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Evaluating the biological effectiveness of boron neutron capture therapy by using microfluidics-based pancreatic tumor spheroids

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Introducing borane clusters into polymeric frameworks: architecture, synthesis, and applications

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Tailored hyaluronic acid-based nanogels as theranostic boron delivery systems for boron neutron cancer therapy

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Coordination-based molecular nanomaterials for biomedically relevant applications

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Extracellular Vesicles Comprising Carborane Prepared by a Host Exchanging Reaction as a Boron Carrier for Boron Neutron Capture Therapy

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Boron Agent Delivery Platforms Based on Natural Products for Boron Neutron Capture Therapy

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ChemMedChem, 2024, 19
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Characteristic evaluation of the thermal neutron irradiation field using a 30 MeV cyclotron accelerator for basic research on neutron capture therapy

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Nuclear Instruments and Methods in Physics Research Section A: Accelerators, Spectrometers, Detectors and Associated Equipment, 2020, 983, 164533
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Targeting the organelle for radiosensitization in cancer radiotherapy

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Asian Journal of Pharmaceutical Sciences, 2024, 19, 100903
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Next generation of boron neutron capture therapy (BNCT) agents for cancer treatment

Paolo Coghi, Jinxin Li, Narayan S. Hosmane and Yinghuai Zhu

Medicinal Research Reviews, 2023, 43, 1809
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Progress in three-dimensional aromatic-like closo-dodecaborate

Xue Zhao, Ziqiong Yang, Hao Chen, Zhenxi Wang, Xiaohai Zhou and Haibo Zhang

Coordination Chemistry Reviews, 2021, 444, 214042
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Peptide-Drug Conjugates and Their Targets in Advanced Cancer Therapies

Paul Hoppenz, Sylvia Els-Heindl and Annette G. Beck-Sickinger

Front. Chem., 2020, 8
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Simple Cytosolic and Nuclear Introduction of Boron Compounds Using Cationic Lipids to Enhance Cancer Cell-Killing Activity in Boron Neutron Capture Therapy

Shiori Hirase, Yurina Araki, Yoshihide Hattori, Ayako Aoki, Daisuke Fujiwara, Masataka Michigami, Tomoka Takatani-Nakase, Ikuo Fujii, Shiroh Futaki, Mitsunori Kirihata and Ikuhiko Nakase

Biological & Pharmaceutical Bulletin, 2025, 48, 344
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Theranostics in Boron Neutron Capture Therapy

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Dodecaborate-Encapsulated Extracellular Vesicles with Modification of Cell-Penetrating Peptides for Enhancing Macropinocytotic Cellular Uptake and Biological Activity in Boron Neutron Capture Therapy

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Carboranes as unique pharmacophores in antitumor medicinal chemistry

Yu Chen, Fukuan Du, Liyao Tang, Jinrun Xu, Yueshui Zhao, Xu Wu, Mingxing Li, Jing Shen, Qinglian Wen, Chi Hin Cho and Zhangang Xiao

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Clinical Viability of Boron Neutron Capture Therapy for Personalized Radiation Treatment

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Cancers, 2022, 14, 2865
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Towards the Application of Purely Inorganic Icosahedral Boron Clusters in Emerging Nanomedicine

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Molecules, 2023, 28, 4449
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Research and development of boron drugs used for cancer boron neutron capture therapy (BNCT)

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Development of a prompt gamma-ray detector with an 8 × 8 array LaBr 3(Ce) scintillator and a multi-pixel photon counter for boron neutron capture therapy

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Nuclear Instruments and Methods in Physics Research Section A: Accelerators, Spectrometers, Detectors and Associated Equipment, 2023, 1055, 168546
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Improving the spatial resolution of a pixelated LaBr3(Ce) scintillator coupled with a multi-pixel photon counter array for boron neutron capture therapy

Keita Okazaki, Hiroki Tanaka, Takushi Takata, Naonori Hu, Tetsuya Mukawa, Yoshinori Sakurai and Minoru Suzuki

Nuclear Instruments and Methods in Physics Research Section A: Accelerators, Spectrometers, Detectors and Associated Equipment, 2021, 992, 165026
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Current Insights into the Radiobiology of Boron Neutron Capture Therapy and the Potential for Further Improving Biological Effectiveness

