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Strategy and Effects of Polyproline Peptide Stapling by Copper(I)‐Catalyzed Alkyne–Azide Cycloaddition Reaction
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Residue‐Selective C−H Sulfenylation Enabled by Acid‐Activated S‐Acetamidomethyl Cysteine Sulfoxide with Application to One‐Pot Stapling and Lipidation Sequence
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Advancements in site-specific modification of peptides based on the chemical reactivity of native amino acids
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Functionalized Double Strain-Promoted Stapled Peptides for Inhibiting the p53-MDM2 Interaction
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Structural Characterization of Receptor–Receptor Interactions in the Allosteric Modulation of G Protein-Coupled Receptor (GPCR) Dimers
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Multicomponent Peptide Stapling as a Diversity‐Driven Tool for the Development of Inhibitors of Protein–Protein Interactions
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Peptide Stapling through Site-Directed Conjugation of Triazine Moieties to the Tyrosine Residues of a Peptide
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Development of a Single-Chain Peptide Agonist of the Relaxin-3 Receptor Using Hydrocarbon Stapling
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Dual In-Tether Chiral Centers Modulate Peptide Helicity
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Ligand‐Enabled Pd‐Catalyzed sp3 C−H Macrocyclization: Synthesis and Evaluation of Macrocyclic Sulfonamide for the Treatment of Parkinson's Disease
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Development of cell‐penetrating peptide‐based drug leads to inhibit MDMX:p53 and MDM2:p53 interactions
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Targeting the Genome‐Stability Hub Ctf4 by Stapled‐Peptide Design
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Development of a Multifunctional Benzophenone Linker for Peptide Stapling and Photoaffinity Labelling
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Targeting the ATG5-ATG16L1 Protein–Protein Interaction with a Hydrocarbon-Stapled Peptide Derived from ATG16L1 for Autophagy Inhibition
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An insight into piscidins: The discovery, modulation and bioactivity of greater amberjack, Seriola dumerili, piscidin
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