Diana V. Aleksanyan, Svetlana G. Churusova, Valentina V. Brunova, Alexander S. Peregudov, Aleksander M. Shakhov, Ekaterina Yu. Rybalkina, Zinaida S. Klemenkova, Elena G. Kononova, Gleb L. Denisov and Vladimir A. Kozlov

Dalton Trans., 2021, 50, 16726
DOI: 10.1039/D1DT03259C

Isocyanates and isothiocyanates as versatile platforms for accessing (thio)amide-type compounds

Vittorio Pace, Serena Monticelli, Karen de la Vega-Hernández and Laura Castoldi

Org. Biomol. Chem., 2016, 14, 7848
DOI: 10.1039/C6OB00766J

NH4I-promoted oxidative formation of benzothiazoles and thiazoles from arylacetic acids and phenylalanines with elemental sulfur

Yujia Xia, Huawen Huang, Wei Hu and Guo-Jun Deng

Org. Biomol. Chem., 2021, 19, 5108
DOI: 10.1039/D1OB00671A

Unprecedented amidation of ‘transient’ aryl thioaldehydes by N,N-dimethylformamide under basic conditions

Basudeb Basu and Samir Kundu

New J. Chem., 2014, 38, 3367
DOI: 10.1039/C4NJ00480A

One‐Pot Synthesis of Thioamides via Nickel‐Catalyzed Coupling of Thiocarbamoyl Fluorides and Boronic Acids

Yasir Mumtaz, Haonan Xiang, Jahangir Khan, Shuaishuai Liang and Wenbin Yi

Eur J Org Chem, 2024, 27
DOI: 10.1002/ejoc.202400742

Visible light-induced catalytic syntheses of thioamides as biomass-based corrosion inhibitors for mild steel

Junda Chen and Jinzhu Chen

Journal of Catalysis, 2025, 448, 116180
DOI: 10.1016/j.jcat.2025.116180

Thioamidation of Arylpropyne Derivatives with Sulfur and Formamides for the Synthesis of Aryl Propanethioamides

Hong‐Hui Xu, Xing‐Guo Zhang and Xiao‐Hong Zhang

Asian J Org Chem, 2020, 9, 111
DOI: 10.1002/ajoc.201900680

Design and Synthesis of 5‐Morpholino‐Thiophene‐Indole/ Oxindole Hybrids as Cytotoxic Agents

Upasana Yadav, Akash P. Sakla, Ramya Tokala, Sai Teja Nyalam, Amit Khurana, Chander Singh Digwal, Venu Talla, Chandraiah Godugu, Nagula Shankaraiah and Ahmed Kamal

ChemistrySelect, 2020, 5, 4356
DOI: 10.1002/slct.201904845

Catalyst‐ and Solvent‐Free Thioamidation of Aromatic Aldehydes through a Willgerodt‐Kindler Reaction

Arun D. Kale and Dipak S. Dalal

ChemistrySelect, 2022, 7
DOI: 10.1002/slct.202203497

Ammonium Salts as Convenient Ammonia Surrogates in the Willgerodt Reaction

E. A. Kvetkin and A. V. Sokolov

Russ J Org Chem, 2025, 61, 561
DOI: 10.1134/S1070428024603273

Direct Synthesis of α-Ketothioamide Derivatives through a One-Pot Reaction of Sulfur Ylides, Nitrosobenzenes, and Thioacetic Acid

Chaowei Xiang, Fang Luo, Zheng Wang, Yunlong Pan, Yu Liu, Linghui Zeng, Chong Zhang, Huajian Zhu, Jiankang Zhang and Jiaan Shao

J. Org. Chem., 2024, 89, 8878
DOI: 10.1021/acs.joc.4c00738

Recent Advances in the Synthesis of Ibuprofen and Naproxen

Min-Woo Ha and Seung-Mann Paek

Molecules, 2021, 26, 4792
DOI: 10.3390/molecules26164792

Enzymatic Thioamide Formation in a Bacterial Antimetabolite Pathway

Agnieszka Litomska, Keishi Ishida, Kyle L. Dunbar, Marco Boettger, Sébastien Coyne and Christian Hertweck

Angewandte Chemie, 2018, 130, 11748
DOI: 10.1002/ange.201804158

Design, synthesis and computational study of new benzofuran hybrids as dual PI3K/VEGFR2 inhibitors targeting cancer

Omar A. El-Khouly, Morkos A. Henen, Magda A.-A. El-Sayed and Shahenda M. El-Messery

Sci Rep, 2022, 12
DOI: 10.1038/s41598-022-21277-2

Study on the synthesis of thioamides from aldehyde N-tert-butylsulfinyl amide and sulfur in aqueous media

Pham Xuan Thao, Tuan and Thuong

J. Mil. Sci. Technol., 2021, 54
DOI: 10.54939/1859-1043.j.mst.76.2021.54-60

Access to 2-Aroylthienothiazoles via C–H/N–O Bond Functionalization of Oximes

Peiqi Zhou, Yubing Huang, Wanqing Wu, Jiaming Zhou, Wentao Yu and Huanfeng Jiang

Org. Lett., 2019, 21, 9976
DOI: 10.1021/acs.orglett.9b03900

Multicomponent Assembly of 1,2,3-Dithiazole-5-thiones via Triple Sulfur Donor Integration

