α,α-Difluoro-β-iminophosphonates, an alternative strategy towards the synthesis of α,α-difluoro-β-aminophosphonate derivatives

M. Z. Szewczyk, M. Rapp, D. Virieux, J.-L. Pirat and H. Koroniak

New J. Chem., 2017, 41, 6322
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Fluoro-C-glycosides and fluoro-carbasugars, hydrolytically stable and synthetically challenging glycomimetics

Eric Leclerc, Xavier Pannecoucke, Mélanie Ethève-Quelquejeu and Matthieu Sollogoub

Chem. Soc. Rev., 2013, 42, 4270
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Visible-light-mediated difluoromethylphosphonation of alkenes for the synthesis of CF2P-containing heterocycles

Qiang Yang, Qing-Qing Lin, Hou-Ying Xing and Zhi-Gang Zhao

Org. Chem. Front., 2019, 6, 3939
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Iminosugars as glycosyltransferase inhibitors

Irene Conforti and Alberto Marra

Org. Biomol. Chem., 2021, 19, 5439
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Synthesis and biological activity of β-fluoroalkyl β-amino alcohols

Pierfrancesco Bravo, Marcello Crucianelli, Taizo Ono and Matteo Zanda

Journal of Fluorine Chemistry, 1999, 97, 27
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A Bis-Glycosylamine Strategy for the Synthesis of Dimeric Iminosugars Based on a DAB-1 Scaffold

Kamilia Ould Lamara, Nathan Noël, Fabien Massicot, Jean-Luc Vasse, Stéphane P. Vincent and Jean-Bernard Behr

Molecules, 2025, 30, 226
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A Facile and Rapid Route to a New Series of Pyrrolizidines Structurally Related to (+)-Alexine and (+)-Australine

Jean-Bernard Behr, Audrey Erard and Georges Guillerm

Eur. J. Org. Chem., 2002, 2002, 1256
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Approaches to the Synthesis of Perfluoroalkyl‐Modified Carbohydrates and Derivatives: Thiosugars, Iminosugars, and Tetrahydro(thio)pyrans

María Laura Uhrig, Erwin W. Mora Flores and Al Postigo

Chemistry A European J, 2021, 27, 7813
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The preparation of α,α-difluoropropargylphosphonates

Xin Zhang and Donald J. Burton

Journal of Fluorine Chemistry, 2002, 116, 15
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Glycoside Mimics from Glycosylamines: Recent Progress

Cyril Nicolas and Olivier Martin

Molecules, 2018, 23, 1612
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A concise synthesis of 2,5-dideoxy-2,5-imino-d-mannitol (DMDP) and HomoDMDP from l-xylose

Jean-Bernard Behr and Georges Guillerm

Tetrahedron Letters, 2007, 48, 2369
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Nucleoside Analogues: Synthesis and Biological Properties of Azanucleoside Derivatives

Dácil Hernández and Alicia Boto

Eur J Org Chem, 2014, 2014, 2201
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An efficient synthesis of functionalized β-amino- and β-hydrazinoalkylphosphonates by three-component reaction between trialkyl phosphites, dialkyl acetylenedicarboxylates and aromatic amines or hydrazines

Akram Ranjbar Derranji, Mohammad Anary-Abbasinejad and Marziyeh Mohammadi

Mol Divers, 2024, 28, 73
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Synthesis of β-Aminophosphonates and -Phosphinates

Francisco Palacios, Concepción Alonso and Jesús M. de los Santos

Chem. Rev., 2005, 105, 899
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Synthesis of 2′,3′-dihydrosolanesyl analogues of β-d-arabinofuranosyl-1-monophosphoryldecaprenol with promising antimycobacterial activity

Michaël Bosco, Philippe Bisseret, Patricia Constant and Jacques Eustache

Tetrahedron Letters, 2007, 48, 153
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Stereoselective Synthesis of 1-C-Diethylphosphonomethyl and -difluoromethyl Iminosugars from Sugar Lactams

Thanh Van Tran, Jérôme Désiré, Nicolas Auberger and Yves Blériot

J. Org. Chem., 2022, 87, 7581
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Synthesis of N-substituted α,α-difluoro-β-aminophosphonates by addition of diethyl lithiodifluoromethylphosphonate to imines

Prabhakar Cherkupally and Petr Beier

Journal of Fluorine Chemistry, 2012, 141, 76
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Tunable Approach for the Stereoselective Synthesis of 1-C-Diethylphosphono(difluoromethyl) Iminosugars as Glycosyl Phosphate Mimics

Chloé Cocaud, Cyril Nicolas, Thomas Poisson, Xavier Pannecoucke, Claude Y. Legault and Olivier R. Martin

J. Org. Chem., 2017, 82, 2753
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A Divergent and Stereoselective Approach for the Syntheses of Some Polyhydroxylated Indolizidine and Pyrrolizidine Iminosugars

