Synthesis of (Z)-Alkene and (E)-Fluoroalkene-Containing Diketopiperazine Mimetics Utilizing Organocopper-Mediated Reduction−Alkylation and Diastereoselectivity Examination Using DFT Calculations

Ayumu Niida, Makiko Mizumoto, Tetsuo Narumi, Eriko Inokuchi, Shinya Oishi, Hiroaki Ohno, Akira Otaka, Kazuo Kitaura and Nobutaka Fujii

J. Org. Chem., 2006, 71, 4118
DOI: 10.1021/jo060202z

Application of tri- and tetrasubstituted alkene dipeptide mimetics to conformational studies of cyclic RGD peptides

Shinya Oishi, Kazuhide Miyamoto, Ayumu Niida, Mikio Yamamoto, Keiichi Ajito, Hirokazu Tamamura, Akira Otaka, Yoshihiro Kuroda, Akira Asai and Nobutaka Fujii

Tetrahedron, 2006, 62, 1416
DOI: 10.1016/j.tet.2005.11.033

Optically Active γ‐Hydroxy Sulfone Julia Reagents for the Synthesis of Peptidyl Olefin Peptidomimetics

Sima Mirilashvili, Naama Chasid‐Rubinstein and Amnon Albeck

Eur J Org Chem, 2008, 2008, 3461
DOI: 10.1002/ejoc.200800334

Optically Active Functionalized Building Blocks for Peptidyl Olefin Peptidomimetics

Ekaterina Lerman, Shlomo Levinger and Amnon Albeck

ChemistrySelect, 2021, 6, 7912
DOI: 10.1002/slct.202102058

Structure-Activity Relationship Studies on Cyclic RGD Peptides Utilizing Novel Alkene Dipeptide Isosteres

Shinya OISHI

YAKUGAKU ZASSHI, 2004, 124, 269
DOI: 10.1248/yakushi.124.269

Structure–Activity Relationship Study of a CXC Chemokine Receptor Type 4 Antagonist, FC131, Using a Series of Alkene Dipeptide Isosteres

Kazuya Kobayashi, Shinya Oishi, Ryoko Hayashi, Kenji Tomita, Tatsuhiko Kubo, Noriko Tanahara, Hiroaki Ohno, Yasushi Yoshikawa, Toshio Furuya, Masaru Hoshino and Nobutaka Fujii

J. Med. Chem., 2012, 55, 2746
DOI: 10.1021/jm2016914

Optically Active N‐ and C‐Terminal Building Blocks for the Synthesis of Peptidyl Olefin Peptidomimetics

Sima Mirilashvili, Naama Chasid‐Rubinstein and Amnon Albeck

Eur J Org Chem, 2010, 2010, 4671
DOI: 10.1002/ejoc.201000539

Application of divergent multi-component reactions in the synthesis of a library of peptidomimetics based on γ-amino-α,β-cyclopropyl acids

Peter Wipf, Stefan Werner, Grace H.C. Woo, Corey R.J. Stephenson, Maciej A.A. Walczak, Claire M. Coleman and Leslie A. Twining

Tetrahedron, 2005, 61, 11488
DOI: 10.1016/j.tet.2005.09.016

Stereoselective Synthesis of 3,6-Disubstituted-3,6-dihydropyridin-2-ones as Potential Diketopiperazine Mimetics Using Organocopper-Mediated anti-SN2‘ Reactions and Their Use in the Preparation of Low-Molecule CXCR4 Antagonists

Ayumu Niida, Hiroaki Tanigaki, Eriko Inokuchi, Yoshikazu Sasaki, Shinya Oishi, Hiroaki Ohno, Hirokazu Tamamura, Zixuan Wang, Stephen C. Peiper, Kazuo Kitaura, Akira Otaka and Nobutaka Fujii

J. Org. Chem., 2006, 71, 3942
DOI: 10.1021/jo060390t

Synthesis of fluorine‐containing bioisosteres corresponding to phosphoamino acids and dipeptide units

Akira Otaka, Etsuko Mitsuyama, Junko Watanabe, Hideaki Watanabe and Nobutaka Fujii

Biopolymers, 2004, 76, 140
DOI: 10.1002/bip.10570

Stereocontrolled Synthesis of Tetrasubstituted Olefins

Alison B. Flynn and William W. Ogilvie

Chem. Rev., 2007, 107, 4698
DOI: 10.1021/cr050051k

Catalytic Asymmetric Conjugate Addition and Allylic Alkylation with Grignard Reagents

Syuzanna R. Harutyunyan, Tim den Hartog, Koen Geurts, Adriaan J. Minnaard and Ben L. Feringa

Chem. Rev., 2008, 108, 2824
DOI: 10.1021/cr068424k

Facile access to (Z)-alkene-containing diketopiperazine mimetics utilizing organocopper-mediated anti-SN2′ reactions

Ayumu Niida, Shinya Oishi, Yoshikazu Sasaki, Makiko Mizumoto, Hirokazu Tamamura, Nobutaka Fujii and Akira Otaka

Tetrahedron Letters, 2005, 46, 4183
DOI: 10.1016/j.tetlet.2005.04.057