Maria Letizia Ciavatta, Florence Lefranc, Marianna Carbone, Ernesto Mollo, Margherita Gavagnin, Tania Betancourt, Ramesh Dasari, Alexander Kornienko and Robert Kiss

Medicinal Research Reviews, 2017, 37, 702
DOI: 10.1002/med.21423

Kinetic Resolution of Racemic Aldehydes through Asymmetric Allenoate γ-Addition: Synthesis of (+)-Xylogiblactone A

Saehansaem Park, Gyungah Pak, Changhwa Oh, Jieun Lee, Jimin Kim and Chan-Mo Yu

Org. Lett., 2019, 21, 7660
DOI: 10.1021/acs.orglett.9b02982

Development of a Concise Synthesis of (+)-Ingenol

Steven J. McKerrall, Lars Jørgensen, Christian A. Kuttruff, Felix Ungeheuer and Phil S. Baran

J. Am. Chem. Soc., 2014, 136, 5799
DOI: 10.1021/ja501881p

Total Syntheses of (−)‐Minovincine and (−)‐Aspidofractinine through a Sequence of Cascade Reactions

Szilárd Varga, Péter Angyal, Gábor Martin, Orsolya Egyed, Tamás Holczbauer and Tibor Soós

Angew Chem Int Ed, 2020, 59, 13547
DOI: 10.1002/anie.202004769

A Personal Perspective on Organic Synthesis: Past, Present, and Future

David Y.‐K. Chen

Israel Journal of Chemistry, 2018, 58, 85
DOI: 10.1002/ijch.201700113

In Pursuit of Synthetic Efficiency: Convergent Approaches

Yang Gao and Dawei Ma

Acc. Chem. Res., 2021, 54, 569
DOI: 10.1021/acs.accounts.0c00727

Fighting evolution with chemical synthesis

Ming Yan and Phil S. Baran

Nature, 2016, 533, 326
DOI: 10.1038/533326a

Photochemical Approaches to Complex Chemotypes: Applications in Natural Product Synthesis

Markus D. Kärkäs, John A. Porco and Corey R. J. Stephenson

Chem. Rev., 2016, 116, 9683
DOI: 10.1021/acs.chemrev.5b00760

An Efficient and Scalable “Second Generation” Total Synthesis of the Marine Polyketide Limaol Endowed with Antiparasitic Activity

Stephan N. Hess and Alois Fürstner

Chemistry A European J, 2024, 30
DOI: 10.1002/chem.202401429

A Systematic Review of Recently Reported Marine Derived Natural Product Kinase Inhibitors

Te Li, Ning Wang, Ting Zhang, Bin Zhang, Thavarool P. Sajeevan, Valsamma Joseph, Lorene Armstrong, Shan He, Xiaojun Yan and C. Benjamin Naman

Marine Drugs, 2019, 17, 493
DOI: 10.3390/md17090493

Natural products on demand

Lawrence G. Hamann

Nature Chem, 2014, 6, 460
DOI: 10.1038/nchem.1964

Total Synthesis and Stereochemical Assignment of Delavatine A: Rh-Catalyzed Asymmetric Hydrogenation of Indene-Type Tetrasubstituted Olefins and Kinetic Resolution through Pd-Catalyzed Triflamide-Directed C–H Olefination

Zhongyin Zhang, Jinxin Wang, Jian Li, Fan Yang, Guodu Liu, Wenjun Tang, Weiwei He, Jian-Jun Fu, Yun-Heng Shen, Ang Li and Wei-Dong Zhang

J. Am. Chem. Soc., 2017, 139, 5558
DOI: 10.1021/jacs.7b01718

Scalable Total Synthesis of Acremolactone B

Mengyu Ba, Fengqi He, Lu Ren, William G. Whittingham, Peng Yang and Ang Li

Angew Chem Int Ed, 2024, 63
DOI: 10.1002/anie.202314800

Multi-gram scale synthesis of hunanamycin A, an antibiotic natural product from the marine source

Rahul D. Shingare, Sa ada Farhana and D. Srinivasa Reddy

Tetrahedron Letters, 2016, 57, 3662
DOI: 10.1016/j.tetlet.2016.07.003

Catalyst-Directed Diastereoselective Isomerization of Allylic Alcohols for the Stereoselective Construction of C(20) in Steroid Side Chains: Scope and Topological Diversification

