Jump to main content
Jump to site search


Benzoazacrown compound: a highly effective chelator for therapeutic bismuth radioisotopes

Author affiliations

Abstract

A new benzoazacrown ligand H4BATA was synthesized and its complexation ability towards bismuth cations was evaluated. Binding of cation occurs at room temperature in a few minutes and formed complex exhibits the same level of inertness as highly stable complex with the well-known H4DOTA in biologically relevant and challenging media under in vivo conditions.

Graphical abstract: Benzoazacrown compound: a highly effective chelator for therapeutic bismuth radioisotopes

Back to tab navigation

Supplementary files

Publication details

The article was received on 29 Apr 2019, accepted on 03 Jul 2019 and first published on 04 Jul 2019


Article type: Research Article
DOI: 10.1039/C9MD00251K
Med. Chem. Commun., 2019, Advance Article

  •   Request permissions

    Benzoazacrown compound: a highly effective chelator for therapeutic bismuth radioisotopes

    E. V. Matazova, B. V. Egorova, E. A. Konopkina, G. Yu. Aleshin, A. D. Zubenko, A. A. Mitrofanov, K. V. Karpov, O. A. Fedorova, Y. V. Fedorov and S. N. Kalmykov, Med. Chem. Commun., 2019, Advance Article , DOI: 10.1039/C9MD00251K

Search articles by author

Spotlight

Advertisements