Recent advances in asymmetric C–H bond functionalization enabled by chiral directing groups

Yun Wang, Shuang Wang, Jiayang Wang and Shaojie Lou

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Isoindolinone synthesis through Rh/Cu-catalyzed oxidative C–H/N–H annulation of N-methoxy benzamides with saturated ketones

Xiao Du, Yuntao Hu, Darun Yang, Decai Huang, Wendi Yang, Hailong Wu and Huaiqing Zhao

Org. Biomol. Chem., 2022, 20, 783
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Separation of a diastereomeric diol pair using the mechanical properties of crystals

Rama Krishna Gamidi, Monica Dandawate, Srinu Tothadi, Rahul Choudhury, Ashwini K. Nangia and D. Srinivasa Reddy

CrystEngComm, 2021, 23, 7056
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Microwave‐Assisted Ruthenium‐ and Rhodium‐Catalyzed Couplings of α‐Amino Acid Ester‐Derived Phosphinamides with Alkynes

Xue‐Hong Li, Jun‐Fang Gong and Mao‐Ping Song

Chemistry An Asian Journal, 2022, 17
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Visible‐Light‐Driven Isocyanide Insertion to o‐Alkenylanilines: A Route to Isoindolinone Synthesis

Anjali Dahiya, Bubul Das, Ashish Kumar Sahoo and Bhisma K. Patel

Adv Synth Catal, 2022, 364, 966
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Rhodium(III)‐Catalyzed Three‐Component Cascade Annulation for Modular Assembly of N‐Alkoxylated Isoindolin‐1‐Ones with Quaternary Carbon Center

Wenbo Hu, Liqin Yan, Youpeng Zuo, Shuwen Kong, Yue Pu, Qiang Tang, Xinyu Wang, Xinwei He and Yongjia Shang

Adv Synth Catal, 2022, 364, 2589
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Discovery and current developments of isoindolinone-based fungal natural products

Christian Bailly

European Journal of Medicinal Chemistry Reports, 2023, 9, 100112
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Recent Advances in Tandem CH Activation and Named Reactions Toward Structurally Diverse Small‐Molecule Heterocycles: Synergistic Effects and Mechanistic Insights

Chenglin Wu, Shiyu Chen, Yabei Long and Xinyu Qiu

Eur J Org Chem, 2026, 29
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Synthesis of Dihydroquinolinone Derivatives via the Cascade Reaction of o-Silylaryl Triflates with Pyrazolidinones

Mengyang Shen, Jie Zhao, Yuanshuang Xu, Xinying Zhang and Xuesen Fan

J. Org. Chem., 2021, 86, 15203
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An Acid-Mediated Multicomponent Domino Reaction for the Synthesis of N-Substituted Isoindolinones

Sudheer Kumar Karu, Meghanath Veludandi and Chandrasekharam Malapaka

Synthesis, 2025, 57, 417
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Synthesis of Chiral Sulfinamides Enabled by Polycyclic Ketone Monooxygenase Catalyzed Asymmetric Oxidation of Sulfenamides

Wanqing Xue, Yuqi Lin, Xiaomin Lin, Xinqi Xu, Jingjing Chen, Juan Lin and Ke-Yin Ye

ACS Catal., 2025, 15, 16247
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Asymmetric CH Functionalization Enabled by a Traceless Oxidizing Chiral Auxiliary

Shuang Wang, Ze‐Feng Luo, Yang‐Jie Mao, Peng Ye, Zhen‐Yuan Xu, Dan‐Qian Xu and Shao‐Jie Lou

Adv Synth Catal, 2025, 367
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Rh(III)-Catalyzed Aminoalkylation of Alkenes with Diazo Compounds toward Functionalized Isoindolinones

Yuying Liu, Zhanwei Fu, Chao Yang, Mupeng Luo, Shurong Ban and Shouguo Wang

Chinese Journal of Organic Chemistry, 2024, 44, 3505
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The application of chiral amide directing group in asymmetric C–H activation

Wenkun Chen and Jun Wang

Sci. Sin.-Chim, 2025, 55, 370
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Asymmetric Synthesis of 3-Substituted Isoindolinones by Direct Alkylation of Chiral N-tert-Butylsulfinyl-isoindolinones

Qiang Yin, Zhilong Li, Jiaxin He, Yang Lai, Qianli Zhang and Haiying Sun

J. Org. Chem., 2025, 90, 3501
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Enantioselective Synthesis of Isoindolinone by Palladium-Catalyzed Aminoalkynylation of O-Phenyl Hydroxamic Ethers with Alkynes

Lei Wang, Yinqiang Wang, Shuaijie Wu, Chao-Guo Yan, Chaoshen Zhang, Junliang Zhang and Ying Han

J. Am. Chem. Soc., 2024, 146, 4320
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Rhodium(III)-Catalyzed Intramolecular Benzylic C(sp3)–H Amidation for the Synthesis of Isoindolinones

Darun Yang, Hongyan Xu, Decai Huang and Huaiqing Zhao

Synthesis, 2023, 55, 481
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Intramolecular reductive Heck reaction in the synthesis of 3,3-disubstituted isoindolin-1-ones

M. A. Ashatkina, A. N. Reznikov, S. Yu. Vostrukhina, D. S. Nikerov and Yu. N. Klimochkin

Russ Chem Bull, 2023, 72, 1809
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Unrevealing the Nitrogen Elusive Chirality of 3‐Sulfanyl and 3‐Sulfinyl N‐Tosyl Isoindolinones by ECD Spectra: An Experimental and Theoretical Investigation

Laura Palombi, Marta Monti, Erica Scarel, Valerio Morlacci, Mauro Stener and Massimiliano Aschi

Chemistry A European J, 2024, 30
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