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Selective alkaline stripping of metal ions after solvent extraction by base-stable 1,2,3-triazolium ionic liquids

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Searching for novel reusable biomass-derived solvents: furfuryl alcohol/water azeotrope as a medium for waste-minimised copper-catalysed azide–alkyne cycloaddition

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A new four-component reaction involving the Michael addition and the Gewald reaction, leading to diverse biologically active 2-aminothiophenes

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Multicomponent cyclization with azides to synthesize N-heterocycles

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Click-chemistry approaches to π-conjugated polymers for organic electronics applications

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Convenient preparation of 4-diazoisochroman-3-imines and 3-subsituted 3,5-dihydroisochromeno[3,4-d][1,2,3]triazoles

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Synthesis of homochiral sulfanyl- and sulfoxide-substituted naphthyltriazoles and study of the conformational stability

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One-Pot MCR-Oxidation Approach toward Indole-Fused Heteroacenes

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1-(4-Nitrophenyl)-1H-1,2,3-Triazole-4-carbaldehyde: Scalable Synthesis and Its Use in the Preparation of 1-Alkyl-4-Formyl-1,2,3-triazoles

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Recent Advances in Multicomponent Synthesis of 1,4,5‐Trisubstituted 1,2,3‐Triazoles

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4,5,6,7-Tetrahydroindol-4-Ones as a Valuable Starting Point for the Synthesis of Polyheterocyclic Structures

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Molecules, 2021, 26, 4596
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Oxidative cyclization of 5-aryl-1-benzyl-1,2,3-triazoles bearing electron-rich aromatic groups: ortho/ortho and ortho/ipso coupling

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Synthesis, biological evaluation and molecular modeling of a novel series of fused 1,2,3-triazoles as potential anti-coronavirus agents

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Bioorganic & Medicinal Chemistry Letters, 2018, 28, 3472
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Structural modification strategies of triazoles in anticancer drug development

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Synthesis of Polycyclic Dihydroindoles by Selective Decomposition of Bis(1,2,3‐triazoles) Mediated by Rhodium Catalysis

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Ring-Degenerate Rearrangement Resulting from the Azo Coupling Reaction of a 3-Aryl-1,3a,6a-triazapentalene

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J. Org. Chem., 2020, 85, 9434
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Site-Selective N-Dealkylation of 1,2,3-Triazolium Salts: A Metal-Free Route to 1,5-Substituted 1,2,3-Triazoles and Related Bistriazoles

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Emerging Aspects of Triazole in Organic Synthesis: Exploring its Potential as a Gelator

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Synthesis of [6,5,5]Ring‐Fused Tricyclic Triazoles by Copper‐Promoted Double Cyclization

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A Multicomponent Approach toward Angularly Fused/Linear Bitriazoles: A Cascade Cornforth Rearrangement and Triazolization

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Heteroannulation of 3-Nitroindoles and 3-Nitrobenzo[b]thiophenes: A Multicomponent Approach toward Pyrrole-Fused Heterocycles

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Triazoles and Their Derivatives: Chemistry, Synthesis, and Therapeutic Applications

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Extending the Application Scope of Organophosphorus(V) Compounds in Palladium(II) Pincer Chemistry

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A Facile One-Pot Synthesis of New Poly Functionalized Pyrrolotriazoles via a Regioselective Multicomponent Cyclisation and Suzuki–Miyaura Coupling Reactions

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A comprehensive review on triazoles as anticancer agents

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Metal-free synthetic approaches to 1,5-disubstituted 1,2,3-triazoles

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Au-catalyzed domino process synthesis of imidazo[1,2-a]pyridines from 2-aminopyridine and N-tosylhydrazones: An efficient C N bond formation reaction

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Catalysis Communications, 2017, 90, 43
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Synthesis of Thieno[2,3‐c]pyridine Derivatives by 1,2,3‐Triazole‐Mediated Metal‐Free Denitrogenative Transformation Reaction

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ChemistryOpen, 2025, 14
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Catalyst-free synthesis of 4-acyl-NH-1,2,3-triazoles by water-mediated cycloaddition reactions of enaminones and tosyl azide

