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Synthesis, conformational stability and molecular structure of 4-aryl- and 4,5-diaryl-1,8-bis(dimethylamino)naphthalenes

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Natural product inspired antibiotics approved for human use – 1943 to 2025

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Trienomycin A-simplified analogs: Synthesis and anti-neuroinflammatory activity

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Design, synthesis, in silico and in vitro investigation of 4-cyano-2-phenyl-1,3-oxazole-5-sulfonamide derivatives

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Cascade Transformation of the Ansamycin Benzoquinone Core into Benzoxazole Influencing Anticancer Activity and Selectivity

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New Structure Activity Relationship Insight into the Role of the C‐3 Extension on Rifamycin Antimycobacterial Activity

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Nagimycins A and B, Antibacterial Ansamycin-Related Macrolactams from Streptomyces sp. NA07423

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Piperidine-containing drugs and recently studied analogs – biological activity, mechanism of action and synthetic cascade access to their scaffolds

Daniel Łowicki and Piotr Przybylski

European Journal of Medicinal Chemistry, 2026, 302, 118213
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The antimicrobial potential of adarotene derivatives against Staphylococcus aureus strains

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Natural occurrence, bioactivity, and biosynthesis of triene-ansamycins

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European Journal of Medicinal Chemistry, 2022, 244, 114815
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Undescribed ansatrienin analogs from Streptomyces flaveolus including two N-acetylcysteine conjugates

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Recent progress toward developing axial chirality bioactive compounds

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Synthesis, characterization and biological influences of rifaximin loaded melanin/zinc oxide nanoparticles

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From dansyl-modified biofilm disruptors to β-cyclodextrin-optimized multifunctional supramolecular nanovesicles: their improved treatment for plant bacterial diseases

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A review of recent advancement in covalent organic framework (COFs) synthesis and characterization with a focus on their applications in antibacterial activity

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Double Bond Geometric Isomers of Pentaketide Ansamycins from Streptomyces sp. S008

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Synthesis, characterization of phenyl (2,4-dinitro-1-naphthyl) thioethers, kinetic and mechanistic study of their hydrazinolysis in methanol

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Can. J. Chem., 2025
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Therapeutic Potential of Heat Shock Protein 90 Inhibitors, Geldanamycin, and Analog Compounds in Precision Cancer Therapy

Atta Mohammed Alzebari, Amjad Mahmood Qadir, Mahmood Sherzad Rafaat and Abbas Salihi

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Evolution and evolvability of rifampicin resistance across the bacterial tree of life

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Flavin-Dependent Monooxygenase Kmy13 Mediates Formation of the Carbocyclic ansa System during Kendomycin B Biosynthesis

Jiang Chen, Hongjie Zhu, Ming Peng, Shanwen Zhang, Qinglian Li, Yu-Cheng Gu and Jianhua Ju

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Iron-catalyzed synthesis of N-heterocycles via intermolecular and intramolecular cyclization reactions: A review

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Microbial diversity in camel milk from Xinjiang, China as revealed by metataxonomic analysis

Miao Sun, Wei Shao, Zhengyu Liu, Xianlan Ma, He Chen, Nan Zheng and Yankun Zhao

Front. Microbiol., 2024, 15
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Comprehensive Overview of Antibacterial Drugs and Natural Antibacterial Compounds Found in Food Plants

Sabine Berteina-Raboin

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