Houhua Li and Clément Mazet

J. Am. Chem. Soc., 2015, 137, 10720
DOI: 10.1021/jacs.5b06281

Harnessing natural product assembly lines: structure, promiscuity, and engineering

Christopher C Ladner and Gavin J Williams

Journal of Industrial Microbiology and Biotechnology, 2016, 43, 371
DOI: 10.1007/s10295-015-1704-8

Scalable Total Synthesis of rac‐Jungermannenones B and C

Weilong Liu, Houhua Li, Pei‐Jun Cai, Zhen Wang, Zhi‐Xiang Yu and Xiaoguang Lei

Angew Chem Int Ed, 2016, 55, 3112
DOI: 10.1002/anie.201511659

Bioinspired Skeletal Reorganization Approach for the Synthesis of Steroid Natural Products

Yu Wang and Jinghan Gui

Acc. Chem. Res., 2024, 57, 568
DOI: 10.1021/acs.accounts.3c00716

Synthesis of 9,11-Secosteroids Pinnisterol E, Glaciasterol B, and 6-Keto-aplidiasterol B

Yinlong Miao, Xinghui Li, Mengqing Zhang, Huafang Fan and Jinghan Gui

Org. Lett., 2022, 24, 1684
DOI: 10.1021/acs.orglett.2c00281

Twelve‐membered macrolactones: privileged scaffolds for the development of new therapeutics

Richard S. Brzozowski and William M. Wuest

Chem Biol Drug Des, 2017, 89, 169
DOI: 10.1111/cbdd.12783

Highly Enantioselective Acylation of Acyclic Meso 1,3-Diols through Synergistic Isothiourea-Catalyzed Desymmetrization/Chiroablative Kinetic Resolution

Jérémy Merad, Prashant Borkar, Tracy Bouyon Yenda, Christèle Roux, Jean-Marc Pons, Jean-Luc Parrain, Olivier Chuzel and Cyril Bressy

Org. Lett., 2015, 17, 2118
DOI: 10.1021/acs.orglett.5b00707

Scalable Total Synthesis of rac‐Jungermannenones B and C

Weilong Liu, Houhua Li, Pei‐Jun Cai, Zhen Wang, Zhi‐Xiang Yu and Xiaoguang Lei

Angewandte Chemie, 2016, 128, 3164
DOI: 10.1002/ange.201511659

Total Synthesis of the Euphorbia Diterpenoid Pepluacetal

Meng Liu, Chuanhua Wu, Xingang Xie, Huilin Li and Xuegong She

Angew Chem Int Ed, 2024, 63
DOI: 10.1002/anie.202400943

Highly Efficient Formal [2+2+2] Strategy for the Rapid Construction of Polycyclic Spiroindolines: A Concise Synthesis of 11‐Demethoxy‐16‐epi‐myrtoidine

Jun Zhu, Yu‐Jing Cheng, Xiao‐Kang Kuang, Lijia Wang, Zhong‐Bo Zheng and Yong Tang

Angewandte Chemie, 2016, 128, 9370
DOI: 10.1002/ange.201603991

Navigating the Chiral Pool in the Total Synthesis of Complex Terpene Natural Products

Zachary G. Brill, Matthew L. Condakes, Chi P. Ting and Thomas J. Maimone

Chem. Rev., 2017, 117, 11753
DOI: 10.1021/acs.chemrev.6b00834

Scalable Total Synthesis of Bastimolide A Enabled by Asymmetric Allylborations Catalyzed by Chiral Brønsted Acids

Shigenobu Umemiya, Naoya Shinagawa, Aisuke Fujimoto and Masahiro Terada

JACS Au, 2025, 5, 3052
DOI: 10.1021/jacsau.5c00630

Plant antibacterials: The challenges and opportunities

Tomayo I. Berida, Yemi A. Adekunle, Hannah Dada-Adegbola, Ayoub Kdimy, Sudeshna Roy and Satyajit D. Sarker