Penghui Ni, Jing Tan, Yuxing Tan, Wujiu Jiang and Guo-Jun Deng

Org. Lett., 2025, 27, 10809
DOI: 10.1021/acs.orglett.5c03433

Tetracoordinate Boron Intermediates Enable Unconventional Transformations

Kai Yang and Qiuling Song

Acc. Chem. Res., 2021, 54, 2298
DOI: 10.1021/acs.accounts.1c00132

Europhtal: An industrial cobalt phthalocyanine complex as the efficient catalyst for synthesis of thioamides by one‐pot reaction of mercaptans and amines

Nasser Zarinderakht, Mohammad Abbasi and Najmeh Nowrouzi

Applied Organom Chemis, 2022, 36
DOI: 10.1002/aoc.6709

Towards More Practical Methods for the Chemical Synthesis of Thioamides Using Sulfuration Agents: A Decade Update

Qiang Zhang, Laurent Soulère and Yves Queneau

Molecules, 2023, 28, 3527
DOI: 10.3390/molecules28083527

Recent Advances in Multicomponent Reactions with Organic and Inorganic Sulfur Compounds

Qinqin Tang, Xianjie Yin, Ratnakar Reddy Kuchukulla and Qingle Zeng

The Chemical Record, 2021, 21, 893
DOI: 10.1002/tcr.202100026

Copper‐catalyzed synthesis of α‐ketothioamides from ketones

Fatemeh Abdollahi and Arash Ghaderi

J Chinese Chemical Soc, 2023, 70, 949
DOI: 10.1002/jccs.202200520

Sulfur promoted decarboxylative thioamidation of carboxylic acids using formamides as amine proxy

Saurabh Kumar, Rajeshwer Vanjari, Tirumaleswararao Guntreddi and Krishna Nand Singh

Tetrahedron, 2016, 72, 2012
DOI: 10.1016/j.tet.2016.02.070

Synthesis of Phosphoryl Thioamides via Three‐Component Reaction of Phosphinic Chlorides with Amines and Sulfur

Mikhail Kozlov, Andrey Kozlov, Alexander Komkov, Konstantin Lyssenko, Igor Zavarzin and Yulia Volkova

Adv Synth Catal, 2019, 361, 2904
DOI: 10.1002/adsc.201900067

Elemental Sulfur in the Synthesis of Organic Compounds (An Update 2019–2025)

Anatoly Y. Chursin, Igor V. Zavarzin and Yulia A. Volkova

Adv Synth Catal, 2026, 368
DOI: 10.1002/adsc.70152

Elemental Sulfur/Base/Water: An Efficient System for the Synthesis of 2-Phosphoryl-Substituted Benzazoles via a Willgerodt-Kindler-Type Reaction

Anatoly Y. Chursin, Konstantin M. Bolshakov, Konstantin A. Lyssenko, Igor V. Zavarzin and Yulia A. Volkova

J. Org. Chem., 2026, 91, 4882
DOI: 10.1021/acs.joc.5c02758

Upcycled Composite Derived from Polyacrylonitrile and Elemental Sulfur: Thermomechanical Properties and Microstructural Insight

Shalini K. Wijeyatunga and Rhett C. Smith

Sustainability, 2025, 17, 3702
DOI: 10.3390/su17083702

Nucleophilic activation of the sulfur S8 cyclic form as a green chemistry tool

N. P. Tarasova, E. G. Krivoborodov and Ya. O. Mezhuev

Russ Chem Bull, 2023, 72, 415
DOI: 10.1007/s11172-023-3809-9

Non-Isocyanide-Based Three-Component Reactions: From Strecker to Nowadays

Ivette Morales-Salazar, Jean-Philippe Bouillon, Eduardo González-Zamora and Alejandro Islas-Jácome

J. Mex. Chem. Soc., 2025, 69, 185
DOI: 10.29356/jmcs.v69i1.2301

Elemental Sulfur-Promoted Oxidative Rearranging Coupling between o-Aminophenols and Ketones: A Synthesis of 2-Alkyl benzoxazoles under Mild Conditions

Thanh Binh Nguyen and Pascal Retailleau

Org. Lett., 2017, 19, 3887
DOI: 10.1021/acs.orglett.7b01775

Synthesis of Benzothiazole‐ and Benzoxazole‐2‐carboxamides by 2‐Chloracetamides and 2‐Amino(thio)phenols Cyclocondensation with Elemental Sulfur in Water

Mikhail A. Kozlov, Konstantin M. Bolshakov, Natalia G. Kolotyrkina and Igor V. Zavarzin

Eur J Org Chem, 2022, 2022
DOI: 10.1002/ejoc.202200586

One‐Pot Synthesis of Ferrocene Thioamides from Ferrocenecarboxaldehyde via the Willgerodt–Kindler Reaction

Henrich Kabzan, Péter Kisszékelyi, Juraj Filo, Marek Cigáň, Erik Rakovský and Radovan Šebesta

Eur J Org Chem, 2025, 28
DOI: 10.1002/ejoc.202500956

Construction of Thioamide Peptides from Chiral Amino Acids

Yanyan Liao, Shunmin Zhang and Xuefeng Jiang

Angew Chem Int Ed, 2023, 62
DOI: 10.1002/anie.202303625

Chemoselective Thioacylation of Amines Enabled by Synergistic Defluorinative Coupling

Yuqi Li, Tongxiang Cao, Rongbin Peng, Shang Zhou, Xujing Long, Huanfeng Jiang and Chuanle Zhu

Org. Lett., 2024, 26, 6438
DOI: 10.1021/acs.orglett.4c02237

S8‐Mediated One‐Pot Synthesis of Thioamides from Benzyl Chlorides and Amines

Xiaotong Li, Qiang Pan, Renhe Hu, Xin Wang, Zhao Yang and Shiqing Han

Asian J Org Chem, 2016, 5, 1353
DOI: 10.1002/ajoc.201600385

Ohne Licht und ohne Hitze? Bei Raumtemperatur hergestellte Schwefelpolymere sind spitze!

