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Issue 5, 2015
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Copper-catalyzed O-arylation of N-protected 1,2-aminoalcohols using functionalized trivalent organobismuth reagents

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Abstract

The O-arylation of 1,2-aminoalcohols using functionalized triarylbismuth reagents is reported. The reaction can be performed using substoichiometric amounts of copper acetate and operates under mild conditions. Good functional group tolerance is observed, giving access to a range of β-aryloxyamines. The effect provided by the amino group in the arylation reaction is investigated.

Graphical abstract: Copper-catalyzed O-arylation of N-protected 1,2-aminoalcohols using functionalized trivalent organobismuth reagents

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Publication details

The article was received on 29 Sep 2014, accepted on 28 Nov 2014 and first published on 09 Dec 2014


Article type: Communication
DOI: 10.1039/C4OB02497D
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Citation: Org. Biomol. Chem., 2015,13, 1322-1327
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    Copper-catalyzed O-arylation of N-protected 1,2-aminoalcohols using functionalized trivalent organobismuth reagents

    P. Petiot, J. Dansereau, M. Hébert, I. Khene, T. Ahmad, S. Samaali, M. Leroy, F. Pinsonneault, C. Y. Legault and A. Gagnon, Org. Biomol. Chem., 2015, 13, 1322
    DOI: 10.1039/C4OB02497D

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