Heliyon, 2024, 10, e31145
DOI: 10.1016/j.heliyon.2024.e31145

ChemInform Abstract: Natural Product Synthesis in the Age of Scalability

Christian A. Kuttruff, Martin D. Eastgate and Phil S. Baran

ChemInform, 2014, 45
DOI: 10.1002/chin.201425249

Total Synthesis, Stereochemical Revision, and Biological Reassessment of Mandelalide A: Chemical Mimicry of Intrafamily Relationships

Jens Willwacher, Berit Heggen, Conny Wirtz, Walter Thiel and Alois Fürstner

Chemistry A European J, 2015, 21, 10416
DOI: 10.1002/chem.201501491

Alkynes From Furans: A General Fragmentation Method Applied to the Synthesis of the Proposed Structure of Aglatomin B

Jiachen Deng, Jingjing Wu, Hailong Tian, Jiajing Bao, Yong Shi, Weisheng Tian and Jinghan Gui

Angewandte Chemie, 2018, 130, 3679
DOI: 10.1002/ange.201712365

Scalable Enantioselective Total Synthesis of (−)‐Goniomitine

Huai‐Yu Bin, Ke Wang, Dan Yang, Xiao‐Hui Yang, Jian‐Hua Xie and Qi‐Lin Zhou

Angew Chem Int Ed, 2019, 58, 1174
DOI: 10.1002/anie.201812822

Unified Total Synthesis of Stemoamide-Type Alkaloids by Chemoselective Assembly of Five-Membered Building Blocks

Makoto Yoritate, Yoshito Takahashi, Hayato Tajima, Chisato Ogihara, Takashi Yokoyama, Yasuki Soda, Takeshi Oishi, Takaaki Sato and Noritaka Chida

J. Am. Chem. Soc., 2017, 139, 18386
DOI: 10.1021/jacs.7b10944

A 11‐Steps Total Synthesis of Magellanine through a Gold(I)‐Catalyzed Dehydro Diels–Alder Reaction

Philippe McGee, Geneviève Bétournay, Francis Barabé and Louis Barriault

Angew Chem Int Ed, 2017, 56, 6280
DOI: 10.1002/anie.201611606

Organocatalytic hydroboration of imines, nitriles, and amides using choline-based ionic liquids

Barbara Krupa, Mateusz Nowicki, Jakub Szyling and Jędrzej Walkowiak

Journal of Catalysis, 2025, 451, 116362
DOI: 10.1016/j.jcat.2025.116362

Short Total Synthesis of [15N5]-Cylindrospermopsins from 15NH4Cl Enables Precise Quantification of Freshwater Cyanobacterial Contamination

Artur K. Mailyan, Joanna L. Chen, Weiwei Li, Arturo A. Keller, Shawn M. Sternisha, Brian G. Miller and Armen Zakarian

J. Am. Chem. Soc., 2018, 140, 6027
DOI: 10.1021/jacs.8b03071

Chemo-enzymatic synthesis of natural products and their analogs

Felix Kaspar and Anett Schallmey

Current Opinion in Biotechnology, 2022, 77, 102759
DOI: 10.1016/j.copbio.2022.102759

On Scalability, Synthetic Efficiency, and Convergency

Vittorio Farina

Org. Process Res. Dev., 2025, 29, 979
DOI: 10.1021/acs.oprd.5c00030

Versatile Butenolide Syntheses via a Structure-Oriented C–H Activation Reaction

Yu-Kun Lin, Donghyeon Kim, Yuxin Ouyang and Jin-Quan Yu

J. Am. Chem. Soc., 2025, 147, 26019
DOI: 10.1021/jacs.5c09040

Highly Efficient Formal [2+2+2] Strategy for the Rapid Construction of Polycyclic Spiroindolines: A Concise Synthesis of 11‐Demethoxy‐16‐epi‐myrtoidine

Jun Zhu, Yu‐Jing Cheng, Xiao‐Kang Kuang, Lijia Wang, Zhong‐Bo Zheng and Yong Tang

Angew Chem Int Ed, 2016, 55, 9224
DOI: 10.1002/anie.201603991

Cyanthiwigin Natural Product Core as a Complex Molecular Scaffold for Comparative Late-Stage C–H Functionalization Studies