Lirong He, Hui Zhao and Patrick Theato

Angewandte Chemie, 2018, 130, 13194
DOI: 10.1002/ange.201807005

C2-Transformation of calcium carbide trigered by hydrogen sulfide

Yunzhe Du, Siliu Cheng, Shuyi Li, Junping Niu, Yuan Gou, Ligang Yan, Tian-Xing Zhang, Ruijun Xie, Limin Han, Tiezheng Jia and Ning Zhu

Chinese Chemical Letters, 2025, 36, 111233
DOI: 10.1016/j.cclet.2025.111233

A multipathway coupled domino strategy: I2-mediated oxidative thionation for direct synthesis of thiobenzamides from miscellaneous substrates

Hong-Zheng Li, Wei-Jian Xue, Guo-Dong Yin and An-Xin Wu

Tetrahedron Letters, 2015, 56, 5843
DOI: 10.1016/j.tetlet.2015.08.060

Visible‐Light‐Driven Multicomponent Reactions for the Versatile Synthesis of Thioamides by Radical Thiocarbamoylation

Hong‐Mei Guo, Jia‐Jin Wang, Yanjiao Xiong and Xuesong Wu

Angew Chem Int Ed, 2024, 63
DOI: 10.1002/anie.202409605

Dehydrative Beckmann rearrangement and the following cascade reactions

Yongjiao Wei, Yinghui Liu and Lan-Gui Xie

Chinese Chemical Letters, 2022, 33, 2407
DOI: 10.1016/j.cclet.2021.10.020

The Electrogenerated Cyanomethyl Anion: An Old Base Still Smart

Isabella Chiarotto, Leonardo Mattiello and Marta Feroci

Acc. Chem. Res., 2019, 52, 3297
DOI: 10.1021/acs.accounts.9b00465

Copper‐Catalyzed Decarboxylative Synthesis of α‐Ketothioamides Using α,β‐Unsaturated Arylcarboxylic Acids, Alicyclic Secondary Amines and Elemental Sulfur

Anjali Jaiswal, Anup Kumar Sharma, Preeti and Krishna Nand Singh

Asian J Org Chem, 2021, 10, 1748
DOI: 10.1002/ajoc.202100203

Glycerol‐K2CO3 Deep Eutectic Solvent as Environmentally Friendly Media with Basic and Dehumidifier Synergistic Effect for Running of Willgerodt‐Kindler Reaction

Iman Radfar, Sepideh Abbasi, Maryam Kazemi Miraki, Elahe Yazdani, Meghdad Karimi and Akbar Heydari

ChemistrySelect, 2018, 3, 3265
DOI: 10.1002/slct.201702906

Dimethylamine as the key intermediate generated in situ from dimethylformamide (DMF) for the synthesis of thioamides

Weibing Liu, Cui Chen and Hailing Liu

Beilstein J. Org. Chem., 2015, 11, 1721
DOI: 10.3762/bjoc.11.187

MWCNTs/MNPs-adenine-CuI in choline chloride-urea: a sustainable and efficient catalytic system for preparation of thioamides through Willgerodt-Kindler reaction

Reza Mohammadi, Ghada Al Assi, M M Rekha, Shaker Al-Hasnaawei, Subhashree Ray, Amrita Pal and Renu Sharma

Journal of Molecular Structure, 2026, 1351, 144195
DOI: 10.1016/j.molstruc.2025.144195

Thioamide construction via sulfur interrupted Brook rearrangement

Shunmin Zhang, Yanyan Liao and Xuefeng Jiang

Green Synthesis and Catalysis, 2025, 6, 192
DOI: 10.1016/j.gresc.2024.02.006

Three-Component Cascade Bis-heteroannulation of Aryl or Vinyl Methylketoxime Acetates toward Thieno[3,2-c]isoquinolines

Zhenhua Xu, Guo-Jun Deng, Feng Zhang, Hongbiao Chen and Huawen Huang

Org. Lett., 2019, 21, 8630
DOI: 10.1021/acs.orglett.9b03241

Willgerodt‐Kindler Reaction of Benzaldehydes: A Comparative Study for a Sustainable Synthesis of Secondary Thiobenzamides

Maria Papa, Isabella Chiarotto and Marta Feroci

ChemistrySelect, 2017, 2, 3207
DOI: 10.1002/slct.201700507

Green Chemistry in the Synthesis of Pharmaceuticals

Supratik Kar, Hans Sanderson, Kunal Roy, Emilio Benfenati and Jerzy Leszczynski

Chem. Rev., 2022, 122, 3637
DOI: 10.1021/acs.chemrev.1c00631

Multicomponent reactions in crop protection chemistry

Clemens Lamberth

Bioorganic & Medicinal Chemistry, 2020, 28, 115471
DOI: 10.1016/j.bmc.2020.115471

