Nazarov reaction: current trends and recent advances in the synthesis of natural compounds and their analogs

Maxim G. Vinogradov, Olga V. Turova and Sergei G. Zlotin

Org. Biomol. Chem., 2017, 15, 8245
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A one pot three-component reaction for the preparation of dihydroquinolines with two different ketones and aromatic amines

Guobin Yang, Guangxun Li, Jin Huang, Zhuo Tang and Jinzhong Zhao

Org. Biomol. Chem., 2017, 15, 10167
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l-Proline derived nitrogenous steroidal systems: an asymmetric approach to 14-azasteroids

Ritesh Singh and Gautam Panda

RSC Adv., 2013, 3, 19533
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Application of Nazarov type electrocyclization to access [6,5,6] and [6,5,5] core embedded new polycycles: an easy entry to tetrahydrofluorene scaffolds related to Taiwaniaquinoids and C-nor-D homosteroids

Ritesh Singh and Gautam Panda

Org. Biomol. Chem., 2011, 9, 4782
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Trifluoromethylthio-promoted Nazarov cyclization of α-SCF3-vinyl (hetero)aryl ketones

Sugyeong Kim, Yu Jin Pyo, Geon Ryun Park, Hyungu Kang, Heon-Jong Ha, Sang Ho Kim, Ha Yun Nam, Daeheum Cho and Chang-Woo Cho

Org. Biomol. Chem., 2026, 24, 360
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Facile assembly of indeno[1,2-c]chromenes via a palladium-catalyzed reaction of 2-alkynylhalobenzene

Xiaolin Pan, Hongming Nie, Yong Luo, Yueqiu Gao and Jie Wu

Org. Biomol. Chem., 2012, 10, 8244
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Microwave assisted [RuCl2(p-cymene)2]2 catalyzed regioselective endo-tandem cyclization involving imine and alkyne activation: an approach to benzo[4,5]imidazo[2,1-a]pyridine scaffold

Sudipta Kumar Manna and Gautam Panda

RSC Adv., 2014, 4, 21032
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PtI2-Catalyzed tandem 3,3-rearrangement/Nazarov reaction of arylpropargylic esters: synthesis of indanone derivatives

Huaiji Zheng, Xingang Xie, Juan Yang, Changgui Zhao, Peng Jing, Bowen Fang and Xuegong She

Org. Biomol. Chem., 2011, 9, 7755
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Efficient generation of indeno[1,2-c]chromenes via the Pd-catalyzed reaction of 2-alkynylhalobenzenes with 2-alkynylphenols

Yong Luo, Linxiang Hong and Jie Wu

Chem. Commun., 2011, 47, 5298
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Lewis acid-catalyzed tandem acylation–Nazarov cyclization for the syntheses of fused cyclopentenones

Ertong Li, Changwei Li, Jing Wang, Jinqian Wang, Lihong Dong, Xiaohe Guo, Chuanjun Song and Junbiao Chang

Tetrahedron, 2014, 70, 874
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Trapping the Oxyallyl Cation Intermediate Derived from the Nazarov Cyclization of Allenyl Vinyl Ketones with Nitrogen Heterocycles

Vanessa M. Marx, François M. LeFort and D. Jean Burnell

Adv Synth Catal, 2011, 353, 64
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Catalytic Nazarov Cyclization: The State of the Art

Tulaza Vaidya, Richard Eisenberg and Alison J. Frontier

ChemCatChem, 2011, 3, 1531
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Using Nazarov Electrocyclization to Stage Chemoselective [1,2]‐Migrations: Stereoselective Synthesis of Functionalized Cyclopentenones

David Lebœuf, Jie Huang, Vincent Gandon and Alison J. Frontier

Angew Chem Int Ed, 2011, 50, 10981
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Bildung von α‐Ketoradikalen aus Vinylbromiden und molekularem Sauerstoff mit sichtbarem Licht: Synthese von Indenonen und Dihydroindeno[1,2‐c]chromenen

Santosh K. Pagire, Peter Kreitmeier and Oliver Reiser

Angewandte Chemie, 2017, 129, 11068
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Visible‐Light‐Promoted Generation of α‐Ketoradicals from Vinyl‐bromides and Molecular Oxygen: Synthesis of Indenones and Dihydroindeno[1,2‐c]chromenes

Santosh K. Pagire, Peter Kreitmeier and Oliver Reiser

Angew Chem Int Ed, 2017, 56, 10928
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A Catalytic Intramolecular Aldehyde–Alkyne Metathesis Approach to Azepino[1,2‐a]indoles

Upasana Deka, Arup Jyoti Das, Swapnil Kumar Nath and Sajal Kumar Das

Adv Synth Catal, 2024, 366, 4452
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Diastereoselective annulation of 2-substituted 3-nitro-2H-chromenes by phosphine catalyzed [3+2] allenoate cycloaddition: Syntheses of tetrahydrocyclopenta[c]chromenes

Ivan A. Kochnev and Alexey Y. Barkov

Tetrahedron Letters, 2026, 176, 155931
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[RuCl2(p-cymene)2]2 catalyzed cross dehydrogenative coupling (CDC) toward xanthone and fluorenone analogs through intramolecular C–H bond functionalization reaction

