Issue 6, 2025

Dearomative 2,3-diamination of indoles triggered by Rh(iii)-catalyzed Csp2–H activation

Abstract

An Rh(III)-catalyzed dearomative 2,3-diamination of indoles with N-alkoxyamides has been developed. The method provides an efficient approach to access 2-(N-acylimino)-3-aminoindolines with high regioselectivity.

Graphical abstract: Dearomative 2,3-diamination of indoles triggered by Rh(iii)-catalyzed Csp2–H activation

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Article information

Article type
Research Article
Submitted
27 Oct 2024
Accepted
04 Jan 2025
First published
08 Jan 2025

Org. Chem. Front., 2025,12, 1821-1826

Dearomative 2,3-diamination of indoles triggered by Rh(III)-catalyzed Csp2–H activation

C. Wang, H. Jiang and W. Zeng, Org. Chem. Front., 2025, 12, 1821 DOI: 10.1039/D4QO02017K

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