Sulfur Chemistry in Polymer and Materials Science

Hatice Mutlu, Ezgi Berfin Ceper, Xiaohui Li, Jingmei Yang, Wenyuan Dong, Mehmet Murat Ozmen and Patrick Theato

Macromol. Rapid Commun., 2019, 40
DOI: 10.1002/marc.201800650

Mild and Chemoselective Thioacylation of Amines Enabled by the Nucleophilic Activation of Elemental Sulfur

Masato Saito, Sho Murakami, Takeshi Nanjo, Yusuke Kobayashi and Yoshiji Takemoto

J. Am. Chem. Soc., 2020, 142, 8130
DOI: 10.1021/jacs.0c03256

Mechanistic and experimental study on copper-catalyzed C3-sulfenylation of indoles with sulfur powder and aryl iodides

Xin Ge, Lin Cheng, Fengli Sun, Xuemin Liu, Xinzhi Chen, Chao Qian and Shaodong Zhou

Catalysis Communications, 2019, 123, 32
DOI: 10.1016/j.catcom.2019.01.015

A facile access to thieno[2,3-b]indoles via sulfur-mediated decarboxylative cyclization of α, β-unsaturated carboxylic acids with indoles

Hao-Lin Zhang, Fei Wen, Wen-Bing Sheng, Peng Yin, Chun-Tao Zhang, Cai-Yun Peng, Dong-Ming Peng, Duan-Fang Liao and Rong-Geng Fu

Tetrahedron Letters, 2019, 60, 80
DOI: 10.1016/j.tetlet.2018.11.062

Electronic structure and tautomerism of thioamides

Igor Novak, Leo Klasinc and Sean P. McGlynn

Journal of Electron Spectroscopy and Related Phenomena, 2016, 209, 62
DOI: 10.1016/j.elspec.2016.03.005

Visible‐Light‐Promoted Willgerodt–Kindler‐Type Thioamidation Reaction of Amines, α‐Ketoacids, and Elemental Sulfur

Jigang Gao, Taimin Wang, Peng Li, Yun Luo, Lijing Fang, Hongbin Zhai, Jinlin Wang and Bin Cheng

Eur J Org Chem, 2025, 28
DOI: 10.1002/ejoc.202500708

Synthesis of 2‐Nitrothiophenes via Tandem Henry Reaction and Nucleophilic Substitution on Sulfur from β‐Thiocyanatopropenals

Lin Rong, Yingxia Shen, Guoxi Xiong and Yuefa Gong

Journal of Heterocyclic Chem, 2019, 56, 670
DOI: 10.1002/jhet.3446

Thioamidation via Sulfur-Promoted Coupling of N-Methyliminodiacetyl Acylborons and Amines

Hao Yang, Yanyan Liao and Xuefeng Jiang

J. Org. Chem., 2026, 91, 428
DOI: 10.1021/acs.joc.5c02513

A straightforward route to alkyl 5‐arylthiophene‐2‐thiocarboxylates from alkyl 2‐aroyl‐1‐chlorocyclopropanecarboxylates

Long Huang, Xuehui Liu, Duntie Zhang, Chenghao Luo, Jing Zhang, Yikun Chen and Yuefa Gong

Journal of Heterocyclic Chem, 2021, 58, 882
DOI: 10.1002/jhet.4225

A Robust, Eco‐Friendly Access to Secondary Thioamides through the Addition of Organolithium Reagents to Isothiocyanates in Cyclopentyl Methyl Ether (CPME)

Vittorio Pace, Laura Castoldi, Serena Monticelli, Sandra Safranek, Alexander Roller, Thierry Langer and Wolfgang Holzer

Chemistry A European J, 2015, 21, 18966
DOI: 10.1002/chem.201504247

Nickel-Catalyzed Coupling Reaction of Arylboronic Acid with Methyl Dithiocarbamates for the Synthesis of Thioamides

Jinsong Hou, Lirong Han and Qinghan Li

LOC, 2025, 22, 973
DOI: 10.2174/0115701786318561250619115451

Thiol as a Synthon for Preparing Thiocarbonyl: Aerobic Oxidation of Thiols for the Synthesis of Thioamides

Xi Wang, Miran Ji, Seungyeon Lim and Hye-Young Jang

J. Org. Chem., 2014, 79, 7256
DOI: 10.1021/jo501378v

Selective Construction of 2-Substituted Benzothiazoles from o-Iodoaniline Derivatives S8 and N-Tosylhydrazones

Yubing Huang, Peiqi Zhou, Wanqing Wu and Huanfeng Jiang

J. Org. Chem., 2018, 83, 2460
DOI: 10.1021/acs.joc.7b03118

Construction of Thioamide Peptides from Chiral Amino Acids

Yanyan Liao, Shunmin Zhang and Xuefeng Jiang

Angewandte Chemie, 2023, 135
DOI: 10.1002/ange.202303625

Multicomponent Polymerization of Sulfur, Diynes, and Aromatic Diamines and Facile Tuning of Polymer Backbone Structures

