Helical sulfono-γ-AApeptides with predictable functions in protein recognition

Peng Sang, Yan Shi, Lulu Wei and Jianfeng Cai

RSC Chem. Biol., 2022, 3, 805
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Bottom-up design of peptide shapes in water using oligomers of N-methyl-l/d-alanine

Jumpei Morimoto, Marin Yokomine, Yota Shiratori, Takumi Ueda, Takayuki Nakamuro, Kiyofumi Takaba, Saori Maki-Yonekura, Koji Umezawa, Koichiro Miyanishi, Yasuhiro Fukuda, Takumu Watanabe, Mayuko Suga, Ayumi Inayoshi, Takuya Yoshida, Wataru Mizukami, Koh Takeuchi, Koji Yonekura, Eiichi Nakamura and Shinsuke Sando

Chem. Sci., 2025, 16, 10512
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Residue-based program of a β-peptoid twisted strand shape via a cyclopentane constraint

Jungyeon Kim, Hiroka Kobayashi, Marin Yokomine, Yota Shiratori, Takumi Ueda, Koh Takeuchi, Koji Umezawa, Daisuke Kuroda, Kouhei Tsumoto, Jumpei Morimoto and Shinsuke Sando

Org. Biomol. Chem., 2022, 20, 6994
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Fluorescent p53 helix mimetics pairing anticancer and bioimaging properties

Sintu Karmakar, Mimasha Mallik, Sushree Sulava, Unnati Modi, Suryanarayana Allu, Shruti Sangwan, Srinu Tothadi, J. Prakasha Reddy, Rajesh Vasita, Ashwini K. Nangia, Debasmita Pankaj Alone and Panchami Prabhakaran

Biomater. Sci., 2025, 13, 3828
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A high-resolution structural characterization and physicochemical study of how a peptoid binds to an oncoprotein MDM2

Marin Yokomine, Jumpei Morimoto, Yasuhiro Fukuda, Takumi Ueda, Koh Takeuchi, Koji Umezawa, Hideo Ago, Hiroaki Matsuura, Go Ueno, Akinobu Senoo, Satoru Nagatoishi, Kouhei Tsumoto and Shinsuke Sando

Chem. Sci., 2024, 15, 7051
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Selection of MDM2-binding peptides in Escherichia coli using an engineered split intein and aminoglycoside phosphotransferase

Yutaro Watanabe, Chiori Tezuka, Kana Nobusawa and Tsuyoshi Takahashi

Chem. Commun., 2025, 61, 6332
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Oligo(N‐methylalanine) as a Peptide‐Based Molecular Scaffold with a Minimal Structure and High Density of Functionalizable Sites

Marin Yokomine, Jumpei Morimoto, Yasuhiro Fukuda, Yota Shiratori, Daisuke Kuroda, Takumi Ueda, Koh Takeuchi, Kouhei Tsumoto and Shinsuke Sando

Angew Chem Int Ed, 2022, 61
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Review: Structure-Activity Relationship of Antimicrobial Peptoids

Priscilla L. Nyembe, Thandokuhle Ntombela and Maya M. Makatini

Pharmaceutics, 2023, 15, 1506
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Oligo(N‐methylalanine) as a Peptide‐Based Molecular Scaffold with a Minimal Structure and High Density of Functionalizable Sites

Marin Yokomine, Jumpei Morimoto, Yasuhiro Fukuda, Yota Shiratori, Daisuke Kuroda, Takumi Ueda, Koh Takeuchi, Kouhei Tsumoto and Shinsuke Sando

Angewandte Chemie, 2022, 134
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Amide-to-ester substitution as a stable alternative to N-methylation for increasing membrane permeability in cyclic peptides

Yuki Hosono, Satoshi Uchida, Moe Shinkai, Chad E. Townsend, Colin N. Kelly, Matthew R. Naylor, Hsiau-Wei Lee, Kayoko Kanamitsu, Mayumi Ishii, Ryosuke Ueki, Takumi Ueda, Koh Takeuchi, Masatake Sugita, Yutaka Akiyama, Scott R. Lokey, Jumpei Morimoto and Shinsuke Sando

Nat Commun, 2023, 14
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Tackling Undruggable Targets with Designer Peptidomimetics and Synthetic Biologics

Colin S. Swenson, Gunasheil Mandava, Deborah M. Thomas and Raymond E. Moellering

Chem. Rev., 2024, 124, 13020
DOI: 10.1021/acs.chemrev.4c00423

Guidelines for designing peptoid structures: Insights from the Peptoid Data Bank

James R. B. Eastwood, Ethan I. Weisberg, Dana Katz, Ronald N. Zuckermann and Kent Kirshenbaum

Peptide Science, 2023, 115
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Helical Foldamers and Stapled Peptides as New Modalities in Drug Discovery: Modulators of Protein-Protein Interactions

Keisuke Tsuchiya, Takashi Kurohara, Kiyoshi Fukuhara, Takashi Misawa and Yosuke Demizu

Processes, 2022, 10, 924
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Exploration of N‐Arylation of Backbone Amides as a Novel Tool for Conformational Modification in Peptides

Abha Dangi and Udaya Kiran Marelli

Chemistry A European J, 2023, 29
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Well‐Defined Anisotropic Self‐Assembly from Peptoids and Their Biomedical Applications

Yota Okuno and Yasuhiko Iwasaki

ChemMedChem, 2023, 18
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Development of a Systematic and Extensible Force Field for Peptoids (STEPs)

Bradley S. Harris, Karteek K. Bejagam and Marcel D. Baer

J. Phys. Chem. B, 2023, 127, 6573
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