Issue 27, 2015

Synthesis and indole coupling reactions of azetidine and oxetane sulfinate salts

Abstract

Azetidine and oxetane sulfinate salts are easily prepared from commercially available 3-iodoheterocycle precursors in a three-step sequence. They undergo smooth coupling reactions thereby providing an expedient route for the introduction of these four-membered heterocycles into indoles.

Graphical abstract: Synthesis and indole coupling reactions of azetidine and oxetane sulfinate salts

Supplementary files

Article information

Article type
Communication
Submitted
02 fev 2015
Accepted
23 fev 2015
First published
24 fev 2015

Chem. Commun., 2015,51, 5914-5916

Synthesis and indole coupling reactions of azetidine and oxetane sulfinate salts

A. M. A. Nassoy, P. Raubo and J. P. A. Harrity, Chem. Commun., 2015, 51, 5914 DOI: 10.1039/C5CC00975H

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