Anugula Rajender, Jalagam Prasada Rao and Batchu Venkateswara Rao

Eur J Org Chem, 2013, 2013, 1749
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Potent inhibition of chitin synthase by an azasugar—investigation of synergistic effect with UDP

Mounira Djebaili and Jean-Bernard Behr

Journal of Enzyme Inhibition and Medicinal Chemistry, 2005, 20, 123
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Dichotomous Selectivity in Indium-Mediated Aza-Barbier-Type Allylation of 2-N-Acetyl Glycosyl Sulfinylimines in Brine: Convenient Access to Potent Anti-Influenza Agents

Long-Zhi Lin, Sheng Yang, Wan-Hsuan Liu and Jiun-Jie Shie

J. Org. Chem., 2022, 87, 2324
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Fluorinated Phosphonates: Synthesis and Biomedical Application

Vadim D. Romanenko and Valery P. Kukhar

Chem. Rev., 2006, 106, 3868
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Iminosugars as glycosyltransferase inhibitors: synthesis of polyhydroxypyrrolidines and their evaluation on chitin synthase activity

Isabelle Gautier-Lefebvre, Jean-Bernard Behr, Georges Guillerm and Murielle Muzard

European Journal of Medicinal Chemistry, 2005, 40, 1255
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New Chiral Reagent for Installation of Pharmacophoric (S)‐ or (R)‐2‐(Alkoxyphosphono)‐1‐amino‐2,2‐difluoroethyl Groups

Chen Xie, Lijun Zhang, Haibo Mei, Romana Pajkert, Maksym Ponomarenko, Yi Pan, Gerd‐Volker Röschenthaler, Vadim A. Soloshonok and Jianlin Han

Chemistry A European J, 2016, 22, 7036
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Stereoselective synthesis of arabinose-derived phosphonates

Claire Bouix, Philippe Bisseret and Jacques Eustache

Tetrahedron Letters, 1998, 39, 825
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ChemInform Abstract: Synthesis of (Difluoromethyl)phosphonate Azasugars Designed as Inhibitors for Glycosyl Transferases.

J.‐B. BEHR, C. M. EVINA, PHUNG NGA PHUNG NGA and G. GUILLERM

ChemInform, 1997, 28
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Diastereoselective addition of diethyl difluoromethylphosphonate to enantiopure sulfinimines: synthesis of α,α-difluoro-β-aminophosphonates, phosphonic acids, and phosphonamidic acids

Gerd-Volker Röschenthaler, Valery P. Kukhar, Michael Yu. Belik, Kateryna I. Mazurenko and Alexander E. Sorochinsky

Tetrahedron, 2006, 62, 9902
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An unprecedented access to trifluoromethylthiosugar derivatives from thiocyanate precursors upon treatment with trifluoromethyltrimethylsilane

Marie-Noëlle Bouchu, Sylvie Large, Michaela Steng, Bernard Langlois and Jean-Pierre Praly

Carbohydrate Research, 1998, 314, 37
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Recent Advances on the Synthesis and Application of α,α-Difluoro-β-aminophosphonates

Youlong Du, Qian Wang, Haibo Mei, Romana Pajkert, Gerd-Volker Röschenthaler and Jianlin Han

Chinese Journal of Organic Chemistry, 2024, 44, 3686
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New asymmetric strategy for the total synthesis of naturally occurring (+)-alexine and (−)-7-epi-alexine

Masaki Takahashi, Tetsuya Maehara, Tetsuya Sengoku, Norifumi Fujita, Kunihiko Takabe and Hidemi Yoda

Tetrahedron, 2008, 64, 5254
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Selective Synthesis of α-Fluoro-β-keto- and α-Fluoro-β-aminophosphonates via Electrophilic Fluorination by Selectfluor

Kinga Radwan-Olszewska, Francisco Palacios and Pawel Kafarski

J. Org. Chem., 2011, 76, 1170
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Synthesis and Fucosidase Inhibitory Study of Unnatural Pyrrolidine Alkaloid 4-epi-(+)-Codonopsinine

Alexis Kotland, Fabien Accadbled, Koen Robeyns and Jean-Bernard Behr

J. Org. Chem., 2011, 76, 4094
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Concise Synthesis ofP-Glycosyl Alkenylphosphonates andP,C-di andP,P,Ctri-Glycosyl Phosphonates

Claude Grison and Hicham Chibli

Journal of Carbohydrate Chemistry, 2009, 28, 12
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1-C-phosphonomethyl- and 1-C-difluorophosphonomethyl-1,4-imino-l-arabinitols as Galf transferase inhibitors: A comparison

Chloé Cocaud, Ruixiang B. Zheng, Todd L. Lowary, Thomas Poisson, Xavier Pannecoucke, Cyril Nicolas and Olivier R. Martin

Carbohydrate Research, 2018, 461, 45
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C-Difluoromethylene-containing, C-trifluoromethyl and C-perfluoroalkyl carbohydrates. Synthesis by carbohydrate transformation or building block methods

Richard Plantier-Royon and Charles Portella

Carbohydrate Research, 2000, 327, 119
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