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Issue 19, 2016

Copper-catalyzed borylative coupling of vinylazaarenes and N-Boc imines

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Abstract

Cu-catalyzed three-component couplings of vinylazaarenes, B2(pin)2, and N-Boc imines are described. Oxidation of the initially formed boronate gives azaarene-containing, Boc-protected amino alcohols with reasonable to good diastereoselectivities.

Graphical abstract: Copper-catalyzed borylative coupling of vinylazaarenes and N-Boc imines

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Article information


Submitted
21 Jan 2016
Accepted
09 Feb 2016
First published
17 Feb 2016

This article is Open Access

Chem. Commun., 2016,52, 3770-3772
Article type
Communication

Copper-catalyzed borylative coupling of vinylazaarenes and N-Boc imines

J. J. Smith, D. Best and H. W. Lam, Chem. Commun., 2016, 52, 3770 DOI: 10.1039/C6CC00603E

This article is licensed under a Creative Commons Attribution 3.0 Unported Licence. You can use material from this article in other publications without requesting further permissions from the RSC, provided that the correct acknowledgement is given.

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