A method to identify small molecule/protein pairs susceptible to protein ubiquitination by the CRBN E3 ligase

Pinwen Cai, Chiara Disraeli, Basilius Sauter, Saule Zhanybekova and Dennis Gillingham

Chem. Sci., 2025, 16, 7730
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Incorporation of viridicatin alkaloid-like scaffolds into DNA-encoded chemical libraries

Xianfu Fang, Huilin Liao, Xiaohong Fan, Yiting Wang, Huihong Wang, Gong Zhang, Wei Fang, Yangfeng Li and Yizhou Li

Org. Biomol. Chem., 2023, 21, 2162
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Recent advances in DNA-encoded libraries

Yuting Gao, Jinlu Liu, Sijie Huang, Nana Du, Gong Zhang and Yizhou Li

Chem. Commun., 2025, 61, 10952
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Covalent Capture and Selection of DNA‐Encoded Chemical Libraries via Photo‐Activated Lysine‐Selective Crosslinkers

Haimei Wei, Tianyang Zhang, Yangfeng Li, Gong Zhang and Yizhou Li

Chemistry An Asian Journal, 2023, 18
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Affinity-Driven Aryl Diazonium Labeling of Peptide Receptors on Living Cells

Sheryl Sharma, Michael J. Naldrett, Makayla J. Gill and James W. Checco

J. Am. Chem. Soc., 2024, 146, 13676
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Challenges and Prospects of DNA-Encoded Library Data Interpretation

Moreno Wichert, Laura Guasch and Raphael M. Franzini

Chem. Rev., 2024, 124, 12551
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Advancing small-molecule drug discovery by encoded dual-display technologies

Alice Lessing, Dimitar Petrov and Jörg Scheuermann

Trends in Pharmacological Sciences, 2023, 44, 817
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Discovering Cell‐Targeting Ligands and Cell‐Surface Receptors by Selection of DNA‐Encoded Chemical Libraries against Cancer Cells without Predefined Targets

Yuhan Gui, Rui Hou, Yuchen Huang, Yu Zhou, Shihao Liu, Ling Meng, Ying Li, Fong Sang Lam, Ruoyun Ding, Yan Cao, Gang Li, Xiaojie Lu and Xiaoyu Li

Angewandte Chemie, 2025, 137
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Evolution of chemistry and selection technology for DNA-encoded library

Peixiang Ma, Shuning Zhang, Qianping Huang, Yuang Gu, Zhi Zhou, Wei Hou, Wei Yi and Hongtao Xu

Acta Pharmaceutica Sinica B, 2024, 14, 492
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Enzymatic Cleavage of Double‐Stranded DNA‐Encoded Libraries (DELs) to Single‐Stranded DELs with Compounds at the 3′ End: Its Application in Photo‐Crosslinking Selection

Masatoshi Niwa, Jun Hayashida, Munefumi Tokugawa, Takeshi Nanya, Masako Tanabe, Naoko Honda, Takehiko Inohana, Hajime Fukano, Yukihiro Shigeta, Takeshi Kuboyama and Shin Itoh

Chemistry A European J, 2024, 30
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Recording Binding Information Directly into DNA-Encoded Libraries Using Terminal Deoxynucleotidyl Transferase

Lukas A. Schneider, Basilius Sauter, Koder Dagher and Dennis Gillingham

J. Am. Chem. Soc., 2023, 145, 20874
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Mask and Release Strategy‐Enabled Diversity‐Oriented Synthesis for DNA‐Encoded Library

Silin Zhang, Haiman Zhang, Xiawen Liu, Ping Qi, Tingting Tan, Shengdong Wang, Hui Gao, Hongtao Xu, Zhi Zhou and Wei Yi

Advanced Science, 2024, 11
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Discovering Cell‐Targeting Ligands and Cell‐Surface Receptors by Selection of DNA‐Encoded Chemical Libraries against Cancer Cells without Predefined Targets

Yuhan Gui, Rui Hou, Yuchen Huang, Yu Zhou, Shihao Liu, Ling Meng, Ying Li, Fong Sang Lam, Ruoyun Ding, Yan Cao, Gang Li, Xiaojie Lu and Xiaoyu Li

Angew Chem Int Ed, 2025, 64
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Agonist Discovery for Membrane Proteins on Live Cells by Using DNA-encoded Libraries

Yiran Huang, Rui Hou, Fong Sang Lam, Yunxuan Jia, Yu Zhou, Xun He, Gang Li, Feng Xiong, Yan Cao, Dongyao Wang and Xiaoyu Li

J. Am. Chem. Soc., 2024, 146, 24638
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DNA‐Encoded Noncanonical Substrate Library for Protease Profiling

Huiya Zhang, Yuyu Xing, Yixuan Yang, Bixi Tang, Zhaoyun Zong, Jia Li, Yi Zang, Matthew Bogyo, Xiaojie Lu and Shiyu Chen

ChemBioChem, 2024, 25
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Direct Selection of DNA-Encoded Libraries for Biased Agonists of GPCRs on Live Cells

Bo Cai, Amal El Daibani, Yuntian Bai, Tao Che and Casey J. Krusemark

JACS Au, 2023, 3, 1076
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The Furan–Thiol–Amine Reaction Facilitates DNA-Compatible Thiopyrrole-Grafted Macrocyclization and Late-Stage Amine Transformation

Qigui Nie, Tingting Xu, Xianfu Fang, Yanrong Dan, Gong Zhang, Yangfeng Li, Jianbo Li and Yizhou Li

Org. Lett., 2025, 27, 498
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Fusion of enzymatic proteins: Enhancing biological activities and facilitating biological modifications

Agnieszka Rybarczyk, Talha Sultan, Nazim Hussain, Hafiz Muhammad Husnain Azam, Safa Rafique, Jakub Zdarta and Teofil Jesionowski

Advances in Colloid and Interface Science, 2025, 340, 103473
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