Synthesis and characterization of nitrogen-based ionic liquids bearing allyl groups and examples of their application

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New J. Chem., 2020, 44, 12274
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A sialosyl sulfonate as a potent inhibitor of influenza virus replication

Ádám Hadházi, Mauro Pascolutti, Benjamin Bailly, Jeffrey C. Dyason, Anikó Borbás, Robin J. Thomson and Mark von Itzstein

Org. Biomol. Chem., 2017, 15, 5249
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Using batch reactor results to calculate optimal flow rates for the scale-up of UV photochemical reactions

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React. Chem. Eng., 2018, 3, 86
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Conformationally locked sugar derivatives and analogues as potential neuraminidase inhibitors

Yogesh Yadav, Rajdeep Tyagi, Ramesh Kumar and Ram Sagar

European Journal of Medicinal Chemistry, 2023, 255, 115410
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Process Intensification for the Synthesis of 6-Allyl-6-azabicyclo[3.1.0]hex-3-en-2-ol from 1-Allylpyridinium Salt Using a Continuous UV-Light Photoflow Approach

Milene A. G. Fortunato, Chi-Phong Ly, Filipa Siopa and Carlos A. M. Afonso

MPs, 2019, 2, 67
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From Pyridine to (−)‐Agelastatin A

João R. Vale, Milene A. G. Fortunato, Késsia H. S. Andrade, Ângelo M. R. Rocha, Carlos A. M. Afonso and Filipa Siopa

Adv Synth Catal, 2023, 365, 2240
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Ligand‐Controlled Regiodivergence in Nickel‐Catalyzed Vinylcyclopropane Rearrangement

Keiichi Irifune, Ken Yamazaki, Takayuki Nakamuro, Masahiro Murakami and Tomoya Miura

Angew Chem Int Ed, 2023, 62
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Design and synthesis of constrained bicyclic molecules as candidate inhibitors of influenza A neuraminidase

Cinzia Colombo, Črtomir Podlipnik, Leonardo Lo Presti, Masahiro Niikura, Andrew J. Bennet, Anna Bernardi and Joseph J Barchi

PLoS ONE, 2018, 13, e0193623
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Identification of neuraminidase inhibitors against dual H274Y/I222R mutant strains

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Sci Rep, 2017, 7
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Exploration of the 150 cavity and the role of serendipity in the discovery of inhibitors of influenza virus A neuraminidase

Sankar Mohan and B. Mario Pinto

Can. J. Chem., 2018, 96, 91
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Photochemical Rearrangements in Heterocyclic Chemistry

Corentin Lefebvre, Lucas Fortier and Norbert Hoffmann

Eur J Org Chem, 2020, 2020, 1393
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Benzimidazole-based DGAT1 inhibitors with a [3.1.0] bicyclohexane carboxylic acid moiety

Shuwen He, Zhong Lai, Qingmei Hong, Jackie Shang, Mikhail Reibarkh, Jeffrey T. Kuethe, Jian Liu, Deodial Guiadeen, Arto D. Krikorian, Timothy A. Cernak, Kevin D. Dykstra, Donald M. Sperbeck, Zhicai Wu, Yang Yu, Ginger X. Yang, Tianying Jian, Andreas Verras, Lisa M. Sonatore, Judyann Wiltsie, Christine C. Chung, Beth A. Murphy, Judith N. Gorski, Jinqi Liu, Jianying Xiao, Michael Wolff, Sharon X. Tong, Maria Madeira, Bindhu V. Karanam, Dong-Ming Shen, James M. Balkovec, Shirly Pinto, Ravi P. Nargund and Robert J. DeVita

Bioorganic & Medicinal Chemistry Letters, 2019, 29, 1182
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Design and synthesis of glycomimetics: Recent advances

Alice Tamburrini, Cinzia Colombo and Anna Bernardi

Medicinal Research Reviews, 2020, 40, 495
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Synthesis and Biological Evaluation of S-Substituted Perhalo-2-nitrobuta-1,3-dienes as Novel Xanthine Oxidase, Tyrosinase, Elastase, and Neuraminidase Inhibitors

Nihal Onul, Onur Ertik, Neşe Mermer and Refiye Yanardag

Journal of Chemistry, 2018, 2018, 1
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Asymmetric Divergent Total Syntheses of (+)-Decursivine and (+)- Serotobenine via Intramolecular Fischer Indole Synthesis

Dong-Hyun Kim, Hyo-Mi Kim, Ji-Su Lim, Hyun-Woo Lee and Cheon-Gyu Cho

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Flow-Assisted Synthesis of Bicyclic Aziridines via Photochemical Transformation of Pyridinium Salts

Filipa Siopa, João P. M. António and Carlos A. M. Afonso

Org. Process Res. Dev., 2018, 22, 551
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N1 neuraminidase of H5N1 avian influenza A virus complexed with sialic acid and zanamivir – A study by molecular docking and molecular dynamics simulation

R. A. Jeyaram and C. Anu Radha

Journal of Biomolecular Structure and Dynamics, 2022, 40, 11434
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Growing impact of sialic acid-containing glycans in future drug discovery

Priyanka Bose, Manoj K. Jaiswal, Sumit K. Singh, Rakesh K. Singh and Vinod K. Tiwari

Carbohydrate Research, 2023, 527, 108804
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Observation of a Tricyclic[4.1.0.02,4]heptane During a Michael Addition-Ring Closure Reaction and a Computational Study on Its Mechanism of Formation

Marco Farren-Dai, John R. Thompson, Anna Bernardi, Cinzia Colombo and Andrew J. Bennet

J. Org. Chem., 2017, 82, 12511
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Discovery of IACS-9779 and IACS-70465 as Potent Inhibitors Targeting Indoleamine 2,3-Dioxygenase 1 (IDO1) Apoenzyme

Matthew M. Hamilton, Faika Mseeh, Timothy J. McAfoos, Paul G. Leonard, Naphtali J. Reyna, Angela L. Harris, Alan Xu, Michelle Han, Michael J. Soth, Barbara Czako, Jay P. Theroff, Pijus K. Mandal, Jason P. Burke, Brett Virgin-Downey, Alessia Petrocchi, Dana Pfaffinger, Norma E. Rogers, Connor A. Parker, Simon S. Yu, Yongying Jiang, Stephan Krapp, Alfred Lammens, Graham Trevitt, Martin R. Tremblay, Keith Mikule, Keith Wilcoxen, Jason B. Cross, Philip Jones, Joseph R. Marszalek and Richard T. Lewis

J. Med. Chem., 2021, 64, 11302
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Palladium-catalyzed allylic substitution between C-based nucleophiles and 6-azabicyclo[3.1.0]-hex-3-en-2-oxy derivatives: A new selectivity paradigm

João A.C. Oliveira, Gredy Kiala, Filipa Siopa, Aurélie Bernard, Geoffrey Gontard, Julie Oble, Carlos A.M. Afonso and Giovanni Poli

Tetrahedron, 2020, 76, 131182
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Ligand‐Controlled Regiodivergence in Nickel‐Catalyzed Vinylcyclopropane Rearrangement

Keiichi Irifune, Ken Yamazaki, Takayuki Nakamuro, Masahiro Murakami and Tomoya Miura

Angewandte Chemie, 2023, 135
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(1R,4S,5S)-5-((3-Hydroxypropyl)amino)-4-((1-methyl-1H-tetrazol-5-yl)thio)cyclopent-2-en-1-ol

Milene Fortunato, Filipa Siopa and Carlos Afonso

Molbank, 2021, 2021, M1199
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