Leah D. Punshon, Maria Rita Fabbrizi, Ben Phoenix, Stuart Green and Jason L. Parsons

Cells, 2024, 13, 2065
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Reaction of Chloroacetyl-Modified Peptides with Mercaptoundecahydrododecaborate (BSH) Is Accelerated by Basic Amino Acid Residues in the Peptide

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Processes, 2022, 10, 2200
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Conceptual design of a target station using a 30-MeV cyclotron accelerator for the basic study of boron neutron capture therapy at KURNS

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Nuclear Instruments and Methods in Physics Research Section A: Accelerators, Spectrometers, Detectors and Associated Equipment, 2022, 1042, 167425
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Boron delivery systems for enhanced boron neutron capture therapy: a comprehensive review

Seungjin Yu, Goeun Choi and Jin-Ho Choy

Medical Lasers, 2023, 12, 71
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Proposal of recommended experimental protocols for in vitro and in vivo evaluation methods of boron agents for neutron capture therapy

Yoshihide Hattori, Tooru Andoh, Shinji Kawabata, Naonori Hu, Hiroyuki Michiue, Hiroyuki Nakamura, Takahiro Nomoto, Minoru Suzuki, Takushi Takata, Hiroki Tanaka, Tsubasa Watanabe and Koji Ono

Journal of Radiation Research, 2023, 64, 859
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A Selective Carborane-Functionalized Gastrin-Releasing Peptide Receptor Agonist as Boron Delivery Agent for Boron Neutron Capture Therapy

Paul Hoppenz, Sylvia Els-Heindl, Martin Kellert, Robert Kuhnert, Stefan Saretz, Hans-Georg Lerchen, Johannes Köbberling, Bernd Riedl, Evamarie Hey-Hawkins and Annette G. Beck-Sickinger

J. Org. Chem., 2020, 85, 1446
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Electrochemical Synthesis of Triphenylphosphine Coinage Metal Complexes stabilized by closo‐Dodecaborates [B12X12]2− (X=H, F, Cl, Br, I)

Rüdiger M. Exner, Carsten Jenne and Bianca Wegener

Zeitschrift anorg allge chemie, 2021, 647, 500
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Design, Synthesis and Biological Evaluation of Boron‐Containing Macrocyclic Polyamine Dimers and Their Zinc(II) Complexes for Boron Neutron Capture Therapy

Hiroki Ueda, Minoru Suzuki, Yoshinori Sakurai, Tomohiro Tanaka and Shin Aoki

Eur J Inorg Chem, 2022, 2022
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Particle and Heavy Ion Transport Code System‐Based Microdosimetry for the Development of Boron Agents for Boron Neutron Capture Therapy

Takafumi Shigehira, Tadashi Hanafusa, Kazuyo Igawa, Tomonari Kasai, Shuichi Furuya, Hisakazu Nishimori, Yoshinobu Maeda, Hiroyuki Michiue and Atsushi Fujimura

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Multi-Functional Boron-Delivery Agents for Boron Neutron Capture Therapy of Cancers

Sebastian O. Oloo, Kevin M. Smith and Maria da Graça H. Vicente

Cancers, 2023, 15, 3277
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Experimental verification of efficacy of pBCT in terms of physical and biological aspects

Mana Hosobuchi, Jun Kataoka, Hiromu Yokokawa, You Okazaki, Ryoichi Hirayama, Taku Inaniwa, Masashi Ueda and Mitsuhiro Kimura

Nuclear Instruments and Methods in Physics Research Section A: Accelerators, Spectrometers, Detectors and Associated Equipment, 2023, 1045, 167537
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Aza-BODIPY: A New Vector for Enhanced Theranostic Boron Neutron Capture Therapy Applications

Ghadir Kalot, Amélie Godard, Benoît Busser, Jacques Pliquett, Mans Broekgaarden, Vincent Motto-Ros, Karl David Wegner, Ute Resch-Genger, Ulli Köster, Franck Denat, Jean-Luc Coll, Ewen Bodio, Christine Goze and Lucie Sancey

Cells, 2020, 9, 1953
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Hyaluronic acid-decorated carborane-TAT conjugation nanomicelles: A potential boron agent with enhanced selectivity of tumor cellular uptake