Kelly E. Kim, Ashley M. Adams, Nicholas D. Chiappini, J. Du Bois and Brian M. Stoltz

J. Org. Chem., 2018, 83, 3023
DOI: 10.1021/acs.joc.7b03291

The Cargill-Type Rearrangement in Natural Product Synthesis

Wen Xun, Deyun Ma, Rimeng Chen, Shaobin Su and Bo Xu

Synthesis, 2025, 57, 2765
DOI: 10.1055/a-2640-7480

Enantioselective Total Syntheses of (+)-Hostmanin A, (−)-Linderol A, (+)-Methyllinderatin and Structural Reassignment of Adunctin E

Dattatraya H. Dethe and Balu D. Dherange

J. Org. Chem., 2015, 80, 4526
DOI: 10.1021/acs.joc.5b00331

Divergent Strategy in Natural Product Total Synthesis

Lei Li, Zhuang Chen, Xiwu Zhang and Yanxing Jia

Chem. Rev., 2018, 118, 3752
DOI: 10.1021/acs.chemrev.7b00653

Unraveling Plant Natural Chemical Diversity for Drug Discovery Purposes

Emmanuelle Lautié, Olivier Russo, Pierre Ducrot and Jean A. Boutin

Front. Pharmacol., 2020, 11
DOI: 10.3389/fphar.2020.00397

Convergent total synthesis of (+)-calcipotriol: A scalable, modular approach to vitamin D analogs

Jieyu Gu, Kevin X. Rodriguez, Yuzuru Kanda, Shenghua Yang, Michal Ociepa, Henrik Wilke, Arteen V. Abrishami, Lars Jørgensen, Tine Skak-Nielsen, Jason S. Chen and Phil S. Baran

Proc. Natl. Acad. Sci. U.S.A., 2022, 119
DOI: 10.1073/pnas.2200814119

Scalable Total Synthesis of Acremolactone B

Mengyu Ba, Fengqi He, Lu Ren, William G. Whittingham, Peng Yang and Ang Li

Angewandte Chemie, 2024, 136
DOI: 10.1002/ange.202314800

Tandem organocatalytic approach to C28–C35 fragment of eribulin mesylate

Lahu N. Chavan, Rambabu Chegondi and Srivari Chandrasekhar

Tetrahedron Letters, 2015, 56, 4286
DOI: 10.1016/j.tetlet.2015.05.075

Natural Products as Sources of New Drugs from 1981 to 2014

David J. Newman and Gordon M. Cragg

J. Nat. Prod., 2016, 79, 629
DOI: 10.1021/acs.jnatprod.5b01055

Intramolecular Electrochemical Oxybromination of Olefins for the Synthesis of Isoxazolines in Batch and Continuous Flow

Ajit Prabhakar Kale, Pavlo Nikolaienko, Kristina Smirnova and Magnus Rueping

Eur J Org Chem, 2021, 2021, 3496
DOI: 10.1002/ejoc.202100640

Reactivity tamed one bond at a time

Matthew T. Villaume and Phil S. Baran

Nature, 2014, 513, 324
DOI: 10.1038/513324a

Emerging R and D Law: The Nagoya Protocol and Its Implications for Researchers

Geoff Burton and Elizabeth A. Evans-Illidge

ACS Chem. Biol., 2014, 9, 588
DOI: 10.1021/cb500045t

Combining the best of both worlds: radical-based divergent total synthesis

Kyriaki Gennaiou, Antonios Kelesidis, Maria Kourgiantaki and Alexandros L Zografos

Beilstein J. Org. Chem., 2023, 19, 1
DOI: 10.3762/bjoc.19.1

Advances in the E → Z Isomerization of Alkenes Using Small Molecule Photocatalysts

Tomáš Neveselý, Max Wienhold, John J. Molloy and Ryan Gilmour

Chem. Rev., 2022, 122, 2650
DOI: 10.1021/acs.chemrev.1c00324

Concise Total Synthesis of Dehaloperophoramidine

Kirill Popov, Anita Hoang and Peter Somfai

Angew Chem Int Ed, 2016, 55, 1801
DOI: 10.1002/anie.201510661

My 50-Plus Years of Academic Research Collaborations with Industry. A Retrospective

