Searching for Suitable Kojic Acid Coformers: From Cocrystals and Salt to Eutectics

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Hydrogen bonding, halogen bonding and C–H…π interactions governing the supramolecular architecture of 1-(4-(4-bromophenyl)piperazin-1-yl)-2-chloroethan-1-one: Insights from X-ray crystallography, DFT calculations and urease inhibitory assessment

Sumera Zaib, Imtiaz Khan, Aliya Ibrar, Nehal Rana, Hafiz Saqib Ali, Christopher John McAdam, Rosa M. Gomila, Islam H. El Azab, M.H.H. Mahmoud, Zeinhom M. El-Bahy and Antonio Frontera

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Neuropharmacological Potential of Different Piperazine Analogs: A Recent Prospective

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1,3,4-Thiadiazole: A Promising Pharmacophore

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Design, Synthesis, and Biological Evaluation of Natural Carbolic Acid‐Pyrazinamide Hybrids as Antimicrobial Agents

Kripa Patel, Afzal Nagani, Moksh Shah and Khyati Patel

ChemistrySelect, 2025, 10
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Multifaced Antifungal Activity of Dialdehyde Chitosan Loaded with Zinc Metal-Organic Framework (Zn-MOF)

Gideon Kiprono Kirui, Edwin Shigwenya Madivoli, Dennis Mwanza Nzilu, Patrick Gachoki Kareru and Walyambillah Waudo

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Synthesis of Fumed-Pr-Pi-TCT as a Fluorescent Chemosensor for the Detection of Cyanide Ions in Aqueous Media

Sepideh Saberi Afshar, Ghodsi Mohammadi Ziarani, Fatemeh Mohajer, Alireza Badiei, Siavash Iravani and Rajender S. Varma

Water, 2022, 14, 4137
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Synthesis of Piperazine-containing Derivatives and their Antimicrobial, Antimycobacterial, Antimalarial and Antioxidant Activities

Navin B. Patel, Pratik N. Maisuria, Akash V. Gujarati and Divyesh K. Patel

CBC, 2024, 20
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Meclizine and Cephalosporin Combination as Promising Antibiotic Drugs: Formulation, Antimicrobial, and In Silico Studies

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Synthesis, characterization and application of piperazine based cationic gemini surfactants as antimicrobial agents

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Journal of Molecular Structure, 2025, 1345, 143053
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Deciphering the biocontrol strategies of Trichoderma yunnanense TM10 against Fusarium oxysporum f. sp. cepae, the causal agent of wilt disease in shallots (Allium cepa var. aggregatum)

Muhammad Adil Awal, Dedat Prismantoro, Reza Fauzi Dwisandi, Kah-Ooi Chua, Muhamad Shakirin Mispan, Nurul Shamsinah Mohd Suhaimi, Ratu Safitri and Febri Doni

Current Research in Microbial Sciences, 2025, 9, 100484
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Designing AI-generated antimicrobials for targeting bacterial microdomains

Mateusz Rzycki and Adam Gruda

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A high-fidelity dual-channel fluorescence probe for benzoyl peroxide detection and toxicity early warning in food, zebrafish, and mice

Pengxu Lin, Xiongjie Zhao, Ting Liu, Xiaomin Yuan and Liyi Zhou

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Antimicrobial polymeric paints: An up‐to‐date review

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Polymers for Advanced Techs, 2021, 32, 4642
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1,2‐Dichloroethane‐Assisted Defluorinative Ring‐Opening Reaction of DABCO and Polyfluoroalkyl Peroxides: Synthesis of Fluorinated N‐Ethyl Piperazines

Yuan‐Yuan Ren, Wen‐Jun Ji, Chi Zhang, Danhua Ge, Mengtao Ma, Zhi‐Liang Shen and Xue‐Qiang Chu

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Novel ionothermal synthesis of PZ-MIL-101 (Cr) at low temperature for CO2 and VOCs adsorption

Sachin Kuchekar, Sanjit Gaikwad and Sangil Han

Journal of Environmental Chemical Engineering, 2025, 13, 116884
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4‐Hydroxycoumarin: A Versatile Substrate for Transition‐metal‐free Multicomponent Synthesis of Bioactive Heterocycles

Biplob Borah, Kartikey Dhar Dwivedi and L. Raju Chowhan

Asian J Org Chem, 2021, 10, 3101
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