Hao Quan, Li Fan, Yushu Huang, Xiaoyan Xia, Yang He, Shiyuan Liu and Jiahui Yu

Colloids and Surfaces B: Biointerfaces, 2021, 204, 111826
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The Dawn of a New Era: Tumor-Targeting Boron Agents for Neutron Capture Therapy

Ting Luo, Wenzhi Huang, Feiyi Chu, Tianyu Zhu, Bin Feng, Shuai Huang, Jing Hou, Liyong Zhu, Shaihong Zhu and Wenbin Zeng

Mol. Pharmaceutics, 2023, 20, 4942
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Design, Synthesis, and Biological Evaluation of Boron-Containing Macrocyclic Polyamines and Their Zinc(II) Complexes for Boron Neutron Capture Therapy

Hiroki Ueda, Minoru Suzuki, Reiko Kuroda, Tomohiro Tanaka and Shin Aoki

J. Med. Chem., 2021, 64, 8523
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Multifunctional high boron content MOFs nano-co-crystals for precise boron neutron capture therapy for brain glioma in situ

Zhijie Wang, Ziteng Chen, Zizhu Zhang, Jiacheng Li, Kui Chen, Haojun Liang, Linwen Lv, Yannan Chang, Sen Liu, Wenjiang Yang, Zhi Yang, Hui Yuan, Xiangxi Meng, Tong Liu, Feng Wang, Juan Li and Gengmei Xing

Nano Today, 2022, 45, 101558
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Improvement of Water Solubility of Mercaptoundecahydrododecaborate (BSH)-Peptides by Conjugating with Ethylene Glycol Linker and Interaction with Cyclodextrin

Mizuki Kitamatsu, Ayaka Nakamura-Tachibana, Yoshimichi Ishikawa and Hiroyuki Michiue

Processes, 2021, 9, 167
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Dodecaborate Conjugates Targeting Tumor Cell Overexpressing Translocator Protein for Boron Neutron Capture Therapy

Yoshihide Hattori, Miki Ishimura, Youichirou Ohta, Hiroshi Takenaka, Shinji Kawabata and Mitsunori Kirihata

ACS Med. Chem. Lett., 2022, 13, 50
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Recent Development of Radiofluorination of Boron Agents for Boron Neutron Capture Therapy of Tumor: Creation of 18F-Labeled C-F and B-F Linkages

Jin-Pei Deng and Chung-Shan Yu

Pharmaceuticals, 2023, 16, 93
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An Improved Method for the Synthesis of M2[B12H12] (M = Na, K) and Their Formation Mechanism

Hui Han, Xin-Ran Liu, Yan-Mei Gao, Sha-Sha Liang, Yi Jing, Hai-Jun Li and Xuenian Chen

Inorg. Chem., 2024, 63, 13886
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In vivo investigation of boron-rich nanodrugs for treating triple-negative breast cancers via boron neutron capture therapy

Kai-Wei Lan, Wei-Yuan Huang, Yi-Lin Chiu, Fang-Tzu Hsu, Yun-Chen Chien, Yong-Yun Hsiau, Tzu-Wei Wang and Pei Yuin Keng

Biomaterials Advances, 2023, 155, 213699
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Copper‐Catalyzed Preparation of Alkenylboronates and Arylboronates

Safiul Alam, Rejaul Karim, Aminur Khan, Amarta Kumar Pal and Antoine Maruani

Eur J Org Chem, 2021, 2021, 6115
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Chemistry of three-dimensional icosahedral boron clusters anions: closo-dodecaborate (2-) [B12H12]2- and carba-closo-dodecaborate(-) [CB11H12]-

Lingyao Wang, Yunjia Jiang, Simon Duttwyler, Furong Lin and Yuanbin Zhang

Coordination Chemistry Reviews, 2024, 516, 215974
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Carborane-containing amino acids and peptides: Synthesis, properties and applications

Dmitry A. Gruzdev, Galina L. Levit, Victor P. Krasnov and Valery N. Charushin

Coordination Chemistry Reviews, 2021, 433, 213753
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Boron-peptide conjugates with angiopep-2 for boron neutron capture therapy

Jing Xiang, Lin Ma, Jianfei Tong, Nan Zuo, Weitao Hu, Yupeng Luo, Junqi Liu, Tianjiao Liang, Qiushi Ren and Qi Liu

Front. Med., 2023, 10
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