Yuzhang Huang, Rongrong Hu and Ben Zhong Tang

Macromolecules, 2024, 57, 6568
DOI: 10.1021/acs.macromol.4c00879

Elemental Sulfur‐Promoted Aerobic Cyclization of Ketones and Aliphatic Amines for Synthesis of Tetrasubstituted Imidazoles

Xiangui Chen, Zhen Wang, Huawen Huang and Guo‐Jun Deng

Adv Synth Catal, 2018, 360, 4017
DOI: 10.1002/adsc.201800765

Organoselenium Compounds: Chemistry and Applications in Organic Synthesis

Juan M. Sonego, Sheila I. de Diego, Sergio H. Szajnman, Carola Gallo‐Rodriguez and Juan B. Rodriguez

Chemistry A European J, 2023, 29
DOI: 10.1002/chem.202300030

Aqueous Compatible Protocol to Both Alkyl and Aryl Thioamide Synthesis

Jianpeng Wei, Yiming Li and Xuefeng Jiang

Org. Lett., 2016, 18, 340
DOI: 10.1021/acs.orglett.5b03541

Synthesis of Thioamides by Catalyst‐Free Three‐Component Reactions in Water

Hualong Xu, Hang Deng, Zhengkai Li, Haifeng Xiang and Xiangge Zhou

Eur J Org Chem, 2013, 2013, 7054
DOI: 10.1002/ejoc.201301148

No Heat, No Light—The Future of Sulfur Polymers Prepared at Room Temperature Is Bright

Lirong He, Hui Zhao and Patrick Theato

Angew Chem Int Ed, 2018, 57, 13012
DOI: 10.1002/anie.201807005

Reactivities and mechanisms in organic reactions involving activation of elemental sulfur under basic conditions

Peter Conen and Michael A.R. Meier

Tetrahedron Chem, 2024, 11, 100086
DOI: 10.1016/j.tchem.2024.100086

Metal-Free Dehydrogenative Double C–H Sulfuration To Access Thieno[2,3-b]indoles Using Elemental Sulfur

Jianming Liu, Yanyan Zhang, Yuanyuan Yue, Zhixian Wang, Huibin Shao, Kelei Zhuo, Qingzhang Lv and Zhiguo Zhang

J. Org. Chem., 2019, 84, 12946
DOI: 10.1021/acs.joc.9b01586

Multicomponent Tandem Cyclization/Aromatization Reaction: Access to 2‐Substituted Naphthothiazoles and Benzothiazoles

Upendra Kumar, Ajay Sharma, Trayambek Nath Chaubey and Satyendra Kumar Pandey

Eur J Org Chem, 2024, 27
DOI: 10.1002/ejoc.202400449

Mild and green thioacylation with dithiocarboxylates via photoredox catalysis

Wen-Chao Gao, Wei Li, Juan Zhang, Hong-Hong Chang and Rong Zhou

Green Synthesis and Catalysis, 2026, 7, 69
DOI: 10.1016/j.gresc.2024.02.008

Elemental-Sulfur-Incorporated Cyclizations of Pyrrolidines Leading to Thienopyrroles

Yuanyuan Yue, Huibin Shao, Zhixian Wang, Ke Wang, Le Wang, Kelei Zhuo and Jianming Liu

J. Org. Chem., 2020, 85, 11265
DOI: 10.1021/acs.joc.0c01363

Direct synthesis of α-ketothioamides from aryl methyl ketones and amines via I2-promoted sp3 C–H functionalization

Hong-Zheng Li, Wei-Jian Xue and An-Xin Wu

Tetrahedron, 2014, 70, 4645
DOI: 10.1016/j.tet.2014.05.045

Direct Transamidation of Thioamides with Amines via Acetophenone-Promoted Enamine Catalysis under Metal-Free Conditions

Yuxing Tan, Penghui Ni, Wu-jiu Jiang, Yang Fu and Qiuping Ding

J. Org. Chem., 2024, 89, 2939
DOI: 10.1021/acs.joc.3c02352

Decarboxylative Thioamidation of Arylacetic and Cinnamic Acids: A New Approach to Thioamides

Tirumaleswararao Guntreddi, Rajeshwer Vanjari and Krishna Nand Singh

Org. Lett., 2014, 16, 3624
DOI: 10.1021/ol501482g

Enantioselective Synthesis of Thiazole‐Derived α‐Perfluoroalkylated 5–7‐Membered Amines

Natalia G. Voznesenskaia, Olga I. Shmatova, Mikhail M. Ilyin, Mikhail M. Ilyin and Valentine G. Nenajdenko

Eur J Org Chem, 2019, 2019, 1893
DOI: 10.1002/ejoc.201801845

Synthesis of 2-carboxamide-substituted benzimidazoles via S8-promoted multicomponent reaction in aqueous media

Valentina Birukova, Anatoly Y. Chursin, Igor V. Zavarzin and Yulia A. Volkova

Tetrahedron, 2026, 193, 135130
DOI: 10.1016/j.tet.2025.135130

Synthesis of copper(i) chelates based on heterocyclic thioamides

Anatoliy Ranskiy, Natalia Didenko, Оlga Gordienko and Таras Тіtov

ChChT, 2025, 19, 628
DOI: 10.23939/chcht19.04.628

General Construction of Thioamides under Mild Conditions: A Stepwise Proton Transfer Process Mediated by EDTA

