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Advances in pyrazolo[1,5-a]pyrimidines: synthesis and their role as protein kinase inhibitors in cancer treatment

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Recent trends in the synthesis and applications of β-iodovinyl sulfones: a decade of progress

Raju Jannapu Reddy, Jangam Jagadesh Kumar and Arram Haritha Kumari

Org. Biomol. Chem., 2024, 22, 2492
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Cs2CO3‐Promoted aza‐Michael Addition of (E)‐β‐Iodovinyl Sulfones with 5‐Amino‐1H‐pyrazole‐4‐carbaldehydes and Anthranilic Acids/Amides: Synthesis of 5‐Sulfonylpyrazolo[3,4‐b]pyridines and 3‐Sulfonyl‐4‐quinolones

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Advances in Vinyl Sulfone Catalyzed Synthesis: Methods, Mechanisms and Perspectives

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Asian J Org Chem, 2023, 12
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Synthesis of (E)‐β‐Iodovinyl Sulfones via HI‐mediated Vicinal Iodosulfonylation of Alkynes with Sodium Sulfinates

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Asian J Org Chem, 2024, 13
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Pd(II)-Catalyzed Tandem Cycloannulative-Alkenylation of o-Alkynyl-Phenols/Anilines with (E)-β-Iodovinyl Sulfones: A Direct Strategy To Construct 3-(Vinyl sulfonyl)benzoheterole Derivatives

Raju Jannapu Reddy, Nunavath Sharadha and Gamidi Rama Krishna

J. Org. Chem., 2023, 88, 8889
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Enantioconvergent Radical–Radical Cross-Coupling via Magnesium-Mediated Charge-Transfer Photocatalysis

Lei Yan, Hui-Qing Yang, Wan-Lei Yu, Xu-Gang Zhang and Peng-Fei Xu

J. Am. Chem. Soc., 2025, 147, 25264
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Synthesis of Sulfonylthiophenes through [3+2] Cycloaddition of Pyridinium 1,4-Zwitterionic Thiolates with (E)-β-Iodovinyl Sulfones or Bromoallylsulfones

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Unified Radical Sulfonylative-Annulation of 1,6-Enynols with Sodium Sulfinates: A Modular Synthesis of 2,3-Disubstituted Benzoheteroles

Raju Jannapu Reddy, Arram Haritha Kumari and Gamidi Rama Krishna

J. Org. Chem., 2023, 88, 1635
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Transition‐Metal‐Free Annulation of Sulfonyl‐Derived 1,3‐Enynes: Simple and Efficient Construction of 2,4‐Disubstituted Thiophenes and Vinyl Sulfone‐Tethered 1,2,3‐NH‐Triazoles

Nunavath Sharadha, Arram Haritha Kumari and Raju Jannapu Reddy

Asian J Org Chem, 2024, 13
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Recent highlights in the synthesis and biological significance of pyrazole derivatives

Ziad Moussa, Mani Ramanathan, Shaikha Mohammad Alharmoozi, Shahad Ali Saeed Alkaabi, Salamah Hamdan Mohammed Al Aryani, Saleh A. Ahmed and Harbi Tomah Al-Masri

Heliyon, 2024, 10, e38894
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K3PO4‐Promoted Cycloannulation of (E)‐β‐Iodovinyl Sulfones with ortho‐Hydroxy‐Chalcones/Cinnamates for the Synthesis of 2,3,4‐Trisubstituted 4H‐Benzopyran Derivatives

Raju Jannapu Reddy, Jangam Jagadesh Kumar and Gamidi Rama Krishna

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Synthetic and Pharmacological Expedition of Pyrazolo[1,5-a]pyridine: A Comprehensive Review

Neetu Agrawal, Dimple Bansal and Vertika Gautam

LDDD, 2024, 21, 71
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Mn(OAc)3-Mediated Unexpected Cycloannulative Sulfonyl Migration Cascade using (E)-β-Iodovinyl Sulfones and ortho-Alkynylphenols for Direct Synthesis of Chromene-Derived Vinyl Sulfones

Raju Jannapu Reddy, Jangam Jagadesh Kumar and Arram Haritha Kumari

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A bioactive sprite: Recent advances in the application of vinyl sulfones in drug design and organic synthesis

Jiangtao Tong, Jiong Shu, Yuhua Wang, Yajuan Qi and Yumei Wang

Life Sciences, 2024, 352, 122904
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Visible‐Light‐Induced Radical Sulfonylative‐Cyclization Cascade of 1,6‐Enynol Derivatives with Sulfinic Acids: A Sustainable Approach for the Synthesis of 2,3‐Disubstituted Benzoheteroles

Arram Haritha Kumari, Jangam Jagadesh Kumar, Nunavath Sharadha, Gamidi Rama Krishna and Raju Jannapu Reddy

ChemSusChem, 2024
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Simple and green synthesis of 3‐acyl‐pyrazolo[1,5‐a]pyridines: [3+2] through cycloaddition of N‐aminopyridines on enaminones

Sébastien Redon and Patrice Vanelle

Journal of Heterocyclic Chem, 2024, 61, 1200
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