Stephen Hanessian

J. Org. Chem., 2024, 89, 9147
DOI: 10.1021/acs.joc.4c00652

Modular Approach for the Synthesis and Bioactivity Profiling of 8,8′-Biflavones

Moritz K. T. Klischan, Flaminia Mazzone, Lena Berning, Julian Greb, Max Schlamkow, Mona Haase, Wolfgang Frey, Björn Stork, Klaus Pfeffer and Jörg Pietruszka

ACS Omega, 2023, 8, 41816
DOI: 10.1021/acsomega.3c06503

Fixing the Unfixable: The Art of Optimizing Natural Products for Human Medicine

Audrey E. Yñigez-Gutierrez and Brian O. Bachmann

J. Med. Chem., 2019, 62, 8412
DOI: 10.1021/acs.jmedchem.9b00246

Total Synthesis and Stereochemical Assignment of Talaroconvolutin A and Talarofuranone: Gram‐scale Synthesis of Ferroptosis Inducer Talaroconvolutin A

Ming Yao, Wei Yang, Jing Li, Chengyun Huang, Jin Fang, Sulu Qin, Shuzhi Liu and Xiaolong Yang

Chin. J. Chem., 2024, 42, 1509
DOI: 10.1002/cjoc.202400061

Reusable directing groups [8-aminoquinoline, picolinamide, sulfoximine] in C(sp3)–H bond activation: present and future

Raja K. Rit, M. Ramu Yadav, Koushik Ghosh and Akhila K. Sahoo

Tetrahedron, 2015, 71, 4450
DOI: 10.1016/j.tet.2015.03.085

Five-Step Synthesis of Yaequinolones J1 and J2

Johannes Schwan, Merlin Kleoff, Philipp Heretsch and Mathias Christmann

Org. Lett., 2020, 22, 675
DOI: 10.1021/acs.orglett.9b04455

Alkynes From Furans: A General Fragmentation Method Applied to the Synthesis of the Proposed Structure of Aglatomin B

Jiachen Deng, Jingjing Wu, Hailong Tian, Jiajing Bao, Yong Shi, Weisheng Tian and Jinghan Gui

Angew Chem Int Ed, 2018, 57, 3617
DOI: 10.1002/anie.201712365

Synthesis, Molecular Editing, and Biological Assessment of the Potent Cytotoxin Leiodermatolide

Damien Mailhol, Jens Willwacher, Nina Kausch-Busies, Elizabeth E. Rubitski, Zhanna Sobol, Maik Schuler, My-Hanh Lam, Sylvia Musto, Frank Loganzo, Andreas Maderna and Alois Fürstner

J. Am. Chem. Soc., 2014, 136, 15719
DOI: 10.1021/ja508846g

«Synthesis: Science or Technology?» A Few Comments from an Old‐timer

Léon Ghosez

Israel Journal of Chemistry, 2018, 58, 127
DOI: 10.1002/ijch.201700139

An Enantioconvergent and Concise Synthesis of Lasonolide A

Lin Yang, Zuming Lin, Shunjie Shao, Qian Zhao and Ran Hong

Angewandte Chemie, 2018, 130, 16432
DOI: 10.1002/ange.201811093

Scalable Enantioselective Total Synthesis of (−)‐Goniomitine

Huai‐Yu Bin, Ke Wang, Dan Yang, Xiao‐Hui Yang, Jian‐Hua Xie and Qi‐Lin Zhou

Angewandte Chemie, 2019, 131, 1186
DOI: 10.1002/ange.201812822

Identification of novel small molecule inhibitors for endoplasmic reticulum oxidoreductase 1α (ERO1α) enzyme: structure-based molecular docking and molecular dynamic simulation studies

Hussam Albassam, Chetan H. Mehta and Usha Y. Nayak

Journal of Biomolecular Structure and Dynamics, 2022, 40, 13218
DOI: 10.1080/07391102.2021.1984308

Axinellamines as Broad-Spectrum Antibacterial Agents: Scalable Synthesis and Biology

Rodrigo A. Rodriguez, Danielle Barrios Steed, Yu Kawamata, Shun Su, Peter A. Smith, Tyler C. Steed, Floyd E. Romesberg and Phil S. Baran

