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DOI: 10.1016/j.bmc.2014.11.039

Addressing phototoxicity observed in a novel series of biaryl derivatives: Discovery of potent, selective and orally active phosphodiesterase 10A inhibitor ASP9436

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Bioorganic & Medicinal Chemistry, 2015, 23, 3351
DOI: 10.1016/j.bmc.2015.04.052

Novel Formation of Oxazepino[4,5-a]quinolines by Tandem 1,3-Dipolar and Insertion Reaction of Quinoline N-Oxides with Arynes

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