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On the way to potential antifungal compounds: synthesis and in vitro activity of 2-benzofuranylacetic acid amides

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The synthesis and investigation of novel 3-benzoylbenzofurans and pyrazole derivatives for anti-HIV activity

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Synthesis of some new pyrimidine-based pyrene/benzochromene hybrids as EGFR kinase inhibitors in HCT-116 cancer cells through apoptosis

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Synthesis, molecular docking analysis and in vitro evaluation of new heterocyclic hybrids of 4-aza-podophyllotoxin as potent cytotoxic agents

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Synthesis of 2,3-Dialkyl-5-hydroxybenzofurans via a One-pot, Three-step Reaction Sequence of 2-Monosubstituted 1,3-Diketones and 1,4-Benzoquinones

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De Novo Construction of Highly Substituted Chromones and Benzo[b]furans via a Switchable Transformation of 3-Alkynyl-4-pyrones with Active Methylene Compounds

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Diversity-Oriented Approach to Furan Building Blocks and Their Relevance in Organic Synthesis, Materials Science, and Medicinal Chemistry

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Exploration of Medicinal Properties and Metabolite Diversity Between Different Petiole Types of Simarouba Glauca: A Nontargeted Metabolomics Approach

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Isochromene and Dihydroisobenzofuran Electrosynthesis by a Highly Regiodivergent Cyclization of 2-Ethynylbenzaldehydes

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Recent advances on quinoxalines as target‐oriented chemotherapeutic anticancer agents through apoptosis

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New Benzofuran–Pyrazole-Based Compounds as Promising Antimicrobial Agents: Design, Synthesis, DNA Gyrase B Inhibition, and In Silico Studies

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Visible-light-mediated synthesis of functionalized benzofurans: an update

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Regioselective Reversal in One-Pot and Two-Step Reaction of 1-(2-Hydroxyphenyl)-Propargyl Alcohols with Aryl/Alkyl Mercaptan: Construction of 3-(Alkylthio)benzofurans and 2-(Alkylthiomethyl)benzofurans Starting from Identical Materials

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Eco-friendly synthetic routes of benzofuran-integrated pyridine or 1, 3, 4-thiadiazole under solvent-free conditions using the grinding technique

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Design, Synthesis, and Molecular Docking Studies of Triazolylpyridine and Triazolylpyridinylbenzofuran Hybrids as Potential EGFR Inhibitors

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Synthesis of novel benzofuran-4,7-quinones from 4,6-dimethoxybenzofurans specifically targeting breast and lung cancer cells

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Inhibition of Clostridioides difficile toxins TcdA and TcdB by the amiodarone derivative dronedarone

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BM7, a derivative of benzofuran, effectively fights cancer by promoting cancer cell apoptosis and impacting IL-6 levels

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Polygonum barbatum extract induces ER stress-mediated UPR and autophagy to suppress colorectal cancer growth

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Annulated Heterocyclic[g]Coumarin Composites: Synthetic Approaches and Bioactive Profiling

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Brief insight into the in silico properties, structure-activity relationships and biotransformation of fruquintinib, an anticancer drug of a new generation containing a privileged benzofuran scaffold

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Synthesis and Anti-Breast Cancer Potency of Mono- and Bis-(pyrazolyl[1,2,4]triazolo[3,4-b][1,3,4]thiadiazine) Derivatives as EGFR/CDK-2 Target Inhibitors

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Microtubule destabilising activity of selected 7-methoxy-2-phenylbenzo[b]furan derivative against primary and metastatic melanoma cells

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Benzofuran compound from Sophora tonkinensis Gagnep suppresses nasopharyngeal carcinoma growth via PI3K/AKT/mTOR pathway: evidence from molecular dynamics simulation and in vitro experiments

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Targeting sensitive and multidrug resistant leukemia cells with a novel benzofuran-isatin conjugate

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Two series of benzofuran and benzodifuran chelating chromophores with DR/NIR emission and anticancer activity

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Characterization of Volatilized Compounds in Conventional and Organic Vegetable-Source Alternative Meat-Curing Ingredients

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Exploration of Benzofuran/Indole‐Chalcone Conjugated 1,2,3‐Triazole Hybrids as Candida glabrata Agents: Design, Synthesis, Biological Evaluation, Molecular Docking, and In Silico ADMET Analysis

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Anticancer Potential of Halogen Derivatives of Methyl 6-Acetyl-5-Hydroxy-2-Methyl-1-Benzofuran-3-Carboxylate

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Copper-Catalyzed Trifunctionalization of Alkynes: One-Pot Assembly of Antifungal Benzofuro[3,2-d]pyrimidine-Containing Fused Heterocycles