Hao Jin, Xin Ge and Shaodong Zhou

Eur J Org Chem, 2021, 2021, 6015
DOI: 10.1002/ejoc.202101013

2‐Benzoyl Thienothiazoles from Annulation of C−H Bonds in Acetophenone Oximes

Phuc H. Pham, Khang X. Nguyen, Ninh P. Nguyen, Hoai T. B. Pham, Tung T. Nguyen and Nam T. S. Phan

Asian J Org Chem, 2020, 9, 622
DOI: 10.1002/ajoc.202000046

Csp3–H Bond Functionalization of α-Bromo Ketones for the Synthesis of α-Keto Thioamides Using Elemental Sulfur

Haiying Tian, Fang Guo and Xiuling Chen

Russ J Org Chem, 2022, 58, 1260
DOI: 10.1134/S107042802209010X

Elemental‐Sulfur‐Promoted C(sp3)−H Activation of Methyl Heteroarenes Leading to Thioamides

Jianming Liu, Shanshan Zhao, Xuyang Yan, Yanyan Zhang, Shufang Zhao, Kelei Zhuo and Yuanyuan Yue

Asian J Org Chem, 2017, 6, 1764
DOI: 10.1002/ajoc.201700532

Catalyzing the Ring-Opening Polymerization of 1,3-Benzoxazines via Thioamide from Renewable Sources

Zehra Gul Coban, Yusuf Yagci and Baris Kiskan

ACS Appl. Polym. Mater., 2021, 3, 4203
DOI: 10.1021/acsapm.1c00637

2-Oxo-triterpenoids of ursane, oleanane and dammarane types and their α-glucosidase inhibitory properties

Liana Zakirova, Alexander Poptsov, Oxana Kazakova, Irina Smirnova, Yury Gatilov, Dmitriy Polovyanenko, Irina Bagryanskaya, Denis Babkov, Roman Danilov and Andrey Lukyanov

Natural Product Research, 2025, 1
DOI: 10.1080/14786419.2025.2565286

Surface-modified magnetic biochar: Highly efficient adsorbents for removal of Pb(ΙΙ) and Cd(ΙΙ)

Mahboobeh Zahedifar, Neda Seyedi, Saeid Shafiei and Moslem Basij

Materials Chemistry and Physics, 2021, 271, 124860
DOI: 10.1016/j.matchemphys.2021.124860

Efficient synthesis of N b -thioacyltryptamine derivatives by a three-component Willgerodt–Kindler reaction, and their transformation to 1-substituted-3,4-dihydro-β-carbolines

Mátyás Milen, Péter Slégel, Péter Keglevich, György Keglevich, Gyula Simig and Balázs Volk

Tetrahedron Letters, 2015, 56, 5697
DOI: 10.1016/j.tetlet.2015.09.007

Elemental Sulfur and Molecular Iodine as Efficient Tools for Carbon‐Nitrogen Bond Formation through Redox Reactions

Thanh Binh Nguyen

Asian J Org Chem, 2017, 6, 477
DOI: 10.1002/ajoc.201700011

Peculiar Features of the Willgerodt–Kindler Reaction of 1-Adamantylpropan-2-one and Its Derivatives

I. A. Novakov, B. S. Orlinson, E. N. Savel’ev, E. A. Potaenkova, O. V. Vostrikova, D. P. Tarakanov and M. A. Nakhod

Russ J Gen Chem, 2017, 87, 2762
DOI: 10.1134/S1070363217120027

Visible‐Light‐Driven Multicomponent Reactions for the Versatile Synthesis of Thioamides by Radical Thiocarbamoylation

Hong‐Mei Guo, Jia‐Jin Wang, Yanjiao Xiong and Xuesong Wu

Angewandte Chemie, 2024, 136
DOI: 10.1002/ange.202409605

Tri‐Functional Elemental Sulfur Enabling Bis‐Heteroannulation of Methyl Ketoximes with Methyl N‐Heteroarenes

Huawen Huang, Qian Wang, Zhenhua Xu and Guo‐Jun Deng

Adv Synth Catal, 2019, 361, 591
DOI: 10.1002/adsc.201801324

Contemporary Applications of Thioamides and Methods for Their Synthesis

Tobias N. Hansen and Christian A. Olsen

Chemistry A European J, 2024, 30
DOI: 10.1002/chem.202303770

An Efficient Heterobimetallic Lanthanide Alkoxide Catalyst for Transamidation of Amides under Solvent‐Free Conditions

Hongting Sheng, Ruijie Zeng, Wenjuan Wang, Shuwen Luo, Yan Feng, Jing Liu, Weijian Chen, Manzhou Zhu and Qingxiang Guo

Adv Synth Catal, 2017, 359, 302
DOI: 10.1002/adsc.201600373

Efficient Three-Component Tandem Reaction for Synthesizing Thioamide Derivatives via the Ring Opening Reaction of Cyclic Amidines with Aldehydes Promoted by H2S

Yunzhe Du, Shuyi Li, Siliu Cheng, Huijie Jia, Zheng Wang, Limin Han and Ning Zhu

Acta Chimica Sinica, 2026, 84, 93
DOI: 10.6023/A25060234

Multicomponent polymerization of sulfur, chloroform and diamine toward polythiourea

Nan Zheng, He Gao, Zihui Jiang and Wangze Song

Sci. China Chem., 2023
DOI: 10.1007/s11426-022-1483-8

Enzymatic Thioamide Formation in a Bacterial Antimetabolite Pathway

Agnieszka Litomska, Keishi Ishida, Kyle L. Dunbar, Marco Boettger, Sébastien Coyne and Christian Hertweck

