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Jyoti, Rahul Jamra, Naveen Banyal, Pragati Sharma, Rakesh Kumar, Pawan K. Sharma and Virender Singh

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Unravelling the mechanism of apoptosis induced by copper(ii) complexes of NN2-pincer ligands in lung cancer cells

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Recent advancement in the synthesis of quinoline derivatives via multicomponent reactions

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Designing novel anti-plasmodial quinoline–furanone hybrids: computational insights, synthesis, and biological evaluation targeting Plasmodium falciparum lactate dehydrogenase

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Morphology-dependent catalytic performance of Co3O4 nanomaterials in the oxidative dehydrogenation of tetrahydroquinolines

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Analysis of the structural diversity of heterocycles amongst European medicines agency approved pharmaceuticals (2014–2023)

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A molybdenum-catalyzed acceptorless dehydrogenative approach for quinoline synthesis using amino alcohol

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Facile access to tetrazoles and 1-substituted benzimidazoles using zerovalent copper nanoparticles as an inexpensive and efficient nanocatalyst and its anticancer study

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Design, synthesis and cytotoxic activity of molecular hybrids based on quinolin-8-yloxy and cinnamide hybrids and their apoptosis inducing property

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Halogen bonding accelerated aerobic dehydrogenative aromatization for 4-aminoquinoline preparation

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DDQ promoted metal-free oxidative cascade synthesis of acridinyl ketones and 4-benzoylacridinones from C4-functionalized 1,2,3,4-tetrahydroacridines

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Novel quinolinyl-thiazole hybrid candidates bearing N-methyl piperazine as potential anti-breast cancer agents: synthesis, biological evaluation and computational studies

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Divergent synthesis of pyrrolidone fused pyrimido[1,2-b]indazole through selective trapping of an enone intermediate by 1H-indazol-3-amine

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Direct alkylation of quinolines with organolithium-activated 1,1-diborylalkanes

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A trans-palladium dichloride complex with a bulky organosulfur ligand: syntheses, structure, and applications in catalytic alkylation of acetophenone and secondary alcohols using alcohols

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Design, synthesis, and antiproliferative screening of new quinoline derivatives bearing a cis-vinyl triamide motif as apoptosis activators and EGFR-TK inhibitors

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Hydrogenation and dehydrogenation of N-heterocycles under Cp*Co(iii)-catalysis

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Tertiary amines as a C1 synthon: metal-free synthesis of quinolines and 2-substituted quinolinesvia[3+2+1] aerobic cyclization and C–N bond cleavage

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New multifunctional hybrids as modulators of apoptosis markers and topoisomerase II in breast cancer therapy: synthesis, characterization, and in vitro and in silico studies

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Fe(iii)-catalyzed [4+2] annulation of anthranils and maleimides for pyrrolo[3,4-b]quinolinedione synthesis: application to rosettacin

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New 8-hydroxy quinoline-polycyclic aromatic hydrocarbon (PAH) conjugates and their sulfonated derivatives: effects of sulfonation and PAH size on their structural, supramolecular and cytotoxic properties

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Selenium compounds as promising antiviral agents

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Pd-catalyzed intramolecular C–H activation for the synthesis of fused-1,2,3-triazole quinolines and dihydroquinolines

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Exploring transmembrane allostery in the MexB: DB08385 variant as a promising inhibitor-like candidate against Pseudomonas aeruginosa antibiotic resistance: a computational study

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One-pot, efficient synthesis of fused quinoline analogues via room temperature C(sp3)–N cleavage/aromatization reaction

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In(OTf)3-catalysed A3-annulation strategy towards the synthesis of pyrazole-tethered quinoline derivatives and assessment of their luminescent properties

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EDA complex-enabled annulation

Suven Das

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α-Glucosidase and α-Amylase inhibitory potentials of Quinoline–Rhodanine–1,3,4-oxadiazole hybrids with kinetic studies, and computational insights

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Click chemistry in tuberculosis research: From drug design to therapeutic delivery - A systematic review

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The Application of Alkynes as 1,2-Dicarbonyl Substitutes in Organic Synthesis Through Iodination and Kornblum Oxidation

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Advances in Small-molecule Dual Inhibitors Targeting EGFR and HER2 Receptors as Anti-cancer Agents

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ortho-Selective Dearomative [2π + 2σ] Photocycloadditions of Bicyclic Aza-Arenes

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Green Synthesis of Pyridine and their Fused System: Harnessing the Catalytic Power of Ionic Liquids for Sustainable and Efficient Multicomponent Reaction

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An efficient synthesis of 9-phenyl-3,4-dihydroacridin-1(2H)-one analogues: Crystal structures and theoretical physicochemical studies

Satheeshkumar Rajendran, Kailasam Saravana Mani, Arul Murugesan, Thalía Delgado, Kolandaivel Prabha, Werner Kaminsky and Roberto Acevedo

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Recent advances in the chemistry of selenophenoquinoline heterocycles: Synthesis, reactivity and biological activity

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Journal of Organometallic Chemistry, 2023, 1001, 122872
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Investigation of 3-Arylidene-2,3-dihydro-8-nitro-4-quinolone Di-Spiro analogs: Structural elucidation, In-Silico molecular modeling and In-Vitro cytotoxicity against A549 lung cancer cells

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A Facile, One‐Pot, and Sustainable Synthesis of Poly‐Substitute Quinoline Analogs by Ag2O@GO as a Promising Catalyst

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ChemistrySelect, 2025, 10
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Biowaste‐Mediated Synthesis of CeO₂–TiO₂ Nanoparticles: An Efficient Recoverable Nanocatalyst for the Solvent‐Free Synthesis of Antipyrine Derivatives and Their Biological Evaluation

Bhaskar Dwivedi, Diksha Bhardwaj and Deepika Choudhary

ChemistrySelect, 2024, 9
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Amino acid- and peptide-conjugated heterocyclic compounds: A comprehensive review of Synthesis Strategies and biological activities

Fany Sylvianingsih, Unang Supratman and Rani Maharani

European Journal of Medicinal Chemistry, 2025, 290, 117534
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Solvatochromic fluorophores based on 6-fluoro-2-(aryl)quinoline-4-carboxylic acids: Synthesis, optical studies and evaluation of their antimicrobial and larvicidal properties

Tayná Rodrigues Olegário, Lidiane Gomes de Araújo, Bruno Galdino Lopes, Cláudia M. Zaccaron Cristiano, Jéssika de Oliveira Viana, Karen C. Weber, José Roberto Dantas, Edeltrudes de Oliveira Lima, Vanessa Costa Santos, Luana Beatriz Rocha da Silva, Euzébio Guimarães Barbosa, Lucas Ferreira Martins, Luciano Morais Lião, Edilson Beserra de Alencar Filho, Rodrigo Cristiano and Claudio Gabriel Lima-Junior

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Design, synthesis and molecular docking study of novel quinoline–triazole molecular hybrids as anticancer agents

Rajubai D. Bakale, Amruta N. Bhagat, Udhav V. Mhetre, Shyam V. Londhe, Sanket S. Rathod, Prafulla B. Choudhari and Kishan P. Haval

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A Sequential One‐Pot Synthesis of Quinoline‐Fused Benzoxe(Aze)pines via Intramolecular Reductive Heck Cyclisation

Praveen Kumar Rathod, Kukkamudi Mahesh and Panaganti Leelavathi

Journal of Heterocyclic Chem, 2025, 62, 1986
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Synthesis and biological activity of substituted 5-oxo-1,4,5,6,7,8-hexahydroquinoline-3-carboxamides

N. V. Nosova, М. О. Starovoytova, R. R. Mahmudov, V. V. Novikova, М. V. Dmitriev and V. L. Gein

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Design, synthesis, and biological evaluation of schiff base derivatives incorporating quinoline-1,2,3-triazole moieties: Antimicrobial, anticancer activities, DFT simulations, and molecular docking studies

Darshna K. Lakhnotra, Jay B. Maheta, Nargis H. Shaikh, Ila M. Ram, Yogesh O. Bhola, Sahajkumar Gandhi and Sureshkumar B. Koradiya

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A small‑molecule HDAC/PDE modulator activates human adipocyte UCP1 and resolves inflammatory signaling

Mayyasa Rammah, Atilio Reyes Romero, Najeeb Halabi, Sirin Abuaqel, Andrea Guennoun, Alexander Dömling, Jingxuan Shan and Lotfi Chouchane

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Cytotoxic Cu(II) Complexes with a Novel Quinoline Derivative Ligand: Synthesis, Molecular Docking, and Biological Activity Analysis

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ACS Omega, 2024, 9, 25014
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Rational synthesis, activity and mechanism insights of a new aminoquinoline salt against malaria parasites: in vitro and in vivo approaches

Bruno Assis de Oliveira, Felipe Oliveira Raimundo, Wenderson Tinorio de Paula, Jessica Corrêa Bezerra Bellei, Nícolas Glanzmann, Letícia Ferreira Machado, Amanda Luisa da Fonseca, Camila Simões Freitas, Isabelle Karine da Costa Nunes, Adolfo Firmino Neto, Vinícius Novaes Rocha, Henrique Marcelo Gualberto Pereira, Eduardo Antônio Ferraz Coelho, Fernando de Pilla Varotti, Kézia Katiani Gorza Scopel and Adilson David da Silva

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4-Aminoquinolines modulate RNA structure and function: Pharmacophore implications of a conformationally restricted polyamine

Md Ismail Hossain, Mason Myers, Danushika Herath, Ali H. Aldhumani, Hannah Boesger and Jennifer V. Hines

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Mn(OAc)3-Mediated One-Pot Condensation-Oxidative Annulation of 2-Alkynylanilines and 1,3-Ketoesters: Synthesis of 2-Substituted Quinolines

Kunlayanee Punjajom, Sureeporn Ruengsangtongkul, Jumreang Tummatorn, Praneet Paiboonsombat, Somsak Ruchirawat and Charnsak Thongsornkleeb

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One-Pot Synthesis of 4-Chloroquinolines via Bis(trichloromethyl) Carbonate and Triphenylphosphine Oxide-Mediated Cascade Reactions of N-Aryl Enaminones

Wenhao Wang, Daming Feng, Ping Zhang, Peng Huang and Chunhua Ge

J. Org. Chem., 2024, 89, 9949
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Gold-Catalyzed Synthesis of 4-(Trifluoromethyl)quinolinecarboxylates

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Quinoline-based metal complexes: Synthesis and applications

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Catalyzed protocol in the development of new quinoline derivatives: Recent updates

Mohd Arham Siddiqui, Salahuddin, Rajnish Kumar, Avijit Mazumder, Mohamed Jawed Ahsan and Mohammad Shahar Yar

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Synthesis of novel amidines via one-pot three component reactions: Selective topoisomerase I inhibitors with antiproliferative properties

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Front. Chem., 2022, 10
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Activity Profiling of Nitro‐Substituted Di(Hetero)Aryl 1,3,4‐ and 1,2,4‐Oxadiazoles: Antimicrobial, Cholinesterase Inhibition and Antioxidant Potential

Enikő Šikorová, Šárka Štěpánková, Eva Frýbová, Klára Konečná, Jana Korbielová, Markéta Švarcová, Ondřej Janďourek, Václav Pflégr, Szilvia Bősze and Martin Krátký

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Borrowing hydrogen and dehydrogenative/oxidative cyclization reactions catalyzed by a CCC-NHC pincer Re complex: An air stable catalyst for the synthesis of α-alkylated ketones and quinolines

Hoang H. Pham and T. Keith Hollis

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Designed Synthesis of Amino‐Azo‐Quinoline and Their Nickel(II) Complexes: Molecular Structure, Electrochemistry and an Insight Into Their In Vitro Anti‐Cancer Activities

Srijita Naskar, Koushik Sarkar, Supriyo Halder, Bidisha Chatterjee, Debjeet Chakraborty, Arka Laha, Rahul Sharma, Arup Kumar Mitra, Kausikisankar Pramanik and Sanjib Ganguly

Chemistry & Biodiversity, 2025, 22
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I2–DMSO-mediated formal [3 + 1 + 2] synthesis of pyrimido[1,2-b]indazole using 1,4-dithiane-2,5-diol as a surrogate of ethylene

Yong-Dong Du, Jun-Gang Wang, Jin-Yi Liu, Chun-Yan Wu, Run-Feng Hu and An-Xin Wu

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Synthesis of atophane-containing benzocyclopentaquinolines, benzacridines and bisbenzacridines

E. A. Dikusar, E. A. Akishina, S. S. Koval’skaya, S. G. Stepin and V. I. Potkin

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Lateral Deprotometallation‐Trapping Reactions on Methylated Pyridines, Quinolines and Quinoxalines Using Lithium Diethylamide

Mohamed Hasyeoui, Peter M. Chapple, Frédéric Lassagne, Thierry Roisnel, Marie Cordier, Ali Samarat, Yann Sarazin and Florence Mongin

Eur J Org Chem, 2023, 26
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Synthesis and characterization of two Cu(II) complexes of new quinoline-based carboxylic acid

Nurgün Büyükkıdan, Derviş Gök, Halil İlkimen and Musa Sarı

Journal of Molecular Structure, 2024, 1317, 139096
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β-formyl-β-nitroenamine: A user-friendly synthetic tool with versatile reactivities

Nagatoshi Nishiwaki

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Chemistry of Quinolines and their Agrochemical Potential

Divya Utreja, Riddhi Salotra, Gurbir Kaur, Shivali Sharma and Sonia Kaushal

COC, 2023, 26, 1895
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Green Synthesis of Molecules for the Treatment of Neglected Diseases

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CTMC, 2023, 23, 1004
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Three-Step Synthesis of N-(7-chloro-4-morpholinoquinolin-2-yl)benzamide from 4,7-Dichloroquinoline

Deiby F. Aparicio Acevedo, Marlyn C. Ortiz Villamizar and Vladimir V. Kouznetsov

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Aryl-quinoline-4-carbonyl hydrazone bearing different 2-methoxyphenoxyacetamides as potent α-glucosidase inhibitors; molecular dynamics, kinetic and structure–activity relationship studies

Haleh Hamedifar, Mahroo Mirfattahi, Minoo Khalili Ghomi, Homa Azizian, Aida Iraji, Milad Noori, Ali Moazzam, Navid Dastyafteh, Ali Nokhbehzaim, Katayoun Mehrpour, Shahrzad Javanshir, Somayeh Mojtabavi, Mohammad Ali Faramarzi, Bagher Larijani, Mir Hamed Hajimiri and Mohammad Mahdavi

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Synthesis of 2-Organoselenyl Quinolines via Electro-Oxidative Selenocyclization of Isocyanides

Peng-Fei Huang, Jia-Le Fu, Zhi-Gang Quan, Ke-Wen Tang and Yu Liu

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Recent Advances in Metal Complexes Based on Biomimetic and Biocompatible Organic Ligands against Leishmaniasis Infections: State of the Art and Alternatives

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Recent progress in the application of amidines for the synthesis of N-heterocyclic compounds

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Synthesis, Characterization, and Therapeutic Potential of Novel Schiff Base Metal Complexes: Nickel(II) and Copper(II) Complexes Based 2‐[(2‐Chloroquinolin‐3‐yl)methylidene]aminobenzenethiol (CQAT)

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The novel pyridine-fused quinolinone PQ-L5 exhibits antibacterial effects and enhances β-lactam activity by targeting PBP2a in methicillin-resistant Staphylococcus aureus

Wei Feng, Qian Yuan, Xiaowen Wang, Qianmei Wang, Ye Wei and Fengjun Sun

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Quinoline schiff bases (QSBs) and their derivatives: emerging trends in antimicrobial agents

Mansi Gandhi, Vishwajit Chavda and Shashi Ranga

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Biochemical and Computational Insights into the Therapeutic Potencies of Quinoline Appended Imidazole Compounds

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I2‐Promoted Povarov Multicomponent Reaction for the Synthesis of 2,2′‐Biquinolines and N‐Heteroaromatic Benzothiazoles

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Novel quinoline-4-thiazolidinone derivatives as anticancer agents targeting the biological macromolecular protein-EGFR tyrosine kinase with dual anticancer and antioxidant activities

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Dual Role of Choline Azide for One-Pot Synthesis of Quinolines and Quinazolines Using Versatile Magnetic Cu-Oxalate@Fe3O4 Catalyst

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Synthetic Organic Molecules as Metallic Corrosion Inhibitors: General Aspects and Trends

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Quinoline Derivatives with Different Functional Groups: Evaluation of Their Catecholase Activity

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Designing a Simple Quinoline‐Based Chromo‐Fluorogenic Receptor for Highly Specific Quantification of Copper (II) Ions: Environmental and Bioimaging Applications

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Diastereoselective Alkylation of Activated Nitrogen Heterocycles with Alkenyl Boronate Complexes

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2-Arylidene-6-methyl-2H-furo[3,2-c]pyran-3,4-diones: Design, synthesis, and evaluation of Anti-inflammatory, Anti-malarial, and Anti-cancer efficacy

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Design and Synthesis of Novel Fluorescent 2-(aryloxy)-3-(4,5-diaryl)-1H-imidazol-2-yl)quinolines: Solvatochromic, DFT, TD-DFT Studies, COX-1 and COX-2 Inhibition and Antioxidant Properties

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Dihydroquinolinone and Hexahydroacridinone Chalcones: Synthesis, Experimental, and Theoretical Investigations of Their Photophysical and Biological Activities

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Harnessing Electricity in Dehydrogenative Coupling: Transition Metal‐Free Synthesis of Quinoline Derivatives

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Synthesis, Characterization, In Silico and In Vivo Evaluation of Benzimidazole‐Bearing Quinoline Schiff Bases as New Anticonvulsant Agents

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