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Issue 24, 2019
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Recent advances in the direct functionalization of quinoxalin-2(1H)-ones

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Abstract

The direct C3-functionalization of quinoxalin-2(1H)-ones via C–H bond activation has recently attracted considerable attention, due to their diverse biological activities and chemical properties. This review will focus on the recent achievements, mainly including arylation, alkylation, acylation, alkoxycarbonylation, amination, amidation and phosphonation of quinoxalin-2(1H)-ones. Their mechanisms are also discussed.

Graphical abstract: Recent advances in the direct functionalization of quinoxalin-2(1H)-ones

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Publication details

The article was received on 04 Apr 2019, accepted on 18 May 2019 and first published on 23 May 2019


Article type: Review Article
DOI: 10.1039/C9OB00782B
Org. Biomol. Chem., 2019,17, 5863-5881

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    Recent advances in the direct functionalization of quinoxalin-2(1H)-ones

    Q. Ke, G. Yan, J. Yu and X. Wu, Org. Biomol. Chem., 2019, 17, 5863
    DOI: 10.1039/C9OB00782B

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