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Issue 15, 2019
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Gold(I) catalysed regio- and stereoselective intermolecular hydroamination of internal alkynes: towards functionalised azoles

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Abstract

Gold(I) catalysed regio- and stereoselective intermolecular hydroamination of internal alkynes was developed for the effective synthesis of a series of (Z)-functionalised vinylazoles under solvent free conditions. The catalytic hydrogenation of the resulting enamines leads to substituted saturated azoles in good yields.

Graphical abstract: Gold(i) catalysed regio- and stereoselective intermolecular hydroamination of internal alkynes: towards functionalised azoles

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Publication details

The article was received on 12 Mar 2019, accepted on 20 Mar 2019 and first published on 20 Mar 2019


Article type: Paper
DOI: 10.1039/C9OB00587K
Org. Biomol. Chem., 2019,17, 3805-3811

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    Gold(I) catalysed regio- and stereoselective intermolecular hydroamination of internal alkynes: towards functionalised azoles

    C. Michon, J. Gilbert, X. Trivelli, F. Nahra, C. S. J. Cazin, F. Agbossou-Niedercorn and S. P. Nolan, Org. Biomol. Chem., 2019, 17, 3805
    DOI: 10.1039/C9OB00587K

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