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Copper-catalyzed tandem cis-carbometallation/cyclization of imine-ynamides with arylboronic acids

Abstract

An efficient copper-catalyzed tandem regioselective cis-carbometallation/cyclization of imine-ynamides with arylboronic acids has been developed. This method leads to facile and practical synthesis of valuable 2,3-disubstituted indolines in moderate to excellent yields and features a broad substrate scope and wide functional group tolerance. Other significant features of this protocol include the use of readily available starting materials, high flexibility, simple procedure and mild reaction conditions.

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Article information


Submitted
24 Feb 2020
Accepted
23 Mar 2020
First published
24 Mar 2020

Chem. Commun., 2020, Accepted Manuscript
Article type
Communication

Copper-catalyzed tandem cis-carbometallation/cyclization of imine-ynamides with arylboronic acids

H. Wang, E. Huang, C. Luo, W. Luo, Y. Xu, P. Qian, J. Zhou and L. Ye, Chem. Commun., 2020, Accepted Manuscript , DOI: 10.1039/D0CC01424A

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