Sudipta Kumar Manna, Srinivas Lavanya Kumar Manda and Gautam Panda

Tetrahedron Letters, 2014, 55, 5759
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Synthesis of 5-epi-Taiwaniaquinone G

Jinqian Wang, Jing Wang, Changwei Li, Yonggang Meng, Jie Wu, Chuanjun Song and Junbiao Chang

J. Org. Chem., 2014, 79, 6354
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Flow Photo-Nazarov Reactions of 2-Furyl Vinyl Ketones: Cyclizing a Class of Traditionally Unreactive Heteroaromatic Enones

William L. Ashley, Evan L. Timpy and Thomas C. Coombs

J. Org. Chem., 2018, 83, 2516
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An overview of synthetic approaches for heterocyclic steroids

Ritesh Singh and Gautam Panda

Tetrahedron, 2013, 69, 2853
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ChemInform Abstract: Application of Nazarov Cyclization to Access [6‐5‐6] and [6‐5‐5]Tricyclic Core Embedded New Heterocycles: An Easy Entry to Structures Related to Taiwaniaquinoids.

Ritesh Singh, Maloy Kumar Parai and Gautam Panda

ChemInform, 2009, 40
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Synthesis of Heteroarene‐Fused Cyclopentadienes and Related Compounds Suitable for Metallocene Preparation

Ilya E. Nifant'ev and Pavel V. Ivchenko

Adv Synth Catal, 2020, 362, 3727
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Enantioselective Synthesis of Axially Chiral Styrene‐Carboxylic Esters by Rhodium‐Catalyzed Chelation‐Controlled [2+2+2] Cycloaddition

Daisuke Yokose, Yuki Nagashima, Suzuka Kinoshita, Juntaro Nogami and Ken Tanaka

Angew Chem Int Ed, 2022, 61
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Using Nazarov Electrocyclization to Stage Chemoselective [1,2]‐Migrations: Stereoselective Synthesis of Functionalized Cyclopentenones

David Lebœuf, Jie Huang, Vincent Gandon and Alison J. Frontier

Angewandte Chemie, 2011, 123, 11173
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Visible-light-induced, Ir-catalyzed reactions of N-methyl-N-((trimethylsilyl)methyl)aniline with cyclic α,β-unsaturated carbonyl compounds

Dominik Lenhart and Thorsten Bach

Beilstein J. Org. Chem., 2014, 10, 890
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Enantioselective Synthesis of Axially Chiral Styrene‐Carboxylic Esters by Rhodium‐Catalyzed Chelation‐Controlled [2+2+2] Cycloaddition

Daisuke Yokose, Yuki Nagashima, Suzuka Kinoshita, Juntaro Nogami and Ken Tanaka

Angewandte Chemie, 2022, 134
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Trifluoromethanesulfonic Acid Catalyzed Isomerization of Kinetic Enol Derivatives to the Thermodynamically Favored Isomers

Phil Ho Lee, Dongjin Kang, Subin Choi and Sunggak Kim

Org. Lett., 2011, 13, 3470
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Reagent Control of [1,2]‐Wagner–Meerwein Shift Chemoselectivity Following the Nazarov Cyclization: Application to the Total Synthesis of Enokipodin B

David Lebœuf, Christopher M. Wright and Alison J. Frontier

Chemistry A European J, 2013, 19, 4835
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Tandem gem–dichlorination and nitrile oxide generation from chlorochromene aldoximes: synthesis of a new class of room temperature fluxional 4‐chromanone derivatives

Ashutosh K. Dash, Chaitanya K. Jaladanki, Dilip K. Maiti, Deepika Singh, Anil K. Tripathi, Vivek K. Gupta, Prasad V. Bharatam and Debaraj Mukherjee

ChemistrySelect, 2016, 1, 567
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Solvent-Free Mechanosynthesis of Polysubstituted 1,2-Dihydroquinolines from Anilines and Alkyne Esters

Hui Xu and Guan-Wu Wang

J. Org. Chem., 2022, 87, 8480
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Construction of the Bacteriochlorin Macrocycle with Concomitant Nazarov Cyclization To Form the Annulated Isocyclic Ring: Analogues of Bacteriochlorophyll a

Shaofei Zhang and Jonathan S. Lindsey

J. Org. Chem., 2017, 82, 2489
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Synthesis of 4‐Acylchromene via Highly Chemoselective Iodine‐Catalyzed Cyclization of Alkynylarylether Dimethylacetals

Warabhorn Rodphon, Charnsak Thongsornkleeb, Jumreang Tummatorn and Somsak Ruchirawat

Chemistry An Asian Journal, 2020, 15, 3475
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Understanding the Fate of the Oxyallyl Cation following Nazarov Electrocyclization: Sequential Wagner−Meerwein Migrations and the Synthesis of Spirocyclic Cyclopentenones

Jie Huang, David Lebœuf and Alison J. Frontier

J. Am. Chem. Soc., 2011, 133, 6307
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Experimental and Theoretical Studies on the Nazarov Cyclization/Wagner–Meerwein Rearrangement Sequence

David Lebœuf, Vincent Gandon, Jennifer Ciesielski and Alison J. Frontier

J. Am. Chem. Soc., 2012, 134, 6296
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