Angew Chem Int Ed, 2018, 57, 11574
DOI: 10.1002/anie.201804158

Synthesis of Dibenzo[d,f][1,3]Diazepines via Elemental Sulfur-Mediated Cyclocondensation of 2,2′-Biphenyldiamines with 2-Chloroacetic Acid Derivatives

Tatyana A. Tikhonova, Konstantin A. Lyssenko, Igor V. Zavarzin and Yulia A. Volkova

J. Org. Chem., 2019, 84, 15817
DOI: 10.1021/acs.joc.9b02002

Elemental Sulfur‐Promoted [2+3+1] Annulation for Synthesis of Functionalized Thiochromeno[2,3‐b]indoles from Indole Derivatives

Jianming Liu, Zhixian Wang, Ke Wang, Dong Liu, Yan Yang, Junjun Fan, Kelei Zhuo and Yuanyuan Yue

Asian J Org Chem, 2020, 9, 929
DOI: 10.1002/ajoc.202000159

Palladium‐Catalyzed 3‐Aryl‐5‐acyl‐1,2,4‐thiadiazole Formation from Ketones, Amidines, and Sulfur Powder

Zilong Wang, Hao Xie, Fuhong Xiao, Yanjun Guo, Huawen Huang and Guo‐Jun Deng

Eur J Org Chem, 2017, 2017, 1604
DOI: 10.1002/ejoc.201700148

ChemInform Abstract: Recent Advances in the Willgerodt—Kindler Reaction

Daniel L. Priebbenow and Carsten Bolm

ChemInform, 2013, 44
DOI: 10.1002/chin.201348223

One‐Pot Synthesis of 2,3,5‐Trisubstituted Thiophenes through Three‐Component Assembly of Arylacetaldehydes, Elemental Sulfur, and 1,3‐Dicarbonyls

Zilong Wang, Zhonghua Qu, Fuhong Xiao, Huawen Huang and Guo‐Jun Deng

Adv Synth Catal, 2018, 360, 796
DOI: 10.1002/adsc.201701332

Transamidation of thioacetamide catalyzed by SbCl3

Andrea Ojeda-Porras and Diego Gamba-Sánchez

Tetrahedron Letters, 2015, 56, 4308
DOI: 10.1016/j.tetlet.2015.05.067

Flexible Synthesis of Phosphoryl-Substituted Imidazolines, Tetrahydropyrimidines, and Thioamides by Sulfur-Mediated Processes

Mikhail Kozlov, Alexander Komkov, Timofey Losev, Alexey Tyurin, Andrey Dmitrenok, Igor Zavarzin and Yulia Volkova

J. Org. Chem., 2019, 84, 11533
DOI: 10.1021/acs.joc.9b01384

Synthesis, antitumor activity, and molecular docking study of 2-cyclopentyloxyanisole derivatives: mechanistic study of enzyme inhibition

Walaa M. El-Husseiny, Magda A.-A. El-Sayed, Adel S. El-Azab, Nawaf A. AlSaif, Mohammed M. Alanazi and Alaa A.-M. Abdel-Aziz

Journal of Enzyme Inhibition and Medicinal Chemistry, 2020, 35, 744
DOI: 10.1080/14756366.2020.1740695

Late-Stage Molecular Editing Enabled by Ketone Chain-Walking Isomerization

Yannick Brägger, Ori Green, Benjamin N. Bhawal and Bill Morandi

J. Am. Chem. Soc., 2023, 145, 19496
DOI: 10.1021/jacs.3c05680

Advancing Sustainable Chemistry: MWCNTs/MNPs–Triazine/TMA–I₃ as a Novel Heterogeneous Iodine-Based Nanocatalyst for Eco-Friendly Thioamide Synthesis

Ghada Al-Assi, Magdi E.A. Zaki, G. Padma Priya, Israa Abdulhameed Ahmad, Amrita Pal, Renu Sharma, Sobhi M. Gomha and Reza Mohammadi

Journal of Organometallic Chemistry, 2026, 1049, 124055
DOI: 10.1016/j.jorganchem.2026.124055

Transition-Metal-Free Cleavage of C–C Triple Bonds in Aromatic Alkynes with S8 and Amides Leading to Aryl Thioamides

Kai Xu, Ziyi Li, Fangyuan Cheng, Zhenzhen Zuo, Tao Wang, Mincan Wang and Lantao Liu

Org. Lett., 2018, 20, 2228
DOI: 10.1021/acs.orglett.8b00573

Sulfur‐Promoted Synthesis of 2‐Aroylquinazolin‐4(3H)‐ones by Oxidative Condensation of Anthranilamide and Acetophenones

Thanh Binh Nguyen, Jing‐ya Hou and Pascal Retailleau

Adv Synth Catal, 2019, 361, 3337
DOI: 10.1002/adsc.201900371

Synthesis of Agomelatine by One-pot Catalytic Hydrogenation and Acetylation with NiO

Zhijun Yu, Zhengzai Cheng, Cong Xie, Sheng Zeng, Haiying Deng, Panpan Liu, Hai Hu, Guangyao Li, Ling Ding, Mario Gauthier and Shiqian Li