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Lewis Base Controlled (4+3) and (4+2) Annulations of MBH Carbonates with Benzofuran‐Derived Azadienes: Access to Highly Substituted Benzofuro[3,2‐b]Azepines and Spirotetrahydroquinolines

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Phytochemical Investigation and Biological Evaluation of Disynaphia filifolia: A Novel Source of Tremetone in Asteraceae

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Examining the 2-aryl-5-nitrobenzofuran-based hydrazones for anti-breast (MCF-7) cancer activity, potential to induce cell cycle arrest and inhibit receptor tyrosine kinases (VEGFR-2 & EGFR)

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Sustainable sonochemistry in medicinal heterocycle design: Advances and anticancer implications

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Diastereoselective Synthesis of Dihydrobenzofuran Spirooxindoles and Their Transformation into Benzofuroquinolinones by Ring Expansion of Oxindole Core

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Synthesis of novel mono- and bis-pyrazolylthiazole derivatives as anti-liver cancer agents through EGFR/HER2 target inhibition

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Construction of an AND logic gate fluorescent probe for highly efficient detection of formaldehyde and Pim-1 kinase

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Exploiting heterogeneous Pd/C for accessing benzofuran in biomass-derived γ-valerolactone

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Modified chitosan: Insight on biomedical and industrial applications

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Ring-Closing Metathesis as Methodology for the Synthesis of 2- and 3-Arylbenzo[b]furans

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Furan and benzofuran derivatives as privileged scaffolds as anticancer agents: SAR and docking studies (2010 to till date)

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Development of on-DNA Formation of Benzofuran for DNA-Encoded Library Synthesis

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In silico Design, Synthesis and Biological Evaluation of Novel Chalcone Derivatives as Potent Tubulin-Targeting Anticancer Agents

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Metal‐Catalysed Synthesis of Benzofused Five‐Membered N/O/S‐Heterocycles, a Progressive Area in Synthetic Organic Chemistry

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Investigation of the electronic effect of 2-phenylbenzofuran-3-ol derivatives on the protein conformation-induced aggregation

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Benzofuran‐Chalcone Derivatives as VEGFR‐2 Inhibitors: Synthesis and Anticancer Evaluation

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Design, synthesis, computational evaluation and kinetic study of benzofuran-derived thiazolotriazole derivatives as potential anti-urease agents

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A versatile pH-sensitive hydrogel based on a high-performance dye: Monitoring the freshness of milk and chicken meat

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Heteroaryl Group Containing Trisubstituted Alkenes: Synthesis and Anti‐Tumor Activity

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Synthesis, Antimicrobial Evaluation, and Computational Study of Novel Fluorinated Benzofuran Derivatives

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Synthesis of benzofuro[3,2-c]quinolinones via one-pot reaction of 3-chlorooxindoles and salicylaldehydes

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(2Z,5Z)-5-((3-(Benzofuran-2-yl)-1-phenyl-1H-pyrazol-4-yl)methylene)-2-((4-methoxyphenyl)imino)-3-phenylthiazolidin-4-one

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Synthesis of Benzofuran Derivatives via a DMAP-Mediated Tandem Cyclization Reaction Involving ortho-Hydroxy α-Aminosulfones

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Molecules, 2024, 29, 3725
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Chiral vicinal diamines as promising ligands in Pd-catalyzed reductive Heck type cyclizations

Maria A. Ashatkina, Alexander N. Reznikov, Dmitry S. Nikerov, Daria I. Shamshina, Maria V. Sizova, Vadim A. Shiryaev and Yuri N. Klimochkin

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Visible Light‐Driven Iron‐Catalyzed Decarboxylative Cyclization Reaction for Synthesis of 3‐Amino‐2,3‐Dihydrobenzofuran Derivatives from 2‐Carboxymethoxybenzaldehydes and Aryl Amines

Wenli Sheng, Zhenyu Jiang, Qingyan Liu and Junmin Chen

Adv Synth Catal, 2025, 367
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Novel benzofuran/pterostilbene hybrids trigger programmed cell death and impair migration in CRC cells

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Sustainable Synthesis of 3-Acylmethylated Coumarins via Photoredox Catalytic Radical Addition/Cyclization in Aqueous Media

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J. Org. Chem., 2025, 90, 7738
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Discovering a New N‐acylhydrazone Tethered Isatin/Benzofuran Scaffold for Colorectal Cancer: Design, Synthesis, Biological Activity, and ADME‐Tox Modelling

Cristian J. Zambrano‐Forero, Santiago M. Arango, Angie Herrera‐Ramírez, Wilson Cardona‐Galeano, Jorge Quintero‑Saumeth and Andrés F. Yepes

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