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A metal-free route towards 1,5-disubstituted 1,2,3-triazolylmethylene linked disaccharides: Synthesis in a biodegradable hydroxyl-ammonium-based aqueous ionic liquid media

Anirban Kayet and Tanmaya Pathak

Tetrahedron Letters, 2018, 59, 3341
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Transformation of Amides into Highly Functionalized Triazolines

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Synthesis of 1,2,3-Triazolo-Fused Allocolchicine Analogs via Intramolecular Oxidative Biaryl Coupling

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Enamines and their variants as intermediates for synthesis of aza-heterocycles with applications in MCRs

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Synthesis and characterization of novel axially chiral β-linked 1,2,3-triazolyl porphyrins

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Dyes and Pigments, 2018, 156, 61
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Triazolization of Enolizable Ketones with Primary Amines: A General Strategy toward Multifunctional 1,2,3‐Triazoles

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The Chemical Record, 2021, 21, 376
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1,2,3-Triazolium macrocycles in supramolecular chemistry

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Multicomponent Reactions in the Synthesis of Antiviral Compounds

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Antiproliferative effect of mitochondria-targeting allobetulin 1,2,3-triazolium salt derivatives and their mechanism of inducing apoptosis of cancer cells

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Application of the Triazolization Reaction to Afford Dihydroartemisinin Derivatives with Anti-HIV Activity

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Molecules, 2017, 22, 303
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Synthesis and anticancer activity of novel aza-artemisinin derivatives

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Bioorganic & Medicinal Chemistry, 2017, 25, 3671
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Functionalization of tetrahydroindol-4-one derivatives

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Chemical Series, 2022, 6
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Synthesis and Spectroscopic Properties of 1,2,3-Triazole BOPAHY Dyes and Their Water-Soluble Triazolium Salts

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Recent Progress in Catalytic Synthesis of 1,2,3-Triazoles

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Synthesis and Anti-HIV Activity of a Novel Series of Isoquinoline-Based CXCR4 Antagonists

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Molecules, 2021, 26, 6297
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Chiral Fused 1,2,3‐Triazoles: A Synthetic Overview

Manoj Dhameja, Hariom Kumar and Preeti Gupta

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Stitching Triazoles to Arenes via a Transition Metal-Free Aryne Diels–Alder/1,3-Prototropic Shift/Dehydrobromination Cascade

Ranadeep Talukdar, Vikram Singh, Hemlata Mourya, Malik Nasibullah and Bhoopendra Tiwari

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Metal‐Free Three‐Component Assembly of Fully Substituted 1,2,3‐Triazoles

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Asian J Org Chem, 2018, 7, 1698
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Triphenylphosphonium-linked derivative of allobetulin: preparation, anticancer properties and their mechanism of inhibiting SGC-7901 cells proliferation

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Bioorganic Chemistry, 2022, 126, 105853
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Antibacterial and antitumoral properties of 1,2,3-triazolo fused triterpenes and their mechanism of inhibiting the proliferation of HL-60 cells

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European Journal of Medicinal Chemistry, 2021, 224, 113727
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A One-Pot Procedure for the Synthesis of “Click-Ready” Triazoles from Ketones

Sampad Jana, Joice Thomas and Wim Dehaen

J. Org. Chem., 2016, 81, 12426
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Assembly of fully substituted triazolochromenes via a novel multicomponent reaction or mechanochemical synthesis

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The 1,2,3-triazole ring as a bioisostere in medicinal chemistry

Elisa Bonandi, Michael S. Christodoulou, Gaia Fumagalli, Dario Perdicchia, Giulio Rastelli and Daniele Passarella

Drug Discovery Today, 2017, 22, 1572
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Sequential Ugi reaction/base-induced ring closing/IAAC protocol toward triazolobenzodiazepine-fused diketopiperazines and hydantoins

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Beilstein J. Org. Chem., 2018, 14, 626
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The 1,2,3-triazole ‘all-in-one’ ring system in drug discovery: a good bioisostere, a good pharmacophore, a good linker, and a versatile synthetic tool

