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Fatai Afolabi, Wided Souissi, Guillaume Rivière, Clément Lemaitre, S. Mark Roe, Neil Crickmore and Eddy M. E. Viseux

Dalton Trans., 2018, 47, 15338
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Mechanochemical preparation of strongly emissive monosubstituted triarylphosphane gold(i) compounds activated by hydrogen bonding driven aggregations

Lorenzo Luciani, Nicola Sargentoni, Claudia Graiff, Miguel Monge, María Rodríguez-Castillo, José M. López-de-Luzuriaga and Rossana Galassi

RSC Adv., 2023, 13, 25425
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Stabilization of the cyclodecadiene derivative isofuranodiene by silver (I) coordination. Mechanistic and biological aspects

Filippo Maggi, Fabrizio Papa, Stefania Pucciarelli, Massimo Bramucci, Luana Quassinti, Luciano Barboni, Diego Dal Ben, Anna Teresa Ramadori, Claudia Graiff and Rossana Galassi

Fitoterapia, 2017, 117, 52
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A trigonal coordination of Au(I) phosphane complexes stabilized by O–H⋯X (X = Cl–, Br–, I–) interactions

Petra Gründlinger, Cezarina Cela Mardare, Thorsten Wagner and Uwe Monkowius

Monatsh Chem, 2021, 152, 1201
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An Insight into Synthetic Strategies and Recent Developments of Dihydrofolate Reductase Inhibitors

Pooja Chawla, Ghanshyam Teli, Rupinder Kaur Gill and Raj Kumar Narang

ChemistrySelect, 2021, 6, 12101
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Gold metalation of proteins: Structural studies

Anna Giorgio and Antonello Merlino

Coordination Chemistry Reviews, 2020, 407, 213175
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Biological Activity of NHC-Gold-Alkynyl Complexes Derived from 3-Hydroxyflavones

Inés Mármol, Javier Quero, Paula Azcárate, Elena Atrián-Blasco, Carla Ramos, Joana Santos, María Concepción Gimeno, María Jesús Rodríguez-Yoldi and Elena Cerrada

Pharmaceutics, 2022, 14, 2064
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DHFR Inhibitors: Reading the Past for Discovering Novel Anticancer Agents

Maria Valeria Raimondi, Ornella Randazzo, Mery La Franca, Giampaolo Barone, Elisa Vignoni, Daniela Rossi and Simona Collina

Molecules, 2019, 24, 1140
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Statistical Coupling Analysis Predicts Correlated Motions in Dihydrofolate Reductase

Thomas L. Kalmer, Christine Mae F. Ancajas, Cameron I. Cohen, Jade M. McDaniel, Abiodun S. Oyedele, Hannah L. Thirman and Allison S. Walker

J. Phys. Chem. B, 2024, 128, 10373
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Identification of natural DHFR inhibitors in MRSA strains: Structure-based drug design study

Gagandeep Singh, Hemant Soni, Smriti Tandon, Vijay Kumar, Gajji Babu, Vandana Gupta and Pratima Chaudhuri (Chattopadhyay)

Results in Chemistry, 2022, 4, 100292
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Breast Cancer Treatment: The Case of Gold(I)-Based Compounds as a Promising Class of Bioactive Molecules

Rossana Galassi, Lorenzo Luciani, Junbiao Wang, Silvia Vincenzetti, Lishan Cui, Augusto Amici, Stefania Pucciarelli and Cristina Marchini

Biomolecules, 2022, 12, 80
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Dissociative electron attachment to gold(I)-based compounds: 4,5-dichloro-1,3-diethyl-imidazolylidene trifluoromethyl gold(I)

Maria Pintea, Nigel Mason, Anna Peiró-Franch, Ewan Clark, Kushal Samanta, Cristiano Glessi, Inga Lena Schmidtke and Thomas Luxford

Front. Chem., 2023, 11
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Multi-Targeted Anticancer Activity of Imidazolate Phosphane Gold(I) Compounds by Inhibition of DHFR and TrxR in Breast Cancer Cells

Rossana Galassi, Lorenzo Luciani, Valentina Gambini, Silvia Vincenzetti, Giulio Lupidi, Augusto Amici, Cristina Marchini, Junbiao Wang and Stefania Pucciarelli

Front. Chem., 2021, 8
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In vitro and in vivo studies of gold(I) azolate/phosphane complexes for the treatment of basal like breast cancer

Valentina Gambini, Martina Tilio, Eunice Wairimu Maina, Cristina Andreani, Caterina Bartolacci, Junbiao Wang, Manuela Iezzi, Stefano Ferraro, Anna Teresa Ramadori, Oumarou Camille Simon, Stefania Pucciarelli, Guojun Wu, Q. Ping Dou, Cristina Marchini, Rossana Galassi and Augusto Amici

European Journal of Medicinal Chemistry, 2018, 155, 418
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The Anti-Multidrug-Resistant Acinetobacter baumannii Study on 1,3-diamino-7H-pyrrolo[3,2-f]quinazoline Compounds

Han Wu, Hongtong Chen, Jungan Zhang, Xinxin Hu, Chunyang Xie, Weiting Cao, Ziqi Zhao, Zengshuo Xiao, Yixin Ren, Luyao Dong, Peiyi Sun, Xuefu You, Xinyi Yang, Wei Hong and Hao Wang

Molecules, 2022, 27, 8609
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Dihydrofolate reductase inhibitors: patent landscape and phases of clinical development (2001–2021)

Kavita Bhagat, Nitish Kumar, Harmandeep Kaur Gulati, Aanchal Sharma, Amandeep Kaur, Jatinder Vir Singh, Harbinder Singh and Preet Mohinder Singh Bedi

Expert Opinion on Therapeutic Patents, 2022, 32, 1079
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Studies on the Interaction between Poly-Phosphane Gold(I) Complexes and Dihydrofolate Reductase: An Interplay with Nicotinamide Adenine Dinucleotide Cofactor

Stefania Pucciarelli, Silvia Vincenzetti, Massimo Ricciutelli, Oumarou Camille Simon, Anna Teresa Ramadori, Lorenzo Luciani and Rossana Galassi

IJMS, 2019, 20, 1802
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Synchrotron Characterization of Hexagonal and Cubic Lipidic Phases Loaded with Azolate/Phosphane Gold(I) Compounds: A New Approach to the Uploading of Gold(I)-Based Drugs

Paola Astolfi, Michela Pisani, Elisabetta Giorgini, Barbara Rossi, Alessandro Damin, Francesco Vita, Oriano Francescangeli, Lorenzo Luciani and Rossana Galassi

Nanomaterials, 2020, 10, 1851
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Reactivity of (3‐(4‐Fluorophenyl)oxyran‐2‐yl)(naphthalene‐2‐yl)methanone Toward Some Nucleophiles for Preparing Promising Agents with Antimicrobial and Antioxidant Activities

Hemat S. Khalaf, Eman R. Kotb, Nayera A. M. Abdelwahed, Mohamad T. Abdelrahman and Ahmed H. Shamroukh

ChemistrySelect, 2024, 9
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Development of QSAR Models and Web Applications for Predicting hDHFR Inhibitor Bioactivity Using Machine Learning

Ibrahim Maattallaoui, Mahamadou Sakho, Abdellah Maatallaoui, Enrique Barrajón-Catalán and Noureddine Aouad

Molecules, 2025, 30, 4618
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