J. Am. Chem. Soc., 2014, 136, 15403
DOI: 10.1021/ja508632y

Synthetic Organic Electrochemistry: An Enabling and Innately Sustainable Method

Evan J. Horn, Brandon R. Rosen and Phil S. Baran

ACS Cent. Sci., 2016, 2, 302
DOI: 10.1021/acscentsci.6b00091

Biosynthese im Reagenzglas

Tanja Gulder and Tobias A. M. Gulder

Nachr Chem, 2014, 62, 1081
DOI: 10.1002/nadc.201490379

Empowering Synthesis of Complex Natural Products

Lucas W. Hernandez and David Sarlah

Chemistry A European J, 2019, 25, 13248
DOI: 10.1002/chem.201901808

Gram-Scale Synthesis of Bufospirostenin A by a Biomimetic Skeletal Rearrangement Approach

Yu Wang, Hailong Tian and Jinghan Gui

J. Am. Chem. Soc., 2021, 143, 19576
DOI: 10.1021/jacs.1c10067

Biologically Significant and Recently Isolated Alkaloids from Endophytic Fungi

Sharna-kay Daley and Geoffrey A. Cordell

J. Nat. Prod., 2021, 84, 871
DOI: 10.1021/acs.jnatprod.0c01195

Synthesis of natural products and their derivatives using dynamic crystallization

Takaaki Sato

Chemistry Letters, 2025, 54
DOI: 10.1093/chemle/upae244

Optically Active Flavaglines-Inspired Molecules by a Palladium-Catalyzed Decarboxylative Dearomative Asymmetric Allylic Alkylation

Meng-Yue Cao, Bin-Jie Ma, Zhi-Qi Lao, Hongliang Wang, Jing Wang, Juan Liu, Kuan Xing, Yu-Hao Huang, Kang-Ji Gan, Wei Gao, Huaimin Wang, Xin Hong and Hai-Hua Lu

J. Am. Chem. Soc., 2020, 142, 12039
DOI: 10.1021/jacs.0c05113

Treating a Global Health Crisis with a Dose of Synthetic Chemistry

Melissa A. Hardy, Brandon A. Wright, J. Logan Bachman, Timothy B. Boit, Hannah M. S. Haley, Rachel R. Knapp, Robert F. Lusi, Taku Okada, Veronica Tona, Neil K. Garg and Richmond Sarpong

ACS Cent. Sci., 2020, 6, 1017
DOI: 10.1021/acscentsci.0c00637

Synthesis and biological evaluation of novel steroidal pyrazole amides as highly potent anticancer agents

Haibo Huo, Weiqi Jiang, Feifei Sun, Jian Li and Baojun Shi

Steroids, 2021, 176, 108931
DOI: 10.1016/j.steroids.2021.108931

Natural Product Synthesis at the Interface of Chemistry and Biology

Jiyong Hong

Chemistry A European J, 2014, 20, 10204
DOI: 10.1002/chem.201402804

Flow chemistry in the multi-step synthesis of natural products

Li Wan, Gaopan Kong, Minjie Liu, Meifen Jiang, Dang Cheng and Fener Chen

Green Synthesis and Catalysis, 2022, 3, 243
DOI: 10.1016/j.gresc.2022.07.007

Madangamine alkaloids: Madness and tranquility

Ye Tang, Lili Zhu and Ran Hong

Tetrahedron Chem, 2022, 3, 100025
DOI: 10.1016/j.tchem.2022.100025

Computer-Aided Analysis of Multiple SARS-CoV-2 Therapeutic Targets: Identification of Potent Molecules from African Medicinal Plants

Franklyn Nonso Iheagwam and Solomon Oladapo Rotimi

Scientifica, 2020, 2020, 1
DOI: 10.1155/2020/1878410

Mild Friedel–Crafts Reactions Enable a Robust Synthesis of Roseophilin

Xiao Zhang, Cuifang Zhang, Xiaobin Wang and Guangxin Liang

Org. Lett., 2019, 21, 3357
DOI: 10.1021/acs.orglett.9b01100

Molecular complexity as a driving force for the advancement of organic synthesis

Brandon A. Wright and Richmond Sarpong

Nat Rev Chem, 2024, 8, 776
DOI: 10.1038/s41570-024-00645-8

A 11‐Steps Total Synthesis of Magellanine through a Gold(I)‐Catalyzed Dehydro Diels–Alder Reaction

