Jump to main content
Jump to site search
Access to RSC content Close the message box

Continue to access RSC content when you are not at your institution. Follow our step-by-step guide.


Issue 7, 2020
Previous Article Next Article

Concise synthesis of α-amino cyclic boronates via multicomponent coupling of salicylaldehydes, amines, and B2(OH)4

Author affiliations

Abstract

We report here a concise synthesis of α-amino cyclic boronates via multicomponent coupling of readily available salicylaldehydes, amines, and B2(OH)4. The process can be carried out at room temperature in ethanol, does not require catalysts or additives, and is easy to scale up. Aminals and ligated boroxines are intermediates in this reaction.

Graphical abstract: Concise synthesis of α-amino cyclic boronates via multicomponent coupling of salicylaldehydes, amines, and B2(OH)4

Back to tab navigation

Supplementary files

Article information


Submitted
28 Jan 2020
Accepted
05 Mar 2020
First published
05 Mar 2020

Green Chem., 2020,22, 2184-2190
Article type
Communication

Concise synthesis of α-amino cyclic boronates via multicomponent coupling of salicylaldehydes, amines, and B2(OH)4

W. Ming, X. Liu, A. Friedrich, J. Krebs, Y. P. Budiman, M. Huang and T. B. Marder, Green Chem., 2020, 22, 2184
DOI: 10.1039/D0GC00346H

Social activity

Search articles by author

Spotlight

Advertisements