J. Wuhan Univ. Technol.-Mat. Sci. Edit., 2019, 34, 453
DOI: 10.1007/s11595-019-2073-3

Unexpected Reactivity of Nitrones: Catalytic Insertion of CS2

Marcos López-Aguilar, Nicolás Ríos-Lombardía, Daniel Barrena-Espés, Miguel Gallegos, Joaquín García-Álvarez, Carmen Concellón and Vicente del Amo

Org. Lett., 2025, 27, 8338
DOI: 10.1021/acs.orglett.5c02611

Synthesis of N,N'-Disubstituted Dithiooxamide Derivatives by the Modified Willgerodt–Kindler Reaction

T. N. Ponomareva, E. V. Eliseenkov, A. A. Petrov and V. P. Boyarskii

Russ J Org Chem, 2020, 56, 781
DOI: 10.1134/S1070428020050097

Transition‐Metal‐Free, General Construction of Thioamides from Chlorohydrocarbon, Amide and Elemental Sulfur

Hao Jin, Xinzhi Chen, Chao Qian, Xin Ge and Shaodong Zhou

Eur J Org Chem, 2021, 2021, 3403
DOI: 10.1002/ejoc.202100588

Mechanisms of the Reaction of Elemental Sulfur and Polysulfides with Cyanide and Phosphines**

Jyoti Sharma and Pier Alexandre Champagne

Chemistry A European J, 2023, 29
DOI: 10.1002/chem.202203906

Metal-free three-component synthesis of thioamides from β-nitrostyrenes, amines and elemental sulfur

Ling Peng, Li Ma, Ying Ran, Yunfeng Chen and Zhigang Zeng

Tetrahedron Letters, 2021, 74, 153092
DOI: 10.1016/j.tetlet.2021.153092

Catalyst Free Synthesis of Thioamides from Pyrazole Aldehydes using DMSO as Solvent

S. Helen Perci, K. Gunsundari, P. Monisha and S. Jayanthi

Asian J. Chem., 2023, 35, 1417
DOI: 10.14233/ajchem.2023.27721

Mixed bases mediated synthesis of thioamides in water

Jiao Li, Xuanhe Ren, Ganzhong Li, Helong Liang, Yajie Zhao, Zhiwu Wang, Heng Li and Bingxin Yuan

Journal of Sulfur Chemistry, 2020, 41, 229
DOI: 10.1080/17415993.2020.1722818

Synthesis of o-Arylenediamines through Elemental Sulfur-Promoted Aerobic Dehydrogenative Aromatization of Cyclohexanones with Arylamines

Zhen Wang, Xiangui Chen, Hao Xie, Dahan Wang, Huawen Huang and Guo-Jun Deng

Org. Lett., 2018, 20, 5470
DOI: 10.1021/acs.orglett.8b02387

Strained contacts with the cell membrane may influence ligand affinity to G protein coupled receptors: a case of free fatty acid receptor 1 agonists

Alexey Lukin, Anna Bakholdina, Mikhail Chudinov, Oleksandra Onopchenko, Elena Zhuravel, Sergey Zozulya, Maxim Gureev and Mikhail Krasavin

Journal of Enzyme Inhibition and Medicinal Chemistry, 2021, 36, 1650
DOI: 10.1080/14756366.2021.1955874

Synthesis of Thioamides via Decarboxylative/Oxidative Cross‐Coupling Reaction by Visible‐Light Photocatalysis

Subhankar Sarkar, Satyajit Pal, Sougata Santra, Grigory V. Zyryanov, Susanta Ghosh and Adinath Majee

Asian J Org Chem, 2023, 12
DOI: 10.1002/ajoc.202300141

Synthesis, biological evaluation, molecular docking studies and In-silico ADMET evaluation of pyrazines of pentacyclic triterpenes

Fabiola A. López-Huerta, María Teresa Ramírez-Apan, Carlos A. Méndez-Cuesta, Antonio Nieto-Camacho, Simón Hernández-Ortega, Ericka K.P. Almeida-Aguirre, Marco A. Cerbón and Guillermo Delgado

Bioorganic Chemistry, 2022, 125, 105924
DOI: 10.1016/j.bioorg.2022.105924

Palladium-catalyzed Suzuki-Miyaura coupling of thioureas or thioamides

Shaoyu Mai, Wendong Li, Xue Li, Yingwei Zhao and Qiuling Song

Nat Commun, 2019, 10
DOI: 10.1038/s41467-019-13701-5

Microcrystalline Cellulose Decorated with Fe3O4 Nanoparticle Catalysts for the Microwave-Assisted Synthesis of Thioglyoxamides

Dharmesh J. Shah, Anuj S. Sharma, Vinay S. Sharma, Vinod Kumar Vishwakarma, Achalkumar Ammathnadu Sudhakar, Pranav S. Shrivastav and Rajender S. Varma

ACS Appl. Nano Mater., 2023, 6, 4005
DOI: 10.1021/acsanm.3c00324

Site-Specific Incorporation of Multiple Thioamide Substitutions into a Peptide Backbone via Solid Phase Peptide Synthesis

Jinhua Yang, Changliu Wang, Chaochao Yao, Chunqiu Chen, Yafang Hu, Guifeng He and Junfeng Zhao

J. Org. Chem., 2020, 85, 1484
DOI: 10.1021/acs.joc.9b02486