Insights into phosphatase-activated chemical defense in a marine sponge holobiont

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RSC Chem. Biol., 2021, 2, 1600
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Cytotoxic and antitumor peptides as novel chemotherapeutics

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Synthesis, modeling, and biological evaluation of anti-tubulin indole-substituted furanones

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Gatorbulin-1, a distinct cyclodepsipeptide chemotype, targets a seventh tubulin pharmacological site

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Plant-Derived Anti-Cancer Therapeutics and Biopharmaceuticals

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Do Lipid-based Nanoparticles Hold Promise for Advancing the Clinical Translation of Anticancer Alkaloids?

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Cancers, 2021, 13, 5346
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Toward a Template for Synthetic Actin-Targeting Macrolide Analogues That Inhibit Cancer Cell Invasiveness

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Synthesis and Biological Evaluation of Novel 2-Aroyl Benzofuran-Based Hydroxamic Acids as Antimicrotubule Agents

Elena Mariotto, Martina Canton, Chiara Marchioro, Andrea Brancale, Ernest Hamel, Katia Varani, Fabrizio Vincenzi, Tiziano De Ventura, Chiara Padroni, Giampietro Viola and Romeo Romagnoli

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Investigating impacts of the mycothiazole chemotype as a chemical probe for the study of mitochondrial function and aging

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Cytochalasin Q exerts anti-melanoma effect by inhibiting creatine kinase B

Yi Lu, Peng Zhang, Hongdan Chen, Qingyi Tong, Jia Wang, Qing Li, Cheng Tian, Jian Yang, Senlin Li, Zijun Zhang, Huimin Yuan and Ming Xiang

Toxicology and Applied Pharmacology, 2022, 441, 115971
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Marine Pharmacology in 2019–2021: Marine Compounds with Antibacterial, Antidiabetic, Antifungal, Anti-Inflammatory, Antiprotozoal, Antituberculosis and Antiviral Activities; Affecting the Immune and Nervous Systems, and Other Miscellaneous Mechanisms of Action

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Lead optimization of novel quinolone chalcone compounds by a structure–activity relationship (SAR) study to increase efficacy and metabolic stability

James Knockleby, Aïcha Dede Djigo, Indeewari Kalhari Lindamulage, Chandrabose Karthikeyan, Piyush Trivedi and Hoyun Lee

Sci Rep, 2021, 11
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Is a Modified Actin the Key to Toxin Resistance in the Nudibranch Chromodoris? A Biochemical and Molecular Approach

Cora Hertzer, Nani Undap, Adelfia Papu, Dhaka Bhandari, Stefan Aatz, Stefan Kehraus, Fontje Kaligis, Robert Bara, Till Schäberle, Heike Wägele and Gabriele König

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Fluoroindole chalcone analogues targeting the colchicine binding site of tubulin for colorectal oncotherapy

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European Journal of Medicinal Chemistry, 2023, 257, 115540
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Therapeutic strategies to overcome taxane resistance in cancer

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βIII-tubulin overexpression in cancer: Causes, consequences, and potential therapies

Arun Kanakkanthara and John H. Miller

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Alterations to the broad-spectrum formin inhibitor SMIFH2 modulate potency but not specificity

Marina Orman, Maya Landis, Aisha Oza, Deepika Nambiar, Joana Gjeci, Kristen Song, Vivian Huang, Amanda Klestzick, Carla Hachicho, Su Qing Liu, Judith M. Kamm, Francesca Bartolini, Jean J. Vadakkan, Christian M. Rojas and Christina L. Vizcarra

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Actin-Interacting Amphidinolides: Syntheses and Mechanisms of Action of Amphidinolides X, J, and K

Anna M. Costa

Molecules, 2023, 28, 5249
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Tubulysin Production by the Dead Cells of Archangium gephyra KYC5002

Seohui Park, Chaehyeon Park, Yujin Ka and Kyungyun Cho

J Microbiol., 2024, 62, 463
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Probing a distinct druggable tubulin binding site with gatorbulins 1–7, their metabolic and physicochemical properties, and pharmacological consequences

Qi-Yin Chen, Ranjala Ratnayake, Rafael Hortigüela, Gustavo M. Seabra, Michael D. Cameron, J. Fernando Díaz, María Ángela Oliva and Hendrik Luesch

Bioorganic & Medicinal Chemistry, 2023, 95, 117506
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Intermediate filaments and their associated molecules

Jing Gao and Fumihiko Nakamura

J Biomed Res, 2025, 39, 242
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