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Issue 28, 2019
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Synthesis of indoles and quinazolines via additive-controlled selective C–H activation/annulation of N-arylamidines and sulfoxonium ylides

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Abstract

Selective synthesis of indole and quinazoline products was achieved through a precise control of the C–H activation/annulation by changing the additives from NaOAc to CuF2/CsOAc. This strategy constructs indole and quinazoline scaffolds efficiently, and hence is of great interest in pharmaceutical, agricultural and chemical industries.

Graphical abstract: Synthesis of indoles and quinazolines via additive-controlled selective C–H activation/annulation of N-arylamidines and sulfoxonium ylides

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Publication details

The article was received on 08 Feb 2019, accepted on 06 Mar 2019 and first published on 06 Mar 2019


Article type: Communication
DOI: 10.1039/C9CC01146C
Chem. Commun., 2019,55, 4039-4042

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    Synthesis of indoles and quinazolines via additive-controlled selective C–H activation/annulation of N-arylamidines and sulfoxonium ylides

    R. Lai, X. Wu, S. Lv, C. Zhang, M. He, Y. Chen, Q. Wang, L. Hai and Y. Wu, Chem. Commun., 2019, 55, 4039
    DOI: 10.1039/C9CC01146C

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