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Methyltetrazine as a small live-cell compatible bioorthogonal handle for imaging enzyme activities in situ

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Synthetic and Systems Biotechnology, 2018, 3, 34
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Labelled Chemical Probes for Demonstrating Direct Target Engagement in Living Systems

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AMTAC-19, a Spiro-Acridine Compound, Induces In Vitro Antitumor Effect via the ROS-ERK/JNK Signaling Pathway

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Small-Molecule Modulation of Protein Homeostasis

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Determining Cysteines Available for Covalent Inhibition Across the Human Kinome

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Bioorthogonal Reactions in Activity-Based Protein Profiling

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Molecules, 2020, 25, 5994
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Protein Degradation by In-Cell Self-Assembly of Proteolysis Targeting Chimeras

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ACS Cent. Sci., 2016, 2, 927
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ERK1/2 inhibitors: New weapons to inhibit the RAS-regulated RAF-MEK1/2-ERK1/2 pathway

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Synthetic approaches to constructing proteolysis targeting chimeras (PROTACs)

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Structure-Guided Discovery and Preclinical Assessment of Novel (Thiophen-3-yl)aminopyrimidine Derivatives as Potent ERK1/2 Inhibitors

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Discovery of Novel Aromatic Urea-Imidazole Salt Derivatives for Cancer Therapy via Targeting ERK1/2

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Recent Advances about the Applications of Click Reaction in Chemical Proteomics

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Molecules, 2021, 26, 5368
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Visualization of Endogenous ERK1/2 in Cells with a Bioorthogonal Covalent Probe

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Bioconjugate Chem., 2017, 28, 1677
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Protein degradation: a validated therapeutic strategy with exciting prospects

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New Phenylpropanoid from Croton velutinus (Euphorbiaceae) as Potential Anticancer Natural Product Targeting MAPKs: Review with Docking Approach

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