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Diastereoselective addition of anisoles to N-tert-butanesulfinyl imines via four-membered lithium cycles
Leleti Rajender Reddy, Sharadsrikar Kotturi, Yogesh Waman, Chirag Patel, Aditya Patwa and Rajesh Shenoy
Chem. Commun., 2018, 54, 7007
DOI: 10.1039/C8CC03764G

Modern advances in heterocyclic chemistry in drug discovery
Alexandria P. Taylor, Ralph P. Robinson, Yvette M. Fobian, David C. Blakemore, Lyn H. Jones and Olugbeminiyi Fadeyi
Org. Biomol. Chem., 2016, 14, 6611
DOI: 10.1039/C6OB00936K

Asymmetric synthesis of 1-substituted 2-azaspiro[3.3]heptanes: important motifs for modern drug discovery
Leleti Rajender Reddy, Yogesh Waman, Priya Kallure, Kumara Swamy Nalivela, Zubeda Begum, Thumbar Divya and Sharadsrikar Kotturi
Chem. Commun., 2019, 55, 5068
DOI: 10.1039/C9CC00863B

Asymmetric synthesis of 2-arylpyrrolidines starting from γ-chloro N-(tert-butanesulfinyl)ketimines
Erika Leemans, Sven Mangelinckx and Norbert De Kimpe
Chem. Commun., 2010, 46, 3122
DOI: 10.1039/b925209f

Construction of an α-chiral pyrrolidine library with a rapid and scalable continuous flow protocol
Chao Shan, Liming Cao, Jiasheng Yang, Ruihua Cheng, Xiantong Yao, Chaoming Liang, Maolin Sun and Jinxing Ye
React. Chem. Eng., 2022, 7, 1779
DOI: 10.1039/D2RE00145D

A Concise and Stereoselective Synthesis of Hydroxypyrrolidines: Rapid Synthesis of (+)-Preussin
Jason A. Draper and Robert Britton
Org. Lett., 2010, 12, 4034
DOI: 10.1021/ol101631e

Rhodium-Catalyzed Asymmetric Arylation of N-(tert-Butanesulfinyl)imines with Sodium Tetraarylborates
Leleti Rajender Reddy, Aditya P. Gupta, Eric Villhauer and Yugang Liu
J. Org. Chem., 2012, 77, 1095
DOI: 10.1021/jo2024224

A Protocol for an Asymmetric Synthesis of γ-Amino Acids
Leleti Rajender Reddy, Kapa Prasad and Mahavir Prashad
J. Org. Chem., 2012, 77, 6296
DOI: 10.1021/jo301177f

Factors Influencing the Regioselectivity of the Oxidation of Asymmetric Secondary Amines with Singlet Oxygen
Dmitry B. Ushakov , Matthew B. Plutschack , Kerry Gilmore and Peter H. Seeberger 
Chemistry A European J, 2015, 21, 6528
DOI: 10.1002/chem.201500121

Diastereoselective synthesis of α,α,α′-trisubstituted pyrrolidines and piperidines by directed sequential lithiation/alkylation
Timothy K. Beng and Nathan Fox
Tetrahedron Letters, 2015, 56, 119
DOI: 10.1016/j.tetlet.2014.11.031

Enantioselective Imine Reduction Catalyzed by Phosphenium Ions
Travis Lundrigan, Erin N. Welsh, Toren Hynes, Chieh-Hung Tien, Matt R. Adams, Kayelani R. Roy, Katherine N. Robertson and Alexander W. H. Speed
J. Am. Chem. Soc., 2019, 141, 14083
DOI: 10.1021/jacs.9b07293

Mimicking the environment of living organisms to achieve the oxidative coupling of amines to imines catalyzed by water-soluble metalloporphyrins
Xian-Tai Zhou, Qing-Gang Ren and Hong-Bing Ji
Tetrahedron Letters, 2012, 53, 3369
DOI: 10.1016/j.tetlet.2012.04.096

Stereocomplementary Synthesis of Pharmaceutically Relevant Chiral 2-Aryl-Substituted Pyrrolidines Using Imine Reductases
Yu-Hui Zhang, Fei-Fei Chen, Bo-Bo Li, Xin-Yi Zhou, Qi Chen, Jian-He Xu and Gao-Wei Zheng
Org. Lett., 2020, 22, 3367
DOI: 10.1021/acs.orglett.0c00802

Chiral Sulfur Compounds Studied by Raman Optical Activity: tert‐Butanesulfinamide and its Precursor tert‐Butyl tert‐Butanethiosulfinate
Shi Qiu, Guanna Li, Shengmei Lu, Baokun Huang, Zhaochi Feng and Can Li
Chirality, 2012, 24, 731
DOI: 10.1002/chir.22038

