Vajja Krishna Rao, Subarno Paul, Mitchell Gulkis, Zhihang Shen, Haritha Nair, Amandeep Singh, Chenglong Li, Arun K. Sharma, Melike Çağlayan, Chinmay Das, Biswajit Das, Chanakya N. Kundu, Satya Narayan and Sankar K. Guchhait
RSC Med. Chem., 2024,15, 937-962
From themed collection:
Meet the Editor webinar: celebrating our speakers and their contributions to the field
Abstract
In this study, a unique strategy of scaffold-hopping-based molecular editing of a bioactive agent NSC-666719 was investigated, which led to the development of new benzodithiazinedioxide-guanidine based anticancer agents with Polβ inhibition.
Hassan Seyrani, Sorour Ramezanpour, Aref Vaezghaemi and Farzad Kobarfard
New J. Chem., 2023,47, 21577-21577
Meng-Yang Chang and Nai-Chen Hsueh
Org. Biomol. Chem., 2025,23, 3572-3582
Abstract
We report the one-pot two-step synthesis of diaroyl benzothiepine-1,1-dioxides via the rongalite-mediated double sulfination of α-bromoacetophenones followed by double condensation of the resulting 1,3-diaroyl sulfones and o-phthalaldehydes.
Pooja R. Solanke, Prakash Kumar, Prathama S. Mainkar, Kiranmai Nayani and Srivari Chandrasekhar
Chem. Commun., 2024,60, 4234-4237
Abstract
A novel diastereoselective one-pot protocol has been developed through sequential execution of an aza-Piancatelli rearrangement and a Conia-ene type reaction under Lewis acid catalysis.
Boxu Lin, Tianran Liu and Tuoping Luo
Nat. Prod. Rep., 2024,41, 1091-1112
From themed collection:
The Synergy of Synthetic Methods Development and Natural Product Synthesis
Abstract
This review highlights a curated selection of publications utilizing homogeneous gold-catalyzed cycloaddition and cyclization reactions for the total synthesis of natural products reported from 2016 to mid-2023.