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Facile one-pot synthesis of 2-aminoindoles from simple anilines and ynamides

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Abstract

A highly effective and straightforward one-pot synthesis of diversely substituted 2-aminoindoles has been developed, involving sequential Au(I)-catalyzed regioselective hydroamination and CuCl2-mediated oxidative cyclization. This protocol offers an operationally easy, simple, robust, and sustainable approach with the use of readily available starting materials, good functional group tolerance, and high practicality and efficiency.

Graphical abstract: Facile one-pot synthesis of 2-aminoindoles from simple anilines and ynamides

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Article information


Submitted
28 Sep 2020
Accepted
11 Oct 2020
First published
12 Oct 2020

Chem. Commun., 2020, Advance Article
Article type
Communication

Facile one-pot synthesis of 2-aminoindoles from simple anilines and ynamides

Y. H. Kim, H. J. Yoo and S. W. Youn, Chem. Commun., 2020, Advance Article , DOI: 10.1039/D0CC06490D

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