Synthesis and anticancer potential of glycosides

Shaukat Ali, Gul Rukh, Hanan A. Ogaly, Rahaf Ajaj, Abdur Rauf and Syed Adnan Ali Shah

RSC Adv., 2025, 15, 51054
DOI: 10.1039/D5RA07626A

Design, synthesis and in vitro evaluation of coumarin–imidazo[1,2-a]pyridine derivatives against cancer induced osteoporosis

Koneni V. Sashidhara, L. Ravithej Singh, Dharmendra Choudhary, Ashutosh Arun, Sampa Gupta, Sulekha Adhikary, Gopala Reddy Palnati, Rituraj Konwar and Ritu Trivedi

RSC Adv., 2016, 6, 80037
DOI: 10.1039/C6RA15674F

Development of Novel Pt(IV)-Carbohydrate Derivatives as Targeted Anticancer Agents against Osteosarcoma

Eoin Moynihan, Silvia Panseri, Giada Bassi, Arianna Rossi, Elisabetta Campodoni, Eithne Dempsey, Monica Montesi, Trinidad Velasco-Torrijos and Diego Montagner

IJMS, 2023, 24, 6028
DOI: 10.3390/ijms24076028

Carbohydrates: Potential Sweet Tools Against Cancer

Antonio Franconetti, Óscar López and José G. Fernandez-Bolanos

CMC, 2020, 27, 1206
DOI: 10.2174/0929867325666180719114150

Pyranocarbazole derivatives as potent anti-cancer agents triggering tubulin polymerization stabilization induced activation of caspase-dependent apoptosis and downregulation of Akt/mTOR in breast cancer cells

Om P.S. Patel, Ashutosh Arun, Pankaj K. Singh, Deepika Saini, Sharanbasappa Shrimant Karade, Manish K. Chourasia, Rituraj Konwar and Prem P. Yadav

European Journal of Medicinal Chemistry, 2019, 167, 226
DOI: 10.1016/j.ejmech.2019.02.003

Eudesmic acid-polyoxomolybdate organo-conjugate as novel anticancer agent

Maryam Ramezani-Aliakbari, Azim Soltanabadi, Hojjat Sadeghi-aliabadi, Jaleh Varshosaz, Bahram Yadollahi, Farshid Hassanzadeh and Mahboubeh Rostami

Journal of Molecular Structure, 2021, 1240, 130612
DOI: 10.1016/j.molstruc.2021.130612

Cucurbitacin B inhibits breast cancer metastasis and angiogenesis through VEGF-mediated suppression of FAK/MMP-9 signaling axis

Sonam Sinha, Sajid Khan, Samriddhi Shukla, Amar Deep Lakra, Sudhir Kumar, Gunjan Das, Rakesh Maurya and Syed Musthapa Meeran

The International Journal of Biochemistry & Cell Biology, 2016, 77, 41
DOI: 10.1016/j.biocel.2016.05.014

Anti-colon cancer activity of Murraya koenigii leaves is due to constituent murrayazoline and O-methylmurrayamine A induced mTOR/AKT downregulation and mitochondrial apoptosis

Ashutosh Arun, Om P.S. Patel, Deepika Saini, Prem P. Yadav and Rituraj Konwar

Biomedicine & Pharmacotherapy, 2017, 93, 510
DOI: 10.1016/j.biopha.2017.06.065

Base‐Free Copper‐Catalyzed Azide‐Alkyne Click Cycloadditions (CuAAc) in Natural Deep Eutectic Solvents as Green and Catalytic Reaction Media**

Salvatore Vincenzo Giofrè, Matteo Tiecco, Angelo Ferlazzo, Roberto Romeo, Gianluca Ciancaleoni, Raimondo Germani and Daniela Iannazzo

Eur J Org Chem, 2021, 2021, 4777
DOI: 10.1002/ejoc.202100698

New piperidine derivativeDTPEPacts as dual‐acting anti‐breast cancer agent by targetingERα and downregulatingPI3K/Akt‐PKCα leading to caspase‐dependent apoptosis