Philippe McGee, Geneviève Bétournay, Francis Barabé and Louis Barriault

Angewandte Chemie, 2017, 129, 6377
DOI: 10.1002/ange.201611606

Total Synthesis and Structural Plasticity of Kratom Pseudoindoxyl Metabolites**

Péter Angyal, Kristóf Hegedüs, Bence Balázs Mészáros, János Daru, Ádám Dudás, Anna Rita Galambos, Nariman Essmat, Mahmoud Al‐Khrasani, Szilárd Varga and Tibor Soós

Angew Chem Int Ed, 2023, 62
DOI: 10.1002/anie.202303700

Natural Product Synthesis: The Endless Quest for Unreachable Perfection

Nicolas Fay, Cyrille Kouklovsky and Aurélien de la Torre

ACS Org. Inorg. Au, 2023, 3, 350
DOI: 10.1021/acsorginorgau.3c00040

Some Thoughts on Barry M. Trost and Natural Products

Georges Massiot

Israel Journal of Chemistry, 2021, 61, 289
DOI: 10.1002/ijch.202000058

Natural Product Total Synthesis: As Exciting as Ever and Here To Stay

Phil S. Baran

J. Am. Chem. Soc., 2018, 140, 4751
DOI: 10.1021/jacs.8b02266

A semi-synthetic heparan sulfate material that potentiates BMP2-mediated osteogenesis

Liam J. Sargison, Amira Sargison, Susan M. Carnachan, Raymond A.A. Smith, Alison M. Daines, Simon F.R. Hinkley and Simon M. Cool

International Journal of Biological Macromolecules, 2025, 314, 144349
DOI: 10.1016/j.ijbiomac.2025.144349

Total Synthesis of Brazilin

Youngeun Jung and Ikyon Kim

J. Org. Chem., 2015, 80, 2001
DOI: 10.1021/jo502745j

Discovery and resupply of pharmacologically active plant-derived natural products: A review

Atanas G. Atanasov, Birgit Waltenberger, Eva-Maria Pferschy-Wenzig, Thomas Linder, Christoph Wawrosch, Pavel Uhrin, Veronika Temml, Limei Wang, Stefan Schwaiger, Elke H. Heiss, Judith M. Rollinger, Daniela Schuster, Johannes M. Breuss, Valery Bochkov, Marko D. Mihovilovic, Brigitte Kopp, Rudolf Bauer, Verena M. Dirsch and Hermann Stuppner

Biotechnology Advances, 2015, 33, 1582
DOI: 10.1016/j.biotechadv.2015.08.001

Ideality in Context: Motivations for Total Synthesis

David S. Peters, Cody Ross Pitts, Kyle S. McClymont, Thomas P. Stratton, Cheng Bi and Phil S. Baran

Acc. Chem. Res., 2021, 54, 605
DOI: 10.1021/acs.accounts.0c00821

Total Synthesis of the Euphorbia Diterpenoid Pepluacetal

Meng Liu, Chuanhua Wu, Xingang Xie, Huilin Li and Xuegong She

Angewandte Chemie, 2024, 136
DOI: 10.1002/ange.202400943

Electrochemical organic reactions: A tutorial review

Joyeeta Lodh, Shounik Paul, He Sun, Luyang Song, Wolfgang Schöfberger and Soumyajit Roy

Front. Chem., 2023, 10
DOI: 10.3389/fchem.2022.956502

Gram‐Scale Enantioselective Formal Synthesis of Morphine through an ortho–para Oxidative Phenolic Coupling Strategy

Matthieu Tissot, Robert J. Phipps, Catherine Lucas, Rafael M. Leon, Robert D. M. Pace, Tifelle Ngouansavanh and Matthew J. Gaunt

