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Richa Goel, Vijay Luxami and Kamaldeep Paul

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Muscarine, imidazole, oxazole and thiazole alkaloids

Zhong Jin

Nat. Prod. Rep., 2016, 33, 1268
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Total synthesis and 13C NMR revision of nagelamide C

Guanghu Tong, Long V. Nguyen and Timothy F. Jamison

Org. Chem. Front., 2025
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Pyrrole carboxamide introduction in the total synthesis of pyrrole–imidazole alkaloids

Apsara K. Herath and Carl J. Lovely

Org. Biomol. Chem., 2021, 19, 2603
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Targeted suppression of oral squamous cell carcinoma by pyrimidine-tethered quinoxaline derivatives

Asmita Choithramani, Rudradip Das, Gourav Bothra, Priyanka Patel Vatsa, Venkatesh Muthukumar, Bombothu Kavya Sai Bhuvana, Saumya Kapoor, Deepshika Moola, Moumita Ghosh Chowdhury, Amit Mandoli and Amit Shard

RSC Med. Chem., 2024, 15, 2729
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Facile synthesis of 3-substituted imidazo[1,2-a]pyridines through formimidamide chemistry

Rasapalli Sivappa, Vamshikrishna Reddy Sammeta, Yanchang Huang, James A. Golen and Sergey N. Savinov

RSC Adv., 2019, 9, 29659
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Design, synthesis and activities of 4/5-acyl-2-aminoimidazolyl analogues of oroidin for biofilm inhibition

Sivappa Rasapalli, Abasaheb Dhawane, Christiaan Rees, James A. Golen, Bal Ram Singh, Shuowei Cai, Jerry Jasinski, Steven M. Kwasny, Donald T. Moir, Timothy J. Opperman and Terry L. Bowlin

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An aza-Robinson Annulation Strategy for the Synthesis of Fused Bicyclic Amides: Synthesis of (±)-Coniceine and Quinolizidine

Alexander Garay-Talero, Tales A. C. Goulart, Rafael D. C. Gallo, Roberto do C. Pinheiro, Catalina Hoyos-Orozco, Igor D. Jurberg and Diego Gamba-Sánchez

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Heterosubstituted 4-Vinylimidazoles – Preparation and Diels-Alder Reactions

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HETEROCYCLES, 2019, 99, 324
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The Dimroth rearrangement as a probable cause for structural misassignments in imidazo[1,2-a]pyrimidines: A N-labelling study and an easy method for the determination of regiochemistry

Maria Chatzopoulou, R. Fernando Martínez, Nicky J. Willis, Timothy D.W. Claridge, Francis X. Wilson, Graham M. Wynne, Stephen G. Davies and Angela J. Russell

Tetrahedron, 2018, 74, 5280
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Total Synthesis of (±)-Sceptrin

Long V. Nguyen and Timothy F. Jamison

Org. Lett., 2020, 22, 6698
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Synthesis and anticancer activity of focused compound libraries from the natural product lead, oroidin

Lauren Dyson, Anthony D. Wright, Kelly A. Young, Jennette A. Sakoff and Adam McCluskey

Bioorganic & Medicinal Chemistry, 2014, 22, 1690
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Activating Imides with Triflic Acid: A General Intramolecular Aldol Condensation Strategy Toward Indolizidine, Quinolizidine, and Valmerin Alkaloids

Yovanny Quevedo-Acosta, Igor D. Jurberg and Diego Gamba-Sánchez

Org. Lett., 2020, 22, 239
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Toward the Synthesis of Sceptrin and Benzosceptrin: Solvent Effect in Stereo‐ and Regioselective [2+2] Photodimerization and Easy Access to the Fully Substituted Benzobutane

Thanh Binh Nguyen, Le Anh Nguyen, Mathilde Corbin, Pascal Retailleau, Ludmila Ermolenko and Ali Al‐Mourabit

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Substrate Controlled Regioselective Bromination of Acylated Pyrroles Using Tetrabutylammonium Tribromide (TBABr3)

Shuang Gao, Travis K. Bethel, Tayeb Kakeshpour, Grace E. Hubbell, James E. Jackson and Jetze J. Tepe

J. Org. Chem., 2018, 83, 9250
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Towards unbiased and more versatile NMR‐based structure elucidation: A powerful combination of CASE algorithms and DFT calculations

Alexei V. Buevich and Mikhail E. Elyashberg

Magnetic Reson in Chemistry, 2018, 56, 493
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Recent Advances in the Synthesis of Imidazo[1,2‐a]pyridines: A Brief Review

Jasmine Panda, Bishnu P. Raiguru, Mitali Mishra, Seetaram Mohapatra and Sabita Nayak

ChemistrySelect, 2022, 7
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Synthesis and biological evaluation of piperazine derivatives as novel isoform selective voltage-gated sodium (Nav) 1.3 channel modulators

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A Direct Route into Fused Imidazo-diazines and Imidazo-pyridines Using Nucleophilic Nitrenoids in a Gold-Catalyzed Formal [3 + 2]-Dipolar Cycloaddition

Miguel Garzón and Paul W. Davies

Org. Lett., 2014, 16, 4850
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ChemInform Abstract: Total Syntheses of Oroidin (Ia), Hymenidin (Ib) and Clathrodin (Ic).

Sivappa Rasapalli, Venkatreddy Kumbam, Abasaheb N. Dhawane, James A. Golen, Carl J. Lovely and Arnold L. Rheingold

ChemInform, 2013, 44
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Hypervalent Iodine(III) Promoted Direct Synthesis of Imidazo[1,2‐a]pyrimidines

Guangyin Qian, Bingxin Liu, Qitao Tan, Siwen Zhang and Bin Xu

Eur J Org Chem, 2014, 2014, 4837
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Expanding the Cyclopentadienyl Framework: 99mTc/Re Complexes with Orthogonal Functions for Bioconjugation

Raphael Lengacher, Joshua Csucker, Daniel Hernández-Valdés, Bernhard Spingler, Henrik Braband and Roger Alberto

Bioconjugate Chem., 2021, 32, 1393
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Novel imidazopyrimidines-based molecules induce tetramerization of tumor pyruvate kinase M2 and exhibit potent antiproliferative profile

Sagarkumar Patel, Christoph Globisch, Priyanka Pulugu, Prasoon Kumar, Alok Jain and Amit Shard

European Journal of Pharmaceutical Sciences, 2022, 170, 106112
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A convenient strategy for synthesizing the Agelas alkaloids clathrodin, oroidin, and hymenidin and their (un)saturated linker analogs

Aleš Žula, Danijel Kikelj and Janez Ilaš

Tetrahedron Letters, 2014, 55, 3999
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An Updated Review on the Synthesis and Antibacterial Activity of Molecular Hybrids and Conjugates Bearing Imidazole Moiety

Renzo Rossi and Maurizio Ciofalo

Molecules, 2020, 25, 5133
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Draining the moat: disrupting bacterial biofilms with natural products

Madison H. Fletcher, Megan C. Jennings and William M. Wuest

Tetrahedron, 2014, 70, 6373
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Elements as Direct Feedstocks for Organic Synthesis: Fe/I2/O2 for Diamination of 2-Cyclohexenones with 2-Aminopyrimidine and 2-Aminopyridines

Thanh Binh Nguyen, Mathilde Corbin, Pascal Retailleau, Ludmila Ermolenko and Ali Al-Mourabit

Org. Lett., 2015, 17, 4956
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Total Synthesis of Nagelamide W

Dare E. George and Jetze J. Tepe

J. Org. Chem., 2023, 88, 9306
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