Ting Li, Lei Yang, Kaidong Ni, Zhenyu Shi, Fei Li and Dongyin Chen
Org. Biomol. Chem., 2016,14, 6297-6303
DOI:
10.1039/C6OB00819D,
Paper
An efficient copper-catalyzed reaction for the synthesis of benzisothiazol-3(2H)-ones has been developed, starting from easily available 2-halobenzamides and carbon disulfide, which gave the corresponding target products in 30–89% yield for 25 examples. The reaction proceeds via a consecutive process with S–C bond and S–N bond formation.