Angew Chem Int Ed, 2014, 53, 13498
DOI: 10.1002/anie.201408435

Natural product anticipation through synthesis

Belinda E. Hetzler, Dirk Trauner and Andrew L. Lawrence

Nat Rev Chem, 2022, 6, 170
DOI: 10.1038/s41570-021-00345-7

Concise Large-Scale Synthesis of Tomatidine, A Potent Antibiotic Natural Product

Chad Normandin and Pierre-Luc Boudreault

Molecules, 2021, 26, 6008
DOI: 10.3390/molecules26196008

Studies Targeting Ryanodol Result in an Annulation Reaction for the Synthesis of a Variety of Fused Carbocycles

Rajdip Karmakar, Arnold L. Rheingold and Glenn C. Micalizio

Org. Lett., 2019, 21, 6126
DOI: 10.1021/acs.orglett.9b02278

Spirotetronate Polyketides as Leads in Drug Discovery

Michelle H. Lacoske and Emmanuel A. Theodorakis

J. Nat. Prod., 2015, 78, 562
DOI: 10.1021/np500757w

Short Scalable Route to Apiaceae Sesquiterpene Scaffolds: Total Synthesis of 4-epi-Epiguaidiol A

Maria Kourgiantaki, Vera P. Demertzidou and Alexandros L. Zografos

Org. Lett., 2022, 24, 8476
DOI: 10.1021/acs.orglett.2c03215

Total Syntheses of (−)‐Minovincine and (−)‐Aspidofractinine through a Sequence of Cascade Reactions

Szilárd Varga, Péter Angyal, Gábor Martin, Orsolya Egyed, Tamás Holczbauer and Tibor Soós

Angewandte Chemie, 2020, 132, 13649
DOI: 10.1002/ange.202004769

Bioinspired Total Synthesis of Gymnothelignan N

Huilin Li, Yuanyuan Zhang, Xingang Xie, Haichen Ma, Changgui Zhao, Gaoyuan Zhao and Xuegong She

Org. Lett., 2014, 16, 4440
DOI: 10.1021/ol501960j

trans‐Hydrogenation: Application to a Concise and Scalable Synthesis of Brefeldin A

Michael Fuchs and Alois Fürstner

Angewandte Chemie, 2015, 127, 4050
DOI: 10.1002/ange.201411618

An Enantioconvergent and Concise Synthesis of Lasonolide A

Lin Yang, Zuming Lin, Shunjie Shao, Qian Zhao and Ran Hong

Angew Chem Int Ed, 2018, 57, 16200
DOI: 10.1002/anie.201811093

Facile and scalable synthesis of baphicacanthin A by a two-pot procedure

Yalong Cuan, Wenhao Li, Yingchao Dou and Guanyu Yang

Natural Product Research, 2023, 37, 1439
DOI: 10.1080/14786419.2021.2011275

Total Synthesis of (+)-Alstonlarsine A: Old Reactions in Modern Alkaloids Synthesis

Zorana B. Ferjancic and Filip J. Bihelovic

Synlett, 2023, 34, 203
DOI: 10.1055/a-1968-2233

Opportunities for enzyme catalysis in natural product chemistry

Steffen Friedrich and Frank Hahn

Tetrahedron, 2015, 71, 1473
DOI: 10.1016/j.tet.2014.12.026

trans‐Hydrogenation: Application to a Concise and Scalable Synthesis of Brefeldin A

Michael Fuchs and Alois Fürstner

Angew Chem Int Ed, 2015, 54, 3978
DOI: 10.1002/anie.201411618

Concise Total Synthesis of Dehaloperophoramidine

Kirill Popov, Anita Hoang and Peter Somfai

Angewandte Chemie, 2016, 128, 1833
DOI: 10.1002/ange.201510661

Fawcettimine‐Type Lycopodium Alkaloids as a Driving Force for Discoveries in Organic Synthesis

Houhua Li and Xiaoguang Lei

The Chemical Record, 2018, 18, 543
DOI: 10.1002/tcr.201700047

Total Synthesis and Structural Plasticity of Kratom Pseudoindoxyl Metabolites**

Péter Angyal, Kristóf Hegedüs, Bence Balázs Mészáros, János Daru, Ádám Dudás, Anna Rita Galambos, Nariman Essmat, Mahmoud Al‐Khrasani, Szilárd Varga and Tibor Soós

Angewandte Chemie, 2023, 135
DOI: 10.1002/ange.202303700