Pt–Sn/γ‐Al2O3‐Catalyzed Highly Efficient Direct Synthesis of Secondary and Tertiary Amines and Imines
Wei He, Liandi Wang, Chenglin Sun, Kaikai Wu, Songbo He, Jiping Chen, Ping Wu and Zhengkun Yu 
Chemistry A European J, 2011, 17, 13308
DOI: 10.1002/chem.201101725

Synthesis of Enantioenriched Pyrrolidines via Gold-Catalyzed Tandem Cycloisomerization/Hydrogenation of Chiral Homopropargyl Sulfonamides
Yong-Fei Yu, Chao Shu, Tong-De Tan, Long Li, Shahid Rafique and Long-Wu Ye
Org. Lett., 2016, 18, 5178
DOI: 10.1021/acs.orglett.6b02736

Henry–Nef reaction: a practical and versatile chiral pool route to 2-substituted pyrrolidine and piperidine alkaloids
Chinmay Bhat and Santosh G. Tilve
Tetrahedron, 2013, 69, 6129
DOI: 10.1016/j.tet.2013.05.055

Synthesis of Nitrogenated Heterocycles by Asymmetric Transfer Hydrogenation of N-(tert-Butylsulfinyl)haloimines
Óscar Pablo, David Guijarro and Miguel Yus
J. Org. Chem., 2013, 78, 9181
DOI: 10.1021/jo4014386

Straightforward Access to Enantioenriched 2-Allylpiperidine: Application to the Synthesis of Alkaloids
Irene Bosque, José C. González-Gómez, Francisco Foubelo and Miguel Yus
J. Org. Chem., 2012, 77, 780
DOI: 10.1021/jo202211u

Tetrabenzylhafnium as a New Organometallic Reagent for Imine Addition Resulting in α‐Branched Amines
Haibo Mei, Xiaoyun Ji, Jianlin Han and Yi Pan
Eur J Org Chem, 2011, 2011, 5783
DOI: 10.1002/ejoc.201100820

Asymmetric synthesis of 2-substituted cyclic amines
Amit A. Kudale, Prasad Anaspure, Falguni Goswami and Matthew Voss
Tetrahedron Letters, 2014, 55, 7219
DOI: 10.1016/j.tetlet.2014.11.022

Total Synthesis of (−)-Aurantioclavine
Katrien Brak and Jonathan A. Ellman
Org. Lett., 2010, 12, 2004
DOI: 10.1021/ol100470g

ChemInform Abstract: Asymmetric Synthesis of 2‐Substituted Pyrrolidines by Addition of Grignard Reagents to γ‐Chlorinated N‐tert‐Butanesulfinyl Imine.
Leleti Rajender Reddy and Mahavir Prashad
ChemInform, 2010, 41
DOI: 10.1002/chin.201019096

Rapid Synthesis of α-Chiral Piperidines via a Highly Diastereoselective Continuous Flow Protocol
Chao Shan, Jinping Xu, Liming Cao, Chaoming Liang, Ruihua Cheng, Xiantong Yao, Maolin Sun and Jinxing Ye
Org. Lett., 2022, 24, 3205
DOI: 10.1021/acs.orglett.2c00975

Flow Synthesis of Fluorinated α‐Amino Acids
Stella Vukelić, Dmitry B. Ushakov, Kerry Gilmore, Beate Koksch and Peter H. Seeberger
Eur J Org Chem, 2015, 2015, 3036
DOI: 10.1002/ejoc.201500300

A flexible method for the synthesis of 2-substituted 1,2,5,6-tetrahydropyridines and piperidines from chloro-containing propargylamines
Danielle N. Penk, Nathan A. Robinson, Harrison M. Hill and Mark Turlington
Tetrahedron Letters, 2017, 58, 470
DOI: 10.1016/j.tetlet.2016.12.061

Umpolung Synthesis of Vicinal Diamines: Diastereoselective Addition of 2-Azaallyl Anions to Davis–Ellman’s Imines
Leleti Rajender Reddy, Sharadsrikar Kotturi, Rajesh Shenoy, Kumara Swamy Nalivela, Chirag Patel, Poojabahen Raval and Vinkal Zalavadiya
Org. Lett., 2018, 20, 5423
DOI: 10.1021/acs.orglett.8b02331

Recent Advances in Asymmetric Synthesis of Pyrrolidine-Based Organocatalysts and Their Application: A 15-Year Update
Arianna Quintavalla, Davide Carboni and Marco Lombardo
Molecules, 2023, 28, 2234
DOI: 10.3390/molecules28052234