A. Arun, M.I. Ansari, P. Popli, S. Jaiswal, A.K. Mishra, A. Dwivedi, K. Hajela and R. Konwar

Cell Proliferation, 2018, 51
DOI: 10.1111/cpr.12501

Carbohydrate derivatives fight against malaria parasite as anti-plasmodial agents

Kartikey Singh and Rama Pati Tripathi

Carbohydrate Research, 2023, 531, 108887
DOI: 10.1016/j.carres.2023.108887

Synthesis of isatin based N1-alkylated 3-β-C-glycoconjugated-oxopropylidene oxindoles as potent antiplasmodial agents

Ravi Kumar Thakur, Prince Joshi, Kapil Upadhyaya, Kartikey Singh, Gaurav Sharma, Sanjeev K. Shukla, Renu Tripathi and Rama Pati Tripathi

European Journal of Medicinal Chemistry, 2019, 162, 448
DOI: 10.1016/j.ejmech.2018.11.008

Emergence of Fluorescent Glycodots for Biomedical Applications

Kartikey Singh, Tuhin Mandal, Umesh Pratap Pandey and Vikram Singh

ACS Biomater. Sci. Eng., 2025, 11, 742
DOI: 10.1021/acsbiomaterials.4c02018

Discovery of 3,4,6‐Triaryl‐2‐pyridones as Potential Anticancer Agents that Promote ROS‐Independent Mitochondrial‐Mediated Apoptosis in Human Breast Carcinoma Cells

Mohammad Imran Ansari, Ashutosh Arun, Mohammad Kamil Hussain, Rituraj Konwar and Kanchan Hajela

ChemistrySelect, 2016, 1, 4255
DOI: 10.1002/slct.201600893

Design, Synthesis and Evaluation of 2,4‐Diaminoquinazoline Derivatives as Potential Tubulin Polymerization Inhibitors

Frida S. Herrera‐Vázquez, Félix Matadamas‐Martínez, Rodrigo Aguayo‐Ortiz, Laura Dominguez, Teresa Ramírez‐Apan, Lilián Yépez‐Mulia and Francisco Hernández‐Luis

ChemMedChem, 2020, 15, 1802
DOI: 10.1002/cmdc.202000185

Synthesis of Gallic Acid Analogs as Histamine and Pro-Inflammatory Cytokine Inhibitors for Treatment of Mast Cell-Mediated Allergic Inflammation

Xiang Fei, In-Gyu Je, Tae-Yong Shin, Sang-Hyun Kim and Seung-Yong Seo

Molecules, 2017, 22, 898
DOI: 10.3390/molecules22060898

The Goldilocks Principle in Phase Labeling. Minimalist and Orthogonal Phase Tagging for Chromatography-Free Mitsunobu Reaction

Mariann Szigeti, Zoltán Dobi and Tibor Soós

J. Org. Chem., 2018, 83, 2869
DOI: 10.1021/acs.joc.8b00014

Cu(I)-Catalyzed Click Chemistry in Glycoscience and Their Diverse Applications

Anand K. Agrahari, Priyanka Bose, Manoj K. Jaiswal, Sanchayita Rajkhowa, Anoop S. Singh, Srinivas Hotha, Nidhi Mishra and Vinod K. Tiwari

Chem. Rev., 2021, 121, 7638
DOI: 10.1021/acs.chemrev.0c00920

Prevention of articular cartilage degeneration in a rat model of monosodium iodoacetate induced osteoarthritis by oral treatment with Withaferin A

Dharmendra Choudhary, Sulekha Adhikary, Naseer Ahmad, Priyanka Kothari, Ashwni Verma, Prabodh Kumar Trivedi, Prabhat Ranjan Mishra and Ritu Trivedi

Biomedicine & Pharmacotherapy, 2018, 99, 151
DOI: 10.1016/j.biopha.2017.12.113

Click Pt(IV)-Carbohydrates Pro-Drugs for Treatment of Osteosarcoma

Eoin Moynihan, Giada Bassi, Andrea Ruffini, Silvia Panseri, Monica Montesi, Trinidad Velasco-Torrijos and Diego Montagner

Front. Chem., 2021, 9
DOI: 10.3389/fchem.2021.795997

Synthesis of 1,2,3-Triazole and Tetrazole Appended Glycoconjugates Based on 3,6-Anhydroglucofuranose via Click Reaction

Susanta Das, Ratul Hore, Sayanta Paria, Gillian Dcosta, Mrinalkanti Kundu and Joykrishna Maity

ACS Omega, 2025, 10, 39615
DOI: 10.1021/acsomega.5c02564

Organocatalyzed synthesis of 2-deoxyglycosyl azides: Application in 1,2,3-triazole linked 2-deoxyglycosides

Vivek Kumar Sharma and Rima Thakur

Carbohydrate Research, 2025, 558, 109668
DOI: 10.1016/j.carres.2025.109668

In Search of Effective Anticancer Agents—Novel Sugar Esters Based on Polyhydroxyalkanoate Monomers

Wojciech Snoch, Dawid Wnuk, Tomasz Witko, Jakub Staroń, Andrzej J. Bojarski, Ewelina Jarek, Francisco J. Plou and Maciej Guzik

IJMS, 2021, 22, 7238
DOI: 10.3390/ijms22137238

Structural Bias Effect On Azidation at C-1 and C-2 of Alkyl-3,6-anhydro-d-hexofuranosides: Synthetic Approach to Natural Products and Derivatives

Ratul Hore, Koushik Bit, Rajatava Pan, Tapas Halder, Susanta Das, Subhadip Sett, Tapas Bera, Abhinash Subba and Joykrishna Maity

ACS Omega, 2025, 10, 42999
DOI: 10.1021/acsomega.5c05437

New orally active DNA minor groove binding small molecule CT‐1 acts against breast cancer by targeting tumor DNA damage leading to p53‐dependent apoptosis

Karan Singh Saini, Hamidullah, Raghib Ashraf, Dhanaraju Mandalapu, Sharmistha Das, Mohd Quadir Siddiqui, Sonam Dwivedi, Jayanta Sarkar, Vishnu Lal Sharma and Rituraj Konwar

Molecular Carcinogenesis, 2017, 56, 1266
DOI: 10.1002/mc.22588

Studies on phenothiazines: New microtubule-interacting compounds with phenothiazine A-ring as potent antineoplastic agents

Alina Ghinet, Iuliana-Monica Moise, Benoît Rigo, Germain Homerin, Amaury Farce, Joëlle Dubois and Elena Bîcu

Bioorganic & Medicinal Chemistry, 2016, 24, 2307
DOI: 10.1016/j.bmc.2016.04.001

Antifibrotic effects of gallic acid on hepatic stellate cells: In vitro and in vivo mechanistic study

Naglaa M. El-Lakkany, Walaa H. El-Maadawy, Sayed H. Seif el-Din, Samira Saleh, Marwa M. Safar, Shahira M. Ezzat, Salwa H. Mohamed, Sanaa S. Botros, Zeinab Demerdash and Olfat A. Hammam

Journal of Traditional and Complementary Medicine, 2019, 9, 45
DOI: 10.1016/j.jtcme.2018.01.010

Design and Synthesis of New Tubulin Polymerization Inhibitors Inspired from Combretastatin A‐4: An Anticancer Agent

Akanksha Sharma, Doddabasappa Talimarada, Umesh Prasad Yadav, Nidhi Singh, A. Sudharshan Reddy, Debojyoti Bag, Krishna Biswas, Amit Baidya, Asha N Borale, Dhananjay Shinde, Sandeep Singh and Harish Holla

ChemistrySelect, 2020, 5, 11560
DOI: 10.1002/slct.202003170