Deniz Lengerli, Kübra Ibis, Yahya Nural and Erden Banoglu

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Synthesis and Evaluation of Phenoxybenzylpiperidinyl Analogues as Agonists of the Chemokine Receptor CCR8

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Chemistry & Biodiversity, 2025, 22
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Copper-Catalyzed Oxidative Cross-Dehydrogenative Coupling/Oxidative Cycloaddition: Synthesis of 4-Acyl-1,2,3-Triazoles

Yi Liu, Gang Nie, Zhongzhen Zhou, Lihui Jia and Yunfeng Chen

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Multi‐Gram Scale Synthesis of 1,2,3‐Triazolium Ionic Liquids and Assay of Their Resistance towards Bases

Stijn Raiguel, Joice Thomas, Koen Binnemans and Wim Dehaen

Eur J Org Chem, 2018, 2018, 4850
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Transition‐Metal‐Free Annulation of Enamines and Tosyl Azide toward N‐Heterocycle Fused and 5‐Amino‐1,2,3‐Triazoles

Leiling Deng, Yunyun Liu, Yanping Zhu and Jie‐Ping Wan

Eur J Org Chem, 2020, 2020, 5606
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Small-molecule profiling for steroid receptor activity using a universal steroid receptor reporter assay

Roy Eerlings, Nana Barbakadze, Tien Nguyen, Nanuli Nadaraia, Elien Smeets, Lisa Moris, Florian Handle, Sarah El Kharraz, Wout Devlies, Arnout Voet, Wim Dehaen, Frank Claessens and Christine Helsen

The Journal of Steroid Biochemistry and Molecular Biology, 2022, 217, 106043
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DFT Studies on Mechanism of Organocatalytic Metal-Free Click 32CA Reaction for Synthesis of NH-1,2,3-triazoles

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Progress in the Synthesis of Fused 1,2,3‐Triazoles

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ChemistrySelect, 2021, 6, 4889
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Synthesis of Multisubstituted 1,2,3-Triazoles: Regioselective Formation and Reaction Mechanism

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Two-Step Synthesis of Fluorescent 3-Arylated 1,3a,6a-Triazapentalenes via a Three-Component Triazolization Reaction

Bram Verbelen and Wim Dehaen

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Recent Progress on Synthesis of Functionalized 1,5-Disubstituted Triazoles

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Metal‐Free Route for the Synthesis of 4‐Acyl‐1,2,3‐Triazoles from Readily Available Building Blocks

Joice Thomas, Vince Goyvaerts, Sandra Liekens and Wim Dehaen

Chemistry A European J, 2016, 22, 9966
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Betulonic Acid Derivatives Interfering with Human Coronavirus 229E Replication via the nsp15 Endoribonuclease

Annelies Stevaert, Besir Krasniqi, Benjamin Van Loy, Tien Nguyen, Joice Thomas, Julie Vandeput, Dirk Jochmans, Volker Thiel, Ronald Dijkman, Wim Dehaen, Arnout Voet and Lieve Naesens

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5-Formyltriazoles as Valuable Starting Materials for Unsymmetrically Substituted Bi-1,2,3-Triazoles

Robby Vroemans, Tomas Horsten, Maarten Van Espen and Wim Dehaen

Front. Chem., 2020, 8
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The potential of click reactions for the synthesis of bioactive triterpenes

René Csuk and Hans-Peter Deigner

Bioorganic & Medicinal Chemistry Letters, 2019, 29, 949
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On Water Cu@g‐C3N4 Catalyzed Synthesis of NH‐1,2,3‐Triazoles via [2+3] Cycloadditions of Nitroolefins/Alkynes and Sodium Azide

Soumen Payra, Arijit Saha and Subhash Banerjee

ChemCatChem, 2018, 10, 5468
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Organocatalyzed [3 + 2] cycloaddition reaction for regioselective synthesis of N-arylbenzotriazoles: theoretical study

Mohammad Abd Al-Hakim Badawi, Nabil Al-Bani, Raghad Ksaeby, Ali A. Khairbek, Abdullah Yahya Abdullah Alzahrani and Renjith Thomas