Ionic‐Liquid‐Assisted Metal‐Free Oxidative Coupling of Amines To Give Imines
Antonio Monopoli, Pietro Cotugno, Francesco Iannone, Francesco Ciminale, Maria Michela Dell'Anna, Piero Mastrorilli and Angelo Nacci
Eur J Org Chem, 2014, 2014, 5925
DOI: 10.1002/ejoc.201402530

A Kinome-Wide Selective Radiolabeled TrkB/C Inhibitor for in Vitro and in Vivo Neuroimaging: Synthesis, Preclinical Evaluation, and First-in-Human
Vadim Bernard-Gauthier, Justin J. Bailey, Andrew V. Mossine, Simon Lindner, Lena Vomacka, Arturo Aliaga, Xia Shao, Carole A. Quesada, Phillip Sherman, Anne Mahringer, Alexey Kostikov, Marilyn Grand’Maison, Pedro Rosa-Neto, Jean-Paul Soucy, Alexander Thiel, David R. Kaplan, Gert Fricker, Björn Wängler, Peter Bartenstein, Ralf Schirrmacher and Peter J. H. Scott
J. Med. Chem., 2017, 60, 6897
DOI: 10.1021/acs.jmedchem.7b00396

Regio‐ and Diastereoselective and Enantiospecific Metal‐Free C(sp3)H Arylation: Facile Access to Optically Active 5‐Aryl 2,5‐Disubstituted Pyrrolidines
Surajit Haldar, Subhra Kanti Roy, Bholanath Maity, Debasis Koley and Chandan K. Jana
Chemistry A European J, 2015, 21, 15290
DOI: 10.1002/chem.201502297

Subtle Strain-Release-Driven Aroylation of Four-Membered Rings via Decarboxylative Giese-Type Reactions
Rafael D. Hernández, Aishwarya Singh, Marco Caricato and Jon A. Tunge
Org. Lett., 2025, 27, 8574
DOI: 10.1021/acs.orglett.5c02499

Synthesis of 2-arylpyrrolidines by reaction of γ-ureidoacetals with benzene-1,3,5-triol
A. V. Smolobochkin, A. S. Gazizov, A. R. Burilov, M. A. Pudovik, D. G. Khuzyasheva and R. R. Amirov
Russ J Org Chem, 2016, 52, 538
DOI: 10.1134/S1070428016040102

Asymmetric Synthesis 1-Substituted 2,6-Diazaspiro[3.3]heptanes through Addition of 3-Azetidinecarboxylate Anions to Davis–Ellman Imines
Leleti Rajender Reddy, Yogesh Waman, Krishna Nayak, Kasimraza Baharooni and Sharadsrikar Kotturi
Org. Lett., 2019, 21, 3481
DOI: 10.1021/acs.orglett.9b00564

Asymmetric Synthesis of α-Amino Acids by Reduction of N-tert-Butanesulfinyl Ketimine Esters
Leleti Rajender Reddy, Aditya P. Gupta and Yugang Liu
J. Org. Chem., 2011, 76, 3409
DOI: 10.1021/jo200401a

Asymmetric Synthesis of Pyrrolidine‐Containing Chemical Scaffolds via Tsuji–Trost Allylation of N‐tert‐Butanesulfinyl Imines
Rafid S. Dawood, Irene Georgiou, Ross P. Wilkie, William Lewis and Robert A. Stockman
Chemistry A European J, 2017, 23, 11153
DOI: 10.1002/chem.201702616

Highly Enantioselective Arylation of N-Tosylalkylaldimines Catalyzed by Rhodium-Diene Complexes
Zhe Cui, Hong-Jie Yu, Rui-Feng Yang, Wen-Yun Gao, Chen-Guo Feng and Guo-Qiang Lin
J. Am. Chem. Soc., 2011, 133, 12394
DOI: 10.1021/ja2046217

Enantiodivergent Approach to the Synthesis of Cis-2,6-Disubstituted Piperidin-4-ones
Alejandro Lahosa, Miguel Yus and Francisco Foubelo
J. Org. Chem., 2019, 84, 7331
DOI: 10.1021/acs.joc.9b01008

A Facile Asymmetric Synthesis of Either Enantiomer of 2-Substituted Pyrrolidines
Leleti Rajender Reddy, Sonia G. Das, Yugang Liu and Mahavir Prashad
J. Org. Chem., 2010, 75, 2236
DOI: 10.1021/jo902710s

Enantioselective Synthesis of α-Heteroarylpyrrolidines by Copper-Catalyzed 1,3-Dipolar Cycloaddition of α-Silylimines
Ana Pascual-Escudero, María González-Esguevillas, Silvia Padilla, Javier Adrio and Juan C. Carretero
Org. Lett., 2014, 16, 2228
DOI: 10.1021/ol5007373

Enantioselective, Palladium-Catalyzed α-Arylation of N-Boc Pyrrolidine: In Situ React IR Spectroscopic Monitoring, Scope, and Synthetic Applications
Graeme Barker, Julia L. McGrath, Artis Klapars, Darren Stead, George Zhou, Kevin R. Campos and Peter O’Brien
J. Org. Chem., 2011, 76, 5936
DOI: 10.1021/jo2011347

Reaction of 4-chloro- and 4-bromobenzene-1,3-diols with 1-alkyl-3-(4,4-diethoxybutyl)ureas in the presence of trifluoroacetic acid
A. V. Smolobochkin, A. S. Gazizov, A. R. Burilov and M. A. Pudovik
Russ J Org Chem, 2015, 51, 1261
DOI: 10.1134/S1070428015090079

Engineered Imine Reductase for Larotrectinib Intermediate Manufacture
Qi Chen, Bo-Bo Li, Lilan Zhang, Xin-Ru Chen, Xin-Xin Zhu, Fei-Fei Chen, Min Shi, Chun-Chi Chen, Yu Yang, Rey-Ting Guo, Weidong Liu, Jian-He Xu and Gao-Wei Zheng
ACS Catal., 2022, 12, 14795
DOI: 10.1021/acscatal.2c03783

Synthesis and Applications of tert-Butanesulfinamide
MaryAnn T. Robak, Melissa A. Herbage and Jonathan A. Ellman
Chem. Rev., 2010, 110, 3600
DOI: 10.1021/cr900382t

Enantioselective C–H Amination Catalyzed by Nickel Iminyl Complexes Supported by Anionic Bisoxazoline (BOX) Ligands
Yuyang Dong, Colton J. Lund, Gerard J. Porter, Ryan M. Clarke, Shao-Liang Zheng, Thomas R. Cundari and Theodore A. Betley
J. Am. Chem. Soc., 2021, 143, 817
DOI: 10.1021/jacs.0c09839

Highly Enantioselective Rh-Catalyzed Alkenylation of Imines: Synthesis of Chiral Allylic Amines via Asymmetric Addition of Potassium Alkenyltrifluoroborates to N-Tosyl Imines
Balraj Gopula, Chien-Wei Chiang, Way-Zen Lee, Ting-Shen Kuo, Ping-Yu Wu, Julian P. Henschke and Hsyueh-Liang Wu
Org. Lett., 2014, 16, 632
DOI: 10.1021/ol4035897

Asymmetric Synthesis of α-(Diarylmethyl) Alkyl Amines through Regioselective Lithiation of α-Diarylmethanes and the Diastereoselective Addition to Ellman’s Imines
Leleti Rajender Reddy, Sharadsrikar Kotturi, Yogesh Waman, Chirag Patel, Megha Danidharia and Rajesh Shenoy
J. Org. Chem., 2018, 83, 6573
DOI: 10.1021/acs.joc.8b00879

Stereoselective Synthesis of α-Disubstituted β-Homoprolines
Arianna Quintavalla, Davide Carboni, Maria Simeone and Marco Lombardo
Org. Lett., 2023, 25, 7067
DOI: 10.1021/acs.orglett.3c02891

Classical-Reaction-Driven Stereo- and Regioselective C(sp3)-H Functionalization of Aliphatic Amines
Sujit Mahato and Chandan K. Jana
The Chemical Record, 2016, 16, 1477
DOI: 10.1002/tcr.201600001

Asymmetric Synthesis of Either Enantiomer of β-Butadienyl Amines by Isoprenylation of Davis–Ellman Imines
Leleti Rajender Reddy, Venu Aili and Shiva Kumar Koppula
J. Org. Chem., 2025, 90, 8136
DOI: 10.1021/acs.joc.5c00463

Total Syntheses of (−) Epilupinine and (−)-Tashiromine Using Imino-Aldol Reactions
Amanda C. Cutter, Iain R. Miller, John F. Keily, Richard K. Bellingham, Mark E. Light and Richard C. D. Brown
Org. Lett., 2011, 13, 3988
DOI: 10.1021/ol2015048

Metal-free oxidation of benzyl amines to imines
Xiao-Feng Wu, Andranik Petrosyan, Tariel V. Ghochikyan, Ashot S. Saghyan and Peter Langer
Tetrahedron Letters, 2013, 54, 3158
DOI: 10.1016/j.tetlet.2013.04.018

Pyrrolidine and Indolizidine Alkaloids from Chiral N-tert-Butanesulfinyl Imines Derived from 4-Halobutanal
Ana Sirvent, Sandra Hernández-Ibáñez, Miguel Yus and Francisco Foubelo
Synthesis, 2021, 53, 1749
DOI: 10.1055/s-0037-1610763