Issue 42, 2016

A concise approach to indoles via oxidative C–H amination of 2-alkenylanilines using dioxygen as the sole oxidant

Abstract

A novel synthetic method to prepare indole derivatives from N-Ts-2-alkenylanilines has been achieved. This reaction is through an oxidative intramolecular C–H amination by using molecular oxygen as the sole oxidant. This protocol is operationally simple and environmental friendly, and provides a diverse range of substrate scope.

Graphical abstract: A concise approach to indoles via oxidative C–H amination of 2-alkenylanilines using dioxygen as the sole oxidant

Supplementary files

Article information

Article type
Paper
Submitted
05 feb 2016
Accepted
31 mrt 2016
First published
01 apr 2016

RSC Adv., 2016,6, 35764-35770

A concise approach to indoles via oxidative C–H amination of 2-alkenylanilines using dioxygen as the sole oxidant

A. Ma, Y. Li, J. Li and J. Deng, RSC Adv., 2016, 6, 35764 DOI: 10.1039/C6RA03378D

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