Is structural hybridization invoking new dimensions for antimalarial drug discovery research?

Bhawana Sharma, Alka Agarwal and Satish Kumar Awasthi

RSC Med. Chem., 2023, 14, 1227
DOI: 10.1039/D3MD00083D

Synthesis, in vitro potency of inhibition, enzyme kinetics and in silico studies of quinoline-based α-glucosidase inhibitors

Minoo Khalili Ghomi, Navid Dastyafteh, Mohammad Nazari Montazer, Milad Noori, Somayeh Mojtabavi, Mohammad Ali Faramarzi, Seyedeh Mahdieh Hashemi and Mohammad Mahdavi

Sci Rep, 2024, 14
DOI: 10.1038/s41598-023-50711-2

A Sustainable Approach for Palladium and Phosphane‐Free Sonogashira Type Cross‐Coupling of 2‐Chloroquinoline with Terminal Alkynes

Zebabanu Khalifa and Amit B. Patel

ChemistrySelect, 2024, 9
DOI: 10.1002/slct.202403356

Mechanistic and Synergistic Evaluation of Amodiaquine–Isometamidium Combination Against Trypanosoma evansi: Integrated In Silico–In-Vitro Insights

Waqas Ahmad, Naeem Rasool, Mehmood Ahmad, Muhammad Yasin Tipu, Tehreem Fayyaz, Usama Bin Naeem, Sadaf Aroosa and Rana Muhammad Zahid Mushtaq

Acta Parasit., 2026, 71
DOI: 10.1007/s11686-026-01228-x

Unveiling the crystal structure and quantum properties of 6‑bromo-N-pyridin-4-yl-2-thiophen-2-ylquinoline-4-carboxamide: A promising journey towards predicting its anticancer potential

T.S. Shashidhara, C.S. Navyashree, M.K. Hema, K. Mantelingu, R. Jothi Ramalingam, Muthusamy Karnan, M. Umashankar and N.K. Lokanath

Journal of Molecular Structure, 2023, 1293, 136266
DOI: 10.1016/j.molstruc.2023.136266

Quinoline Derivatives with Different Functional Groups: Evaluation of Their Catecholase Activity

Mohamed Moutaouakil, Said Tighadouini, Zainab M. Almarhoon, Maha I. Al-Zaben, Abir Ben Bacha, Vijay H. Masand, Jamal Jamaleddine and Rafik Saddik

Catalysts, 2022, 12, 1468
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Identification of novel DNA gyrase inhibitor by combined pharmacophore modeling, QSAR analysis, molecular docking, molecular dynamics, ADMET and DFT approaches

Anguraj Moulishankar, Murugesan Sankaranarayanan, Sundarrajan Thirugnanasambandam, Jothieswari Dhamotharan, Dhanalakshmi Mohanradja and Ponnurengam Malliappan Sivakumar

Acta Tropica, 2024, 260, 107460
DOI: 10.1016/j.actatropica.2024.107460

Exploring diverse frontiers: Advancements of bioactive 4-aminoquinoline-based molecular hybrids in targeted therapeutics and beyond

Lekkala Ravindar, Siti Aishah Hasbullah, K.P. Rakesh, Saki Raheem, Hani Kartini Agustar, Norzila Ismail, Lau Yee Ling and Nurul Izzaty Hassan

European Journal of Medicinal Chemistry, 2024, 264, 116043
DOI: 10.1016/j.ejmech.2023.116043

Ionic copolymer-modified hexagonal carbon nitride tube as a high-performance catalyst for regioselective synthesis of hexahydroquinoline frameworks

Sara Shafaati, Javad Safaei-Ghomi and Zahra Elyasi

Colloids and Surfaces A: Physicochemical and Engineering Aspects, 2024, 699, 134589
DOI: 10.1016/j.colsurfa.2024.134589

Biannual Account of Anti‐malarial Agents reported in 2021 and 2022: A Comprehensive Coverage

Tejas M. Dhameliya, Diya S. Patel, Deepika Kathuria, Maitri B. Shah, Akshada S. Dabhade, Hetvi S. Dave, Nidhi C. Lad, Amit Z. Chaudhari, Shahnaz Alom, Vivek K. Vyas and Hardik G. Bhatt

ChemistrySelect, 2024, 9
DOI: 10.1002/slct.202303982

In-Silico exploration: Unraveling the anti-cancer potential of 8-Nitroquinoline hydrazides

Sentamil Selvi Ramasamy, Kaviyarasu Adhigaman, Vandana Nandakumar, Amsaveni Sundarasamy, Sundharrajan Jagadeesan, M. Saravanakumar, Jan Grzegorz Malecki, Nalini Easwaran and Suresh Thangaraj

Journal of Molecular Structure, 2025, 1321, 140218
DOI: 10.1016/j.molstruc.2024.140218

A review on quinolines: New green synthetic methods and bioactive potential

Laura M. Ferreira, Pilar García-García, Pablo A. García and María Ángeles Castro

European Journal of Pharmaceutical Sciences, 2025, 209, 107097
DOI: 10.1016/j.ejps.2025.107097

8-Quinoline-oxadiazole ethanone and acetamide hybrids as potential dual HIV-1 entry and mycobacterium tuberculosis inhibitors

Chakes Mashaba, Darian Naidu, Mabuatsela V. Maphoru, Oluwatoba E. Oyeneyin, Hogantharanni Govender, Sibusiso Senzani, Nompumelelo P. Mkhwanazi and Matshawandile Tukulula

Scientific African, 2025, 30, e03100
DOI: 10.1016/j.sciaf.2025.e03100

Recent developments in antimalarial activities of 4-aminoquinoline derivatives

Lekkala Ravindar, Siti Aishah Hasbullah, K.P. Rakesh and Nurul Izzaty Hassan

European Journal of Medicinal Chemistry, 2023, 256, 115458
DOI: 10.1016/j.ejmech.2023.115458

Recent Updates on Interaction Studies and Drug Delivery of Antimalarials with Serum Albumin Proteins

Kashish Azeem, Iram Irfan, Qudsia Rashid, Shailja Singh, Rajan Patel and Mohammad Abid

CMC, 2024, 31, 3925
DOI